NO20092422L - Cykloalkylaminsubstituerte isokinolonderivater - Google Patents

Cykloalkylaminsubstituerte isokinolonderivater

Info

Publication number
NO20092422L
NO20092422L NO20092422A NO20092422A NO20092422L NO 20092422 L NO20092422 L NO 20092422L NO 20092422 A NO20092422 A NO 20092422A NO 20092422 A NO20092422 A NO 20092422A NO 20092422 L NO20092422 L NO 20092422L
Authority
NO
Norway
Prior art keywords
isoquinolone derivatives
substituted isoquinolone
cycloalkylamine
cycloalkylamine substituted
treatment
Prior art date
Application number
NO20092422A
Other languages
English (en)
Inventor
Armin Hofmeister
Oliver Plettenburg
Matthias Lohn
John Weston
Joachim Brendel
Katrin Lorenz
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38565513&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20092422(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of NO20092422L publication Critical patent/NO20092422L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
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Abstract

Oppfinnelsen angår 6-substituerte isokinolonderivater med formel (I), anvendelige for behandling og/eller behandling av sykdommer assosiert med Rho-kinase og/eller Rho-kinase mediert fosforylering av yosinlettkjede fosfatase og sammensetninger som inneholder slike forbindelser.
NO20092422A 2006-12-27 2009-06-25 Cykloalkylaminsubstituerte isokinolonderivater NO20092422L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06026899 2006-12-27
PCT/EP2007/011164 WO2008077551A1 (en) 2006-12-27 2007-12-19 Cycloalkylamine substituted isoquinolone derivatives

Publications (1)

Publication Number Publication Date
NO20092422L true NO20092422L (no) 2009-09-25

Family

ID=38565513

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20092422A NO20092422L (no) 2006-12-27 2009-06-25 Cykloalkylaminsubstituerte isokinolonderivater

Country Status (31)

Country Link
US (1) US8742116B2 (no)
EP (1) EP2125745B1 (no)
JP (1) JP5405314B2 (no)
KR (1) KR101474228B1 (no)
CN (1) CN101595094B (no)
AR (1) AR064492A1 (no)
AU (1) AU2007338407B2 (no)
BR (1) BRPI0722064A2 (no)
CA (1) CA2673917C (no)
CL (1) CL2007003821A1 (no)
CO (1) CO6210726A2 (no)
CR (1) CR10813A (no)
DO (1) DOP2009000164A (no)
EC (1) ECSP099467A (no)
ES (1) ES2625266T3 (no)
GT (1) GT200900179A (no)
HK (1) HK1139390A1 (no)
IL (1) IL199540A (no)
MA (1) MA31075B1 (no)
MX (1) MX2009005966A (no)
MY (1) MY155009A (no)
NI (1) NI200900108A (no)
NO (1) NO20092422L (no)
NZ (1) NZ577980A (no)
RU (1) RU2457203C2 (no)
SV (1) SV2009003318A (no)
TN (1) TN2009000269A1 (no)
TW (1) TWI434689B (no)
UY (1) UY30843A1 (no)
WO (1) WO2008077551A1 (no)
ZA (1) ZA200903551B (no)

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TW201834020A (zh) 2003-10-28 2018-09-16 日商尼康股份有限公司 照明光學裝置、曝光裝置、曝光方法以及元件製造方法
TWI512335B (zh) 2003-11-20 2015-12-11 尼康股份有限公司 光束變換元件、光學照明裝置、曝光裝置、以及曝光方法
TWI412067B (zh) 2004-02-06 2013-10-11 尼康股份有限公司 偏光變換元件、光學照明裝置、曝光裝置以及曝光方法
US7470787B2 (en) 2005-07-11 2008-12-30 Aerie Pharmaceuticals, Inc. Isoquinoline compounds
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