NO317978B1 - Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav - Google Patents
Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav Download PDFInfo
- Publication number
- NO317978B1 NO317978B1 NO20003254A NO20003254A NO317978B1 NO 317978 B1 NO317978 B1 NO 317978B1 NO 20003254 A NO20003254 A NO 20003254A NO 20003254 A NO20003254 A NO 20003254A NO 317978 B1 NO317978 B1 NO 317978B1
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- Norway
- Prior art keywords
- arh
- compound
- hydroxy
- alkyl
- norpregna
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
-
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/04—Drugs for genital or sexual disorders; Contraceptives for inducing labour or abortion; Uterotonics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/14—Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Pregnancy & Childbirth (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/998,877 US6054446A (en) | 1997-12-24 | 1997-12-24 | Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use |
PCT/US1998/027406 WO1999033859A2 (fr) | 1997-12-24 | 1998-12-23 | Nouveaux steroides anti-oestrogenes, compositions pharmaceutiques associees et leur mode d'utilisation |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20003254D0 NO20003254D0 (no) | 2000-06-22 |
NO20003254L NO20003254L (no) | 2000-08-21 |
NO317978B1 true NO317978B1 (no) | 2005-01-17 |
Family
ID=25545637
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20003254A NO317978B1 (no) | 1997-12-24 | 2000-06-22 | Anti-ostrogeniske steroider og farmasoytisk preparat inneholdende samme, samt anvendelse derav |
Country Status (14)
Country | Link |
---|---|
US (3) | US6054446A (fr) |
EP (4) | EP1056768B1 (fr) |
JP (4) | JP2001525855A (fr) |
KR (1) | KR100464739B1 (fr) |
CN (2) | CN1332974C (fr) |
AU (1) | AU749597C (fr) |
BR (1) | BR9814435A (fr) |
CA (1) | CA2281844C (fr) |
DE (2) | DE69812433T2 (fr) |
HU (1) | HUP0100136A3 (fr) |
IL (1) | IL136972A0 (fr) |
NO (1) | NO317978B1 (fr) |
RU (1) | RU2233288C2 (fr) |
WO (1) | WO1999033859A2 (fr) |
Families Citing this family (53)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5504074A (en) | 1993-08-06 | 1996-04-02 | Children's Medical Center Corporation | Estrogenic compounds as anti-angiogenic agents |
US6908910B2 (en) | 1993-08-06 | 2005-06-21 | The Children's Medical Center Corporation | Estrogenic compounds as anti-mitotic agents |
WO2001012206A2 (fr) * | 1999-08-13 | 2001-02-22 | Heinrich Wieland | Substances et moyens permettant d'influencer positivement le collagene |
US7087592B1 (en) | 1999-08-23 | 2006-08-08 | Entre Med, Inc. | Compositions comprising purified 2-methoxyestradiol and methods of producing same |
AUPQ342599A0 (en) * | 1999-10-14 | 1999-11-04 | University Of Melbourne, The | Conjugates and uses thereof |
WO2001058919A2 (fr) * | 2000-02-11 | 2001-08-16 | Sri International | Synthese de steroides anti-oestrogenique et d'autres steroides therapeutiques issus de 21-hydroxy-19-norpregna-4-ene-3-one |
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1997
- 1997-12-24 US US08/998,877 patent/US6054446A/en not_active Expired - Lifetime
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- 1998-12-23 EP EP98964882A patent/EP1056768B1/fr not_active Expired - Lifetime
- 1998-12-23 IL IL13697298A patent/IL136972A0/xx not_active IP Right Cessation
- 1998-12-23 EP EP10177213.5A patent/EP2305694A3/fr not_active Withdrawn
- 1998-12-23 DE DE69812433T patent/DE69812433T2/de not_active Expired - Lifetime
- 1998-12-23 KR KR10-1999-7007640A patent/KR100464739B1/ko not_active IP Right Cessation
- 1998-12-23 DE DE69839893T patent/DE69839893D1/de not_active Expired - Lifetime
- 1998-12-23 AU AU20104/99A patent/AU749597C/en not_active Ceased
- 1998-12-23 EP EP03000183A patent/EP1310509B1/fr not_active Expired - Lifetime
- 1998-12-23 EP EP07015863A patent/EP1847548A3/fr not_active Withdrawn
- 1998-12-23 HU HU0100136A patent/HUP0100136A3/hu unknown
- 1998-12-23 BR BR9814435-9A patent/BR9814435A/pt not_active Application Discontinuation
- 1998-12-23 JP JP53517299A patent/JP2001525855A/ja not_active Withdrawn
- 1998-12-23 WO PCT/US1998/027406 patent/WO1999033859A2/fr active IP Right Grant
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- 1998-12-23 CN CN200710128699XA patent/CN101130567B/zh not_active Expired - Lifetime
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