NO20083304L - Imidazo(1,2-A)pyridin-3-yl-eddiksyrehydrazider, fremgangsmater for deres fremstilling og farmasoytiske anvendelser derav - Google Patents
Imidazo(1,2-A)pyridin-3-yl-eddiksyrehydrazider, fremgangsmater for deres fremstilling og farmasoytiske anvendelser deravInfo
- Publication number
- NO20083304L NO20083304L NO20083304A NO20083304A NO20083304L NO 20083304 L NO20083304 L NO 20083304L NO 20083304 A NO20083304 A NO 20083304A NO 20083304 A NO20083304 A NO 20083304A NO 20083304 L NO20083304 L NO 20083304L
- Authority
- NO
- Norway
- Prior art keywords
- pyridin
- acetic acid
- imidazo
- acid hydrazides
- processes
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Oppfinnelsen tilveiebringer nye imidazo[1,2-a]pyridin-3-yl-eddiksyrehydrazider med formel (I) hvor R1, R2 og R3 har forskjellige betydninger, og farmasøytisk akseptable salter, polymorfer, hydrater, tautomerer, oppløsninger og stereoisomerer av dem. Forbindelser med formel (I) er nyttige for å behandle eller å forebygge, i et menneske eller ikke-humant pattedyr, sykdommer som er assosiert med modulering av GABAA reseptorer, angst, epilepsi, søvnlidelser som inkluderer søvnløshet og for å indusere beroligelse-hypnose, anestesi, søvn og muskelavslapping. Oppfinnelsen tilveiebringer også syntetiske prosesser for å lage nevnte forbindelser.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06100030A EP1803722A1 (en) | 2006-01-03 | 2006-01-03 | Imidazo[1,2-a]pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof |
PCT/EP2006/070130 WO2007077159A1 (en) | 2006-01-03 | 2006-12-21 | Imidazo (1,2-a)pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20083304L true NO20083304L (no) | 2008-09-24 |
Family
ID=36691692
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20083304A NO20083304L (no) | 2006-01-03 | 2008-07-25 | Imidazo(1,2-A)pyridin-3-yl-eddiksyrehydrazider, fremgangsmater for deres fremstilling og farmasoytiske anvendelser derav |
Country Status (23)
Country | Link |
---|---|
US (2) | US7943611B2 (no) |
EP (2) | EP1803722A1 (no) |
JP (1) | JP2009522327A (no) |
KR (1) | KR20080083194A (no) |
CN (1) | CN101395156B (no) |
AR (1) | AR058738A1 (no) |
AT (1) | ATE430748T1 (no) |
AU (1) | AU2006334364B2 (no) |
BR (1) | BRPI0620885A2 (no) |
CA (1) | CA2635802A1 (no) |
DE (1) | DE602006006725D1 (no) |
DK (1) | DK1973907T3 (no) |
ES (1) | ES2327278T3 (no) |
HK (1) | HK1123792A1 (no) |
IL (1) | IL192563A0 (no) |
NO (1) | NO20083304L (no) |
PE (1) | PE20071059A1 (no) |
PL (1) | PL1973907T3 (no) |
PT (1) | PT1973907E (no) |
RU (1) | RU2008131798A (no) |
TW (1) | TW200800992A (no) |
UY (1) | UY30066A1 (no) |
WO (1) | WO2007077159A1 (no) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1845098A1 (en) * | 2006-03-29 | 2007-10-17 | Ferrer Internacional, S.A. | Imidazo[1,2-b]pyridazines, their processes of preparation and their use as GABA receptor ligands |
CN109053726A (zh) * | 2018-09-14 | 2018-12-21 | 烟台万润药业有限公司 | 一种唑吡坦酸的制备方法 |
KR102349934B1 (ko) | 2020-10-19 | 2022-01-12 | 신해찬 | 층간소음방지부재 및 이를 이용한 층간소음방지층 시공방법 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU532001B2 (en) * | 1978-11-20 | 1983-09-15 | Sumitomo Chemical Company, Limited | Polycyclic indole derivatives |
FR2492382A1 (fr) * | 1980-10-22 | 1982-04-23 | Synthelabo | Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique |
