NO325709B1 - Anvendelse av (+)-1-(3,4-diklorfenyl)-3-azabicyklo[3.1.0]heksan for fremstilling av medikamenter - Google Patents
Anvendelse av (+)-1-(3,4-diklorfenyl)-3-azabicyklo[3.1.0]heksan for fremstilling av medikamenter Download PDFInfo
- Publication number
- NO325709B1 NO325709B1 NO20033165A NO20033165A NO325709B1 NO 325709 B1 NO325709 B1 NO 325709B1 NO 20033165 A NO20033165 A NO 20033165A NO 20033165 A NO20033165 A NO 20033165A NO 325709 B1 NO325709 B1 NO 325709B1
- Authority
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- Norway
- Prior art keywords
- depression
- azabicyclo
- dichlorophenyl
- hexane
- disorder
- Prior art date
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Classifications
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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PCT/US2002/000845 WO2002066427A2 (en) | 2001-01-11 | 2002-01-11 | (+)-1-(3,4-dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions and uses thereof |
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EP (1) | EP1349835B1 (hu) |
JP (4) | JP2005500983A (hu) |
KR (1) | KR20030081384A (hu) |
CN (2) | CN1496349A (hu) |
AU (1) | AU2002251758B2 (hu) |
BR (1) | BR0206434A (hu) |
CA (1) | CA2434616C (hu) |
CZ (1) | CZ306143B6 (hu) |
HU (1) | HUP0302613A3 (hu) |
IL (2) | IL156889A0 (hu) |
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NZ (1) | NZ527101A (hu) |
PL (1) | PL364837A1 (hu) |
RU (1) | RU2294926C2 (hu) |
SK (1) | SK10122003A3 (hu) |
WO (1) | WO2002066427A2 (hu) |
ZA (1) | ZA200305440B (hu) |
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US6372919B1 (en) * | 2001-01-11 | 2002-04-16 | Dov Pharmaceutical, Inc. | (+)-1-(3,4-dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions thereof, and uses as an anti-depressant agent |
US20060173064A1 (en) * | 2001-08-24 | 2006-08-03 | Lippa Arnold S | (-)-1-(3,4-Dichlorophenyl)-3-azabi cyclo[3.1.0]hexane, compositions thereof, and uses for treating alcohol-related disorders |
US6569887B2 (en) * | 2001-08-24 | 2003-05-27 | Dov Pharmaceuticals Inc. | (−)-1-(3,4-Dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions thereof, and uses as a dopamine-reuptake |
US20070225351A1 (en) * | 2002-01-11 | 2007-09-27 | Lippa Arnold S | Methods and compositions for controlling body weight and appetite |
US20080081834A1 (en) | 2002-07-31 | 2008-04-03 | Lippa Arnold S | Methods and compositions employing bicifadine for treating disability or functional impairment associated with acute pain, chronic pain, or neuropathic disorders |
NZ527142A (en) * | 2003-07-23 | 2006-03-31 | Douglas Pharmaceuticals Ltd | A stable suspension formulation |
CZ2006427A3 (cs) * | 2003-12-29 | 2006-11-15 | Sepracor Inc. | Pyrrolové a pyrazolové inhibitory DAAO |
JP2008507550A (ja) * | 2004-07-22 | 2008-03-13 | ワイス | 神経系障害及び状態の処置方法 |
AU2005266996A1 (en) * | 2004-07-22 | 2006-02-02 | Wyeth | Method for treating nervous system disorders and conditions |
CN101022794A (zh) * | 2004-07-22 | 2007-08-22 | 惠氏公司 | 治疗神经系统障碍和病症的方法 |
KR20130108489A (ko) * | 2004-08-18 | 2013-10-02 | 도브 파마슈티칼 인코포레이티드 | 아자비사이클로헥산의 신규한 다형체 |
AU2012203400B2 (en) * | 2004-08-18 | 2015-01-15 | Euthymics Bioscience, Inc. | Novel polymorphs of azabicyclohexane |
US20070043100A1 (en) | 2005-08-16 | 2007-02-22 | Hagen Eric J | Novel polymorphs of azabicyclohexane |
US20060100263A1 (en) * | 2004-11-05 | 2006-05-11 | Anthony Basile | Antipyretic compositions and methods |
AU2006214443C1 (en) * | 2005-02-15 | 2011-11-24 | Alkermes Pharma Ireland Limited | Aerosol and injectable formulations of nanoparticulate benzodiazepine |
JP2009500425A (ja) | 2005-07-06 | 2009-01-08 | セプラコア インコーポレーテッド | エスゾピクロン及びトランス4−(3,4−ジクロロフェニル)−1,2,3,4−テトラヒドロ−n−メチル−1−ナフタレンアミン又はトランス4−(3,4−ジクロロフェニル)−1,2,3,4−テトラヒドロ−1−ナフタレンアミンの組み合わせ、並びに閉経期並びに気分、不安、及び認知障害の治療方法 |
US20070021488A1 (en) * | 2005-07-21 | 2007-01-25 | Wyeth | Method for treating nervous system disorders and conditions |
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