NO325089B1 - Isoksazoler og deres anvendelse som inhibitorer av ERK - Google Patents

Isoksazoler og deres anvendelse som inhibitorer av ERK Download PDF

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Publication number
NO325089B1
NO325089B1 NO20031192A NO20031192A NO325089B1 NO 325089 B1 NO325089 B1 NO 325089B1 NO 20031192 A NO20031192 A NO 20031192A NO 20031192 A NO20031192 A NO 20031192A NO 325089 B1 NO325089 B1 NO 325089B1
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Prior art keywords
disease
optionally substituted
compound
hydrogen
group
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NO20031192A
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English (en)
Norwegian (no)
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NO20031192D0 (no
NO20031192L (no
Inventor
Jingrong Cao
Michael Hale
Francois Maltais
Robert Mashal
James Janetka
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Vertex Pharma
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Publication of NO20031192D0 publication Critical patent/NO20031192D0/no
Publication of NO20031192L publication Critical patent/NO20031192L/no
Publication of NO325089B1 publication Critical patent/NO325089B1/no

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
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  • Neurosurgery (AREA)
  • Diabetes (AREA)
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NO20031192A 2000-09-15 2003-03-14 Isoksazoler og deres anvendelse som inhibitorer av ERK NO325089B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23295600P 2000-09-15 2000-09-15
PCT/US2001/028790 WO2002022610A1 (fr) 2000-09-15 2001-09-14 Soxazoles et leur utilisation comme inhibiteur d'erk

Publications (3)

Publication Number Publication Date
NO20031192D0 NO20031192D0 (no) 2003-03-14
NO20031192L NO20031192L (no) 2003-05-13
NO325089B1 true NO325089B1 (no) 2008-01-28

Family

ID=22875248

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20031192A NO325089B1 (no) 2000-09-15 2003-03-14 Isoksazoler og deres anvendelse som inhibitorer av ERK

Country Status (16)

Country Link
US (3) US6495582B1 (fr)
EP (1) EP1317453B1 (fr)
JP (1) JP4052573B2 (fr)
AT (1) ATE335737T1 (fr)
AU (1) AU2001290940A1 (fr)
CA (1) CA2422376A1 (fr)
DE (1) DE60122176T2 (fr)
ES (1) ES2269458T3 (fr)
HK (1) HK1052934B (fr)
HU (1) HUP0302991A3 (fr)
IL (1) IL154710A0 (fr)
MX (1) MXPA03002296A (fr)
NO (1) NO325089B1 (fr)
NZ (1) NZ525016A (fr)
WO (1) WO2002022610A1 (fr)
ZA (1) ZA200301696B (fr)

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NO20031192D0 (no) 2003-03-14
HK1052934A1 (en) 2003-10-03
WO2002022610A1 (fr) 2002-03-21
NO20031192L (no) 2003-05-13
HUP0302991A2 (hu) 2003-12-29
US6495582B1 (en) 2002-12-17
EP1317453B1 (fr) 2006-08-09
US6649640B2 (en) 2003-11-18
JP2004509119A (ja) 2004-03-25
ATE335737T1 (de) 2006-09-15
MXPA03002296A (es) 2003-06-06
US20020177618A1 (en) 2002-11-28
US20030195241A1 (en) 2003-10-16
ES2269458T3 (es) 2007-04-01
HUP0302991A3 (en) 2009-10-28
CA2422376A1 (fr) 2002-03-21
ZA200301696B (en) 2004-04-28
HK1052934B (zh) 2007-01-12
DE60122176T2 (de) 2007-07-05
AU2001290940A1 (en) 2002-03-26
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US7354919B2 (en) 2008-04-08
US20050090536A1 (en) 2005-04-28

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