ZA200903551B - Cycloalkylamine substituted isoquinolone derivatives - Google Patents

Cycloalkylamine substituted isoquinolone derivatives

Info

Publication number
ZA200903551B
ZA200903551B ZA200903551A ZA200903551A ZA200903551B ZA 200903551 B ZA200903551 B ZA 200903551B ZA 200903551 A ZA200903551 A ZA 200903551A ZA 200903551 A ZA200903551 A ZA 200903551A ZA 200903551 B ZA200903551 B ZA 200903551B
Authority
ZA
South Africa
Prior art keywords
isoquinolone derivatives
substituted isoquinolone
cycloalkylamine
cycloalkylamine substituted
derivatives
Prior art date
Application number
ZA200903551A
Other languages
English (en)
Inventor
Oliver Plettenburg
Armin Hofmeister
Katrin Lorenz
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38565513&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200903551(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of ZA200903551B publication Critical patent/ZA200903551B/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pregnancy & Childbirth (AREA)
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ZA200903551A 2006-12-27 2009-05-22 Cycloalkylamine substituted isoquinolone derivatives ZA200903551B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP06026899 2006-12-27

Publications (1)

Publication Number Publication Date
ZA200903551B true ZA200903551B (en) 2010-03-31

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ID=38565513

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200903551A ZA200903551B (en) 2006-12-27 2009-05-22 Cycloalkylamine substituted isoquinolone derivatives

Country Status (31)

Country Link
US (1) US8742116B2 (xx)
EP (1) EP2125745B1 (xx)
JP (1) JP5405314B2 (xx)
KR (1) KR101474228B1 (xx)
CN (1) CN101595094B (xx)
AR (1) AR064492A1 (xx)
AU (1) AU2007338407B2 (xx)
BR (1) BRPI0722064A2 (xx)
CA (1) CA2673917C (xx)
CL (1) CL2007003821A1 (xx)
CO (1) CO6210726A2 (xx)
CR (1) CR10813A (xx)
DO (1) DOP2009000164A (xx)
EC (1) ECSP099467A (xx)
ES (1) ES2625266T3 (xx)
GT (1) GT200900179A (xx)
HK (1) HK1139390A1 (xx)
IL (1) IL199540A (xx)
MA (1) MA31075B1 (xx)
MX (1) MX2009005966A (xx)
MY (1) MY155009A (xx)
NI (1) NI200900108A (xx)
NO (1) NO20092422L (xx)
NZ (1) NZ577980A (xx)
RU (1) RU2457203C2 (xx)
SV (1) SV2009003318A (xx)
TN (1) TN2009000269A1 (xx)
TW (1) TWI434689B (xx)
UY (1) UY30843A1 (xx)
WO (1) WO2008077551A1 (xx)
ZA (1) ZA200903551B (xx)

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