NO317978B1 - Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav - Google Patents

Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav Download PDF

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Publication number
NO317978B1
NO317978B1 NO20003254A NO20003254A NO317978B1 NO 317978 B1 NO317978 B1 NO 317978B1 NO 20003254 A NO20003254 A NO 20003254A NO 20003254 A NO20003254 A NO 20003254A NO 317978 B1 NO317978 B1 NO 317978B1
Authority
NO
Norway
Prior art keywords
arh
compound
hydroxy
alkyl
norpregna
Prior art date
Application number
NO20003254A
Other languages
English (en)
Norwegian (no)
Other versions
NO20003254L (no
NO20003254D0 (no
Inventor
Masato Tanabe
Richard H Peters
Wan-Ru Chao
Ling Jong
Original Assignee
Stanford Res Inst Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Stanford Res Inst Int filed Critical Stanford Res Inst Int
Publication of NO20003254D0 publication Critical patent/NO20003254D0/no
Publication of NO20003254L publication Critical patent/NO20003254L/no
Publication of NO317978B1 publication Critical patent/NO317978B1/no

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/02Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/04Drugs for genital or sexual disorders; Contraceptives for inducing labour or abortion; Uterotonics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/14Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/02Suppositories; Bougies; Bases therefor; Ovules

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
NO20003254A 1997-12-24 2000-06-22 Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav NO317978B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/998,877 US6054446A (en) 1997-12-24 1997-12-24 Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
PCT/US1998/027406 WO1999033859A2 (fr) 1997-12-24 1998-12-23 Nouveaux steroides anti-oestrogenes, compositions pharmaceutiques associees et leur mode d'utilisation

Publications (3)

Publication Number Publication Date
NO20003254D0 NO20003254D0 (no) 2000-06-22
NO20003254L NO20003254L (no) 2000-08-21
NO317978B1 true NO317978B1 (no) 2005-01-17

Family

ID=25545637

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20003254A NO317978B1 (no) 1997-12-24 2000-06-22 Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav

Country Status (14)

Country Link
US (3) US6054446A (fr)
EP (4) EP1056768B1 (fr)
JP (4) JP2001525855A (fr)
KR (1) KR100464739B1 (fr)
CN (2) CN1332974C (fr)
AU (1) AU749597C (fr)
BR (1) BR9814435A (fr)
CA (1) CA2281844C (fr)
DE (2) DE69812433T2 (fr)
HU (1) HUP0100136A3 (fr)
IL (1) IL136972A0 (fr)
NO (1) NO317978B1 (fr)
RU (1) RU2233288C2 (fr)
WO (1) WO1999033859A2 (fr)

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KR100464739B1 (ko) 2005-01-05
JP2001525855A (ja) 2001-12-11
WO1999033859A3 (fr) 1999-12-23
BR9814435A (pt) 2004-08-10
HUP0100136A2 (hu) 2001-08-28
US6455517B1 (en) 2002-09-24
CN101130567A (zh) 2008-02-27
AU749597C (en) 2003-02-20
CA2281844C (fr) 2007-06-19
JP2007031446A (ja) 2007-02-08
US6054446A (en) 2000-04-25
EP1056768A2 (fr) 2000-12-06
US6281205B1 (en) 2001-08-28
JP2007051148A (ja) 2007-03-01
NO20003254L (no) 2000-08-21
WO1999033859A2 (fr) 1999-07-08
CA2281844A1 (fr) 1999-07-08
EP1847548A3 (fr) 2012-09-12
CN101130567B (zh) 2011-11-23
DE69812433T2 (de) 2004-02-12
KR20000075580A (ko) 2000-12-15
CN1291196A (zh) 2001-04-11
NO20003254D0 (no) 2000-06-22
DE69812433D1 (de) 2003-04-24
AU749597B2 (en) 2002-06-27
JP4718512B2 (ja) 2011-07-06
EP2305694A2 (fr) 2011-04-06
EP1310509A3 (fr) 2004-12-08
JP4959276B2 (ja) 2012-06-20
EP1310509A2 (fr) 2003-05-14
AU2010499A (en) 1999-07-19
RU2233288C2 (ru) 2004-07-27
WO1999033859A9 (fr) 1999-09-23
EP1056768B1 (fr) 2003-03-19
CN1332974C (zh) 2007-08-22
IL136972A0 (en) 2001-06-14
DE69839893D1 (de) 2008-09-25
EP1310509B1 (fr) 2008-08-13
JP2007269797A (ja) 2007-10-18
EP1847548A2 (fr) 2007-10-24
EP2305694A3 (fr) 2013-04-17
HUP0100136A3 (en) 2002-04-29
JP3968114B2 (ja) 2007-08-29

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