NO324873B1 - 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom - Google Patents

3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom Download PDF

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Publication number
NO324873B1
NO324873B1 NO20025106A NO20025106A NO324873B1 NO 324873 B1 NO324873 B1 NO 324873B1 NO 20025106 A NO20025106 A NO 20025106A NO 20025106 A NO20025106 A NO 20025106A NO 324873 B1 NO324873 B1 NO 324873B1
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compound
compound according
mmol
substituted
solution
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NO20025106A
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English (en)
Norwegian (no)
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NO20025106L (no
NO20025106D0 (no
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Jeffery R Raymond
Claudia E Kasserra
Yaning Shen
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Inflazyme Pharm Ltd
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Publication of NO20025106D0 publication Critical patent/NO20025106D0/no
Publication of NO20025106L publication Critical patent/NO20025106L/no
Publication of NO324873B1 publication Critical patent/NO324873B1/no

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0011Unsubstituted amino radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036Nitrogen-containing hetero ring
    • C07J71/0042Nitrogen only
    • C07J71/0047Nitrogen only at position 2(3)
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036Nitrogen-containing hetero ring
    • C07J71/0057Nitrogen and oxygen
    • C07J71/0063Nitrogen and oxygen at position 2(3)
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Vascular Medicine (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20025106A 2000-04-28 2002-10-24 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom NO324873B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20061700P 2000-04-28 2000-04-28
PCT/CA2001/000581 WO2001083512A1 (en) 2000-04-28 2001-04-30 3-nitrogen-6,7-dioxygen steroids and uses related thereto

Publications (3)

Publication Number Publication Date
NO20025106D0 NO20025106D0 (no) 2002-10-24
NO20025106L NO20025106L (no) 2002-12-18
NO324873B1 true NO324873B1 (no) 2007-12-17

Family

ID=22742458

Family Applications (1)

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NO20025106A NO324873B1 (no) 2000-04-28 2002-10-24 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom

Country Status (34)

Country Link
US (4) US20040034216A1 (et)
EP (1) EP1278763B1 (et)
JP (1) JP2003531916A (et)
KR (1) KR20030045671A (et)
CN (1) CN1214039C (et)
AP (1) AP1825A (et)
AT (1) ATE353909T1 (et)
AU (2) AU2001252084B2 (et)
BG (1) BG107289A (et)
BR (1) BR0110419A (et)
CA (1) CA2418748A1 (et)
CO (1) CO5590904A2 (et)
DE (1) DE60126597T2 (et)
DK (1) DK1278763T3 (et)
DZ (1) DZ3355A1 (et)
EE (1) EE200200613A (et)
ES (1) ES2282247T3 (et)
HK (1) HK1050694A1 (et)
HR (1) HRP20020944A2 (et)
HU (1) HUP0300908A2 (et)
IL (2) IL152448A0 (et)
MA (1) MA25808A1 (et)
MX (1) MXPA02010645A (et)
NO (1) NO324873B1 (et)
NZ (1) NZ522181A (et)
OA (1) OA12255A (et)
PL (1) PL365798A1 (et)
PT (1) PT1278763E (et)
RU (1) RU2291873C2 (et)
SK (1) SK15692002A3 (et)
UA (1) UA79229C2 (et)
WO (1) WO2001083512A1 (et)
YU (1) YU88102A (et)
ZA (1) ZA200208631B (et)

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KR20070007766A (ko) * 2003-10-20 2007-01-16 인플라자임 파마슈티칼즈 리미티드 3-베타-아미노 17-메틸렌 안드로스테인-6-알파 7-베타-디올하이드로클로라이드의 결정질 형태
FR2861077B1 (fr) * 2003-10-20 2006-03-03 Aventis Pharma Sa Formes cristallines du chlorydrate de 3-beta-amino, 17-methylene, androstane-6-alpha, 7-beta-diol
US20050227927A1 (en) * 2004-03-31 2005-10-13 Robinson Cynthia B Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a glucocorticosteroid for treatment of asthma, chronic obstructive pulmonary disease or allergic rhinitis
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ES2282247T3 (es) 2007-10-16
US7112580B2 (en) 2006-09-26
CN1430625A (zh) 2003-07-16
BR0110419A (pt) 2004-02-25
ATE353909T1 (de) 2007-03-15
PL365798A1 (en) 2005-01-10
AP1825A (en) 2008-02-03
HK1050694A1 (en) 2003-07-04
AU2001252084B2 (en) 2006-07-06
AU5208401A (en) 2001-11-12
HRP20020944A2 (en) 2004-02-29
US20050215534A9 (en) 2005-09-29
JP2003531916A (ja) 2003-10-28
RU2291873C2 (ru) 2007-01-20
KR20030045671A (ko) 2003-06-11
PT1278763E (pt) 2007-05-31
DE60126597D1 (de) 2007-03-29
NO20025106L (no) 2002-12-18
BG107289A (bg) 2003-07-31
DZ3355A1 (fr) 2001-11-08
EP1278763A1 (en) 2003-01-29
US20070060553A1 (en) 2007-03-15
US6635629B2 (en) 2003-10-21
DE60126597T2 (de) 2007-10-31
EP1278763B1 (en) 2007-02-14
US20040138186A1 (en) 2004-07-15
ZA200208631B (en) 2004-02-23
AP2002002659A0 (en) 2002-12-31
OA12255A (en) 2006-05-11
WO2001083512A1 (en) 2001-11-08
US20020072510A1 (en) 2002-06-13
SK15692002A3 (sk) 2003-11-04
CA2418748A1 (en) 2001-11-08
NZ522181A (en) 2005-04-29
DK1278763T3 (da) 2007-06-11
HUP0300908A2 (hu) 2003-07-28
NO20025106D0 (no) 2002-10-24
CO5590904A2 (es) 2005-12-30
EE200200613A (et) 2004-04-15
IL152448A0 (en) 2003-05-29
US20040034216A1 (en) 2004-02-19
MA25808A1 (fr) 2003-07-01
IL152448A (en) 2006-12-31
MXPA02010645A (es) 2004-04-20
UA79229C2 (en) 2007-06-11
YU88102A (sh) 2006-01-16
CN1214039C (zh) 2005-08-10

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