NO311934B1 - Benzocykloheptatiofenforbindelser - Google Patents
Benzocykloheptatiofenforbindelser Download PDFInfo
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- NO311934B1 NO311934B1 NO19994823A NO994823A NO311934B1 NO 311934 B1 NO311934 B1 NO 311934B1 NO 19994823 A NO19994823 A NO 19994823A NO 994823 A NO994823 A NO 994823A NO 311934 B1 NO311934 B1 NO 311934B1
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- 235000020357 syrup Nutrition 0.000 description 1
- 239000000454 talc Substances 0.000 description 1
- 229910052623 talc Inorganic materials 0.000 description 1
- 235000012222 talc Nutrition 0.000 description 1
- 229960000195 terbutaline Drugs 0.000 description 1
- 229960000337 tetryzoline Drugs 0.000 description 1
- 238000011287 therapeutic dose Methods 0.000 description 1
- 238000002560 therapeutic procedure Methods 0.000 description 1
- RTKIYNMVFMVABJ-UHFFFAOYSA-L thimerosal Chemical compound [Na+].CC[Hg]SC1=CC=CC=C1C([O-])=O RTKIYNMVFMVABJ-UHFFFAOYSA-L 0.000 description 1
- 229940033663 thimerosal Drugs 0.000 description 1
- 210000001519 tissue Anatomy 0.000 description 1
- 239000000606 toothpaste Substances 0.000 description 1
- 231100000027 toxicology Toxicity 0.000 description 1
- 210000003437 trachea Anatomy 0.000 description 1
- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
- 230000032258 transport Effects 0.000 description 1
- 235000015112 vegetable and seed oil Nutrition 0.000 description 1
- 239000008158 vegetable oil Substances 0.000 description 1
- 238000005406 washing Methods 0.000 description 1
- 238000005303 weighing Methods 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Ophthalmology & Optometry (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Curing Cements, Concrete, And Artificial Stone (AREA)
- Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US4390597P | 1997-04-03 | 1997-04-03 | |
| PCT/US1998/006576 WO1998043640A1 (fr) | 1997-04-03 | 1998-04-02 | Composes de benzocycloheptathiophene |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO994823D0 NO994823D0 (no) | 1999-10-04 |
| NO994823L NO994823L (no) | 1999-10-07 |
| NO311934B1 true NO311934B1 (no) | 2002-02-18 |
Family
ID=21929513
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19994823A NO311934B1 (no) | 1997-04-03 | 1999-10-04 | Benzocykloheptatiofenforbindelser |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US6207683B1 (fr) |
| EP (1) | EP0977568B1 (fr) |
| JP (1) | JP2001519789A (fr) |
| KR (1) | KR20010005791A (fr) |
| CN (1) | CN1128789C (fr) |
| AT (1) | ATE319450T1 (fr) |
| AU (1) | AU733325B2 (fr) |
| BR (1) | BR9807911A (fr) |
| CA (1) | CA2283663C (fr) |
| DE (1) | DE69833748T2 (fr) |
| HK (1) | HK1027961A1 (fr) |
| ID (1) | ID24487A (fr) |
| IL (1) | IL131999A (fr) |
| NO (1) | NO311934B1 (fr) |
| NZ (1) | NZ337843A (fr) |
| PL (1) | PL336007A1 (fr) |
| RU (1) | RU2193557C2 (fr) |
| WO (1) | WO1998043640A1 (fr) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9908014D0 (en) * | 1999-04-08 | 1999-06-02 | Scherer Corp R P | Pharmaceutical compositions |
| EP1218007B1 (fr) | 1999-09-13 | 2011-07-20 | Bridge Pharma, Inc. | Isomeres de ketotifene optiquement actifs et metabolites therapeutiquement actifs |
| US20100166804A1 (en) * | 2007-05-23 | 2010-07-01 | Dennis Penn | Methods |
| WO2009096080A1 (fr) * | 2008-01-30 | 2009-08-06 | Nippon Zoki Pharmaceutical Co., Ltd. | Dérivé de piperidine |
| WO2009142772A2 (fr) | 2008-05-23 | 2009-11-26 | Mastcell Pharmaceuticals, Inc. | Méthodes et traitement d’allergies et inflammations associées à des pathologies gastro-intestinales |
| JP5083989B2 (ja) * | 2008-11-20 | 2012-11-28 | 日本臓器製薬株式会社 | ピペリジン誘導体を含有する医薬 |
| WO2010107525A1 (fr) * | 2009-03-17 | 2010-09-23 | Aciex Therapeutics, Inc. | Formulations ophtalmiques de kétotifène et procédés d'utilisation |
| CN103619839B (zh) * | 2011-06-28 | 2016-06-01 | 福建省闽东力捷迅药业有限公司 | 抗-变态反应的苯并环庚并噻吩衍生物 |
| US8557846B1 (en) | 2012-10-23 | 2013-10-15 | Bridge Pharma, Inc. | Medicinal treatment of dermal diseases in dogs |
| US8778971B2 (en) | 2012-10-23 | 2014-07-15 | Bridge Pharma, Inc. | Medicinal treatment of dermal diseases in companion animals |
| US20150272941A1 (en) | 2012-10-30 | 2015-10-01 | Bridge Pharma, Inc. | Medicinal treatment of chronic pulmonary inflammatory diseases with norketotifen |
