NO20083836L - N-hydroksyakrylamidforbindelser - Google Patents

N-hydroksyakrylamidforbindelser

Info

Publication number
NO20083836L
NO20083836L NO20083836A NO20083836A NO20083836L NO 20083836 L NO20083836 L NO 20083836L NO 20083836 A NO20083836 A NO 20083836A NO 20083836 A NO20083836 A NO 20083836A NO 20083836 L NO20083836 L NO 20083836L
Authority
NO
Norway
Prior art keywords
novel
pharmaceutically acceptable
acceptable salts
same
hdac
Prior art date
Application number
NO20083836A
Other languages
English (en)
Norwegian (no)
Inventor
Fumiyuki Shirai
Hideo Tsutsumi
Hiromichi Itani
Yoshihiro Kozuki
Yoshiteru Eikyu
Taro Masunaga
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2006900588A external-priority patent/AU2006900588A0/en
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of NO20083836L publication Critical patent/NO20083836L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
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NO20083836A 2006-02-07 2008-09-05 N-hydroksyakrylamidforbindelser NO20083836L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AU2006900588A AU2006900588A0 (en) 2006-02-07 HDAC inhibitor
PCT/JP2007/052447 WO2007091703A1 (en) 2006-02-07 2007-02-06 N-hydroxyacrylamide compounds

Publications (1)

Publication Number Publication Date
NO20083836L true NO20083836L (no) 2008-11-05

Family

ID=38038616

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083836A NO20083836L (no) 2006-02-07 2008-09-05 N-hydroksyakrylamidforbindelser

Country Status (19)

Country Link
US (1) US7750155B2 (es)
EP (1) EP1981877B1 (es)
JP (1) JP5218057B2 (es)
KR (1) KR20080091297A (es)
CN (1) CN101379059A (es)
AT (1) ATE554084T1 (es)
AU (1) AU2007213018A1 (es)
BR (1) BRPI0707693A2 (es)
CA (1) CA2641579A1 (es)
ES (1) ES2384121T3 (es)
IL (1) IL193252A0 (es)
MX (1) MX2008010035A (es)
NO (1) NO20083836L (es)
PL (1) PL1981877T3 (es)
PT (1) PT1981877E (es)
RU (1) RU2008135979A (es)
TW (1) TW200806652A (es)
WO (1) WO2007091703A1 (es)
ZA (1) ZA200806778B (es)

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WO2009118370A1 (en) 2008-03-27 2009-10-01 Janssen Pharmaceutica Nv Aza-bicyclohexyl substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
WO2011017448A1 (en) * 2009-08-05 2011-02-10 The Trustees Of The University Of Pennsylvania Use of histone deacetylase inhibitors for treatment of autoimmune diseases
US8614223B2 (en) * 2010-11-16 2013-12-24 Acetylon Pharmaceuticals, Inc. Pyrimidine hydroxy amide compounds as protein deacetylase inhibitors and methods of use thereof
ES2929576T3 (es) 2013-10-08 2022-11-30 Acetylon Pharmaceuticals Inc Combinaciones de inhibidores de histona deacetilasa 6 y el inhibidor de Her2 lapatinib para el uso en el tratamiento del cáncer de mama
EP3055299B1 (en) 2013-10-10 2021-01-06 Acetylon Pharmaceuticals, Inc. Pyrimidine hydroxy amide compounds as histone deacetylase inhibitors
JP2016534069A (ja) 2013-10-24 2016-11-04 メイヨ・ファウンデーション・フォー・メディカル・エデュケーション・アンド・リサーチ Ｈｄａｃ６阻害剤での多嚢胞性疾患の治療
PE20161030A1 (es) 2013-12-03 2016-11-06 Acetylon Pharmaceuticals Inc Combinaciones de inhibidores de histona deacetilasa y farmacos inmunomoduladores
US9464073B2 (en) 2014-02-26 2016-10-11 Acetylon Pharmaceuticals, Inc. Pyrimidine hydroxy amide compounds as HDAC6 selective inhibitors
EP3166603B1 (en) 2014-07-07 2020-02-12 Acetylon Pharmaceuticals, Inc. Treatment of leukemia with histone deacetylase inhibitors
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PT1981877E (pt) 2012-05-24
RU2008135979A (ru) 2010-03-20
BRPI0707693A2 (pt) 2011-05-10
EP1981877A1 (en) 2008-10-22
ATE554084T1 (de) 2012-05-15
WO2007091703A1 (en) 2007-08-16
EP1981877B1 (en) 2012-04-18
ZA200806778B (en) 2009-11-25
AU2007213018A1 (en) 2007-08-16
US20090054465A1 (en) 2009-02-26
JP5218057B2 (ja) 2013-06-26
PL1981877T3 (pl) 2012-12-31
ES2384121T3 (es) 2012-06-29
KR20080091297A (ko) 2008-10-09
JP2009525945A (ja) 2009-07-16
US7750155B2 (en) 2010-07-06
IL193252A0 (en) 2009-02-11
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CN101379059A (zh) 2009-03-04
CA2641579A1 (en) 2007-08-16

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