ES2151834B1 (es) * | 1998-08-06 | 2001-08-16 | Sint Quimica Sa | Procedimiento para preparar n,n,6-trimetil-2-(4-metilfenil)-imidazo-(1,2-a)-piridina-3-acetamida y sus sales. |
CA2544213A1 (en) * | 2003-10-28 | 2005-05-19 | Sepracor Inc. | Imidazo[1,2-a]pyridine anxiolytics |
-
2006
- 2006-01-03 EP EP06100030A patent/EP1803722A1/en not_active Withdrawn
- 2006-12-21 RU RU2008131798/04A patent/RU2008131798A/ru unknown
- 2006-12-21 BR BRPI0620885-1A patent/BRPI0620885A2/pt not_active IP Right Cessation
- 2006-12-21 DK DK06841585T patent/DK1973907T3/da active
- 2006-12-21 KR KR1020087018796A patent/KR20080083194A/ko not_active Application Discontinuation
- 2006-12-21 PL PL06841585T patent/PL1973907T3/pl unknown
- 2006-12-21 AT AT06841585T patent/ATE430748T1/de active
- 2006-12-21 WO PCT/EP2006/070130 patent/WO2007077159A1/en active Application Filing
- 2006-12-21 JP JP2008548979A patent/JP2009522327A/ja not_active Ceased
- 2006-12-21 EP EP06841585A patent/EP1973907B1/en not_active Not-in-force
- 2006-12-21 AU AU2006334364A patent/AU2006334364B2/en not_active Ceased
- 2006-12-21 US US12/087,423 patent/US7943611B2/en not_active Expired - Fee Related
- 2006-12-21 ES ES06841585T patent/ES2327278T3/es active Active
- 2006-12-21 DE DE602006006725T patent/DE602006006725D1/de active Active
- 2006-12-21 CA CA002635802A patent/CA2635802A1/en not_active Abandoned
- 2006-12-21 CN CN2006800536332A patent/CN101395156B/zh not_active Expired - Fee Related
- 2006-12-21 PT PT06841585T patent/PT1973907E/pt unknown
- 2006-12-22 PE PE2006001689A patent/PE20071059A1/es not_active Application Discontinuation
- 2006-12-26 UY UY30066A patent/UY30066A1/es unknown
- 2006-12-26 AR ARP060105781A patent/AR058738A1/es not_active Application Discontinuation
- 2006-12-27 TW TW095149148A patent/TW200800992A/zh unknown
-
2008
- 2008-07-01 IL IL192563A patent/IL192563A0/en unknown
- 2008-07-25 NO NO20083304A patent/NO20083304L/no not_active Application Discontinuation
-
2009
- 2009-02-18 HK HK09101530.6A patent/HK1123792A1/xx not_active IP Right Cessation
-
2011
- 2011-01-24 US US13/012,258 patent/US20110118256A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
PL1973907T3 (pl) | 2009-10-30 |
AU2006334364B2 (en) | 2011-09-29 |
AU2006334364A1 (en) | 2007-07-12 |
US20110118256A1 (en) | 2011-05-19 |
BRPI0620885A2 (pt) | 2011-11-29 |
AR058738A1 (es) | 2008-02-20 |
CN101395156A (zh) | 2009-03-25 |
EP1803722A1 (en) | 2007-07-04 |
DE602006006725D1 (de) | 2009-06-18 |
UY30066A1 (es) | 2007-04-30 |
JP2009522327A (ja) | 2009-06-11 |
CA2635802A1 (en) | 2007-07-12 |
DK1973907T3 (da) | 2009-08-24 |
ATE430748T1 (de) | 2009-05-15 |
EP1973907B1 (en) | 2009-05-06 |
EP1973907A1 (en) | 2008-10-01 |
CN101395156B (zh) | 2011-12-14 |
PT1973907E (pt) | 2009-07-28 |
IL192563A0 (en) | 2009-02-11 |
ES2327278T3 (es) | 2009-10-27 |
WO2007077159A1 (en) | 2007-07-12 |
US7943611B2 (en) | 2011-05-17 |
KR20080083194A (ko) | 2008-09-16 |
US20090176777A1 (en) | 2009-07-09 |
PE20071059A1 (es) | 2007-10-26 |
TW200800992A (en) | 2008-01-01 |
RU2008131798A (ru) | 2010-02-10 |
HK1123792A1 (en) | 2009-06-26 |
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Legal Events
Date | Code | Title | Description |
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FC2A | Withdrawal, rejection or dismissal of laid open patent application |