| US20140120121A1 (en) | 2012-10-30 | 2014-05-01 | Bridge Pharma, Inc. | Medicinal treatment of atopic inflammatory diseases |
| US9439895B2 (en) | 2013-08-06 | 2016-09-13 | Bridge Pharma, Inc. | Methods of treating pruritic conditions mediated through non-histaminergic mechanisms in diabetic patients |
| US9345697B2 (en) | 2013-08-06 | 2016-05-24 | Bridge Pharma, Inc. | Methods of treatment of non-histaminic pruritus |
| US9138431B2 (en) | 2013-08-06 | 2015-09-22 | Bridge Pharma, Inc. | Methods of treatment of histamine H-4 receptor-related pruritus |
| CN104045633B (zh) * | 2014-06-26 | 2017-07-21 | 福建省闽东力捷迅药业有限公司 | 一种富马酸卢帕替芬晶型a及其制备方法 |
| CN104031035B (zh) * | 2014-06-26 | 2017-08-25 | 福建省闽东力捷迅药业有限公司 | 一种富马酸卢帕替芬混晶及其制备方法 |
| ES2703693T3 (es) * | 2015-06-11 | 2019-03-12 | Bridge Pharma Inc | Métodos de tratamiento del prurito no histamínico en mamíferos |
| JP2019529541A (ja) | 2016-09-08 | 2019-10-17 | エマーゴ セラピューティクス，インク． | 高サイトカイン血症及びウィルス感染の処置の為の肥満細胞安定剤 |
| WO2018075574A1 (fr) | 2016-10-18 | 2018-04-26 | Emergo Therapeutics, Inc. | Stabilisateurs de mastocytes pour le traitement d'états inflammatoires chroniques |
| CN109180666A (zh) * | 2018-09-07 | 2019-01-11 | 福建省闽东力捷迅药业有限公司 | 一种富马酸卢帕替芬的杂质c及其制备方法和检测方法 |
| CN115960135A (zh) * | 2022-07-21 | 2023-04-14 | 华创合成制药股份有限公司 | 抗组胺类化合物及其制备方法和用途 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1470263A1 (de) * | 1963-12-19 | 1969-05-29 | Sandoz Ag | Neue Heterocyclische Verbindungen und Verfahren zu ihrer Herstellung |
| DE2626583A1 (de) * | 1975-06-24 | 1977-01-13 | Sandoz Ag | Neue benzocycloheptathiophenderivate ihre herstellung und ihre verwendung als heilmittel |
| US4355036A (en) * | 1980-06-19 | 1982-10-19 | Schering Corporation | Tricyclic-substituted piperidine antihistamines |
| US5250681A (en) | 1988-06-02 | 1993-10-05 | Ajinomoto Co., Inc. | Piperidine derivatives and hypotensives containing the same |
-
1998
- 1998-04-02 AU AU68812/98A patent/AU733325B2/en not_active Ceased
- 1998-04-02 JP JP54201898A patent/JP2001519789A/ja not_active Ceased
- 1998-04-02 RU RU99123048/04A patent/RU2193557C2/ru not_active IP Right Cessation
- 1998-04-02 KR KR1019997008863A patent/KR20010005791A/ko not_active Application Discontinuation
- 1998-04-02 NZ NZ337843A patent/NZ337843A/en unknown
- 1998-04-02 EP EP98914461A patent/EP0977568B1/fr not_active Expired - Lifetime
- 1998-04-02 US US09/381,351 patent/US6207683B1/en not_active Expired - Lifetime
- 1998-04-02 BR BR9807911-5A patent/BR9807911A/pt not_active IP Right Cessation
- 1998-04-02 CN CN98805506A patent/CN1128789C/zh not_active Expired - Fee Related
- 1998-04-02 DE DE69833748T patent/DE69833748T2/de not_active Expired - Fee Related
- 1998-04-02 CA CA002283663A patent/CA2283663C/fr not_active Expired - Fee Related
- 1998-04-02 ID IDW991141A patent/ID24487A/id unknown
- 1998-04-02 PL PL98336007A patent/PL336007A1/xx unknown
- 1998-04-02 AT AT98914461T patent/ATE319450T1/de not_active IP Right Cessation
- 1998-04-02 IL IL13199998A patent/IL131999A/en active IP Right Grant
- 1998-04-02 WO PCT/US1998/006576 patent/WO1998043640A1/fr active IP Right Grant
-
1999
- 1999-10-04 NO NO19994823A patent/NO311934B1/no unknown
-
2000
- 2000-11-15 HK HK00107262A patent/HK1027961A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0977568A4 (fr) | 2001-03-21 |
| NO994823D0 (no) | 1999-10-04 |
| CA2283663A1 (fr) | 1998-10-08 |
| HK1027961A1 (en) | 2001-02-02 |
| US6207683B1 (en) | 2001-03-27 |
| BR9807911A (pt) | 2000-02-22 |
| CN1128789C (zh) | 2003-11-26 |
| NZ337843A (en) | 2001-11-30 |
| CA2283663C (fr) | 2006-07-25 |
| EP0977568B1 (fr) | 2006-03-08 |
| DE69833748D1 (de) | 2006-05-04 |
| AU733325B2 (en) | 2001-05-10 |
| EP0977568A1 (fr) | 2000-02-09 |
| WO1998043640A1 (fr) | 1998-10-08 |
| JP2001519789A (ja) | 2001-10-23 |
| KR20010005791A (ko) | 2001-01-15 |
| PL336007A1 (en) | 2000-06-05 |
| NO994823L (no) | 1999-10-07 |
| ATE319450T1 (de) | 2006-03-15 |
| IL131999A (en) | 2004-06-20 |
| CN1258219A (zh) | 2000-06-28 |
| ID24487A (id) | 2000-07-20 |
| RU2193557C2 (ru) | 2002-11-27 |
| DE69833748T2 (de) | 2006-11-23 |
| IL131999A0 (en) | 2001-03-19 |
| AU6881298A (en) | 1998-10-22 |
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