NO20080002L - Formuleringer av konjugerte ostrogener og bazedoxifen - Google Patents

Formuleringer av konjugerte ostrogener og bazedoxifen

Info

Publication number
NO20080002L
NO20080002L NO20080002A NO20080002A NO20080002L NO 20080002 L NO20080002 L NO 20080002L NO 20080002 A NO20080002 A NO 20080002A NO 20080002 A NO20080002 A NO 20080002A NO 20080002 L NO20080002 L NO 20080002L
Authority
NO
Norway
Prior art keywords
bazedoxifene
conjugated estrogens
formulations
salt
estrogens
Prior art date
Application number
NO20080002A
Other languages
English (en)
Inventor
Arwinder Nagi
Ramarao S Chatlapalli
Lawrence Van Pelt
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37401610&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20080002(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of NO20080002L publication Critical patent/NO20080002L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens

Abstract

Det beskrives faste doseringsformuleringer som inneholder konjugerte østrogener og bazedoxifen eller et salt derav. I enkelte utførelsesformer inkluderer blandingene en kjerne som omfatter konjugerte østrogener og minst ett overtrekk som omfatter bazedoxifen eller et salt derav.
NO20080002A 2005-06-29 2008-01-02 Formuleringer av konjugerte ostrogener og bazedoxifen NO20080002L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69488905P 2005-06-29 2005-06-29
PCT/US2006/025348 WO2007002823A2 (en) 2005-06-29 2006-06-28 Formulations of conjugated estrogens and bazedoxifene

Publications (1)

Publication Number Publication Date
NO20080002L true NO20080002L (no) 2008-03-12

Family

ID=37401610

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20080002A NO20080002L (no) 2005-06-29 2008-01-02 Formuleringer av konjugerte ostrogener og bazedoxifen

Country Status (19)

Country Link
US (1) US20070003623A1 (no)
EP (1) EP1898888A2 (no)
JP (1) JP2008545012A (no)
KR (1) KR20080031037A (no)
CN (1) CN101252921A (no)
AR (1) AR054806A1 (no)
AU (1) AU2006263638A1 (no)
BR (1) BRPI0612586A2 (no)
CA (1) CA2613102A1 (no)
CR (1) CR9597A (no)
EC (1) ECSP078057A (no)
IL (1) IL188223A0 (no)
NI (1) NI200700331A (no)
NO (1) NO20080002L (no)
PA (1) PA8684501A1 (no)
PE (1) PE20070188A1 (no)
RU (1) RU2395286C2 (no)
TW (1) TW200738283A (no)
WO (1) WO2007002823A2 (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2400227C2 (ru) * 2004-04-08 2010-09-27 Вайет Состав, содержащий твердую дисперсию базедоксифен ацетата
US20080175905A1 (en) * 2006-11-29 2008-07-24 Wyeth Estrogen/serm and estrogen/progestin bi-layer tablets
AU2008206476A1 (en) * 2007-01-12 2008-07-24 Wyeth Tablet-in-tablet compositions
PE20090100A1 (es) * 2007-03-30 2009-02-26 Wyeth Corp Metodos de separacion y deteccion de acetato de bacedoxifeno en composiciones farmaceuticas
TW201127386A (en) * 2009-10-27 2011-08-16 Wyeth Llc Bazedoxifene formulations with antioxidants
CN102985072A (zh) * 2010-04-20 2013-03-20 希普拉有限公司 药物组合物
CN103119878B (zh) * 2010-07-29 2016-11-16 熵通信有限公司 用于消除交叉极化干扰和交叉卫星干扰的方法和装置
CN109908099B (zh) * 2011-05-13 2021-10-29 Eb Ip希博里塔布斯有限责任公司 药物递送系统
CN104013630B (zh) * 2014-05-23 2018-08-21 合肥九研医药科技开发有限公司 一种复方醋酸巴多昔芬雌激素组合物
US11147771B2 (en) 2015-06-18 2021-10-19 Estetra Sprl Orodispersible dosage unit containing an estetrol component
KR20220144885A (ko) 2016-08-05 2022-10-27 에스테트라, 소시에떼 아 레스폰서빌리떼 리미떼 월경통 및 생리통의 관리방법
WO2018182205A1 (ko) * 2017-03-30 2018-10-04 한미약품 주식회사 바제독시펜 아세테이트를 함유하는 안정화된 약제학적 조성물
JOP20200260A1 (ar) * 2018-04-19 2019-10-19 Estetra Sprl مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث
TWI801561B (zh) * 2018-04-19 2023-05-11 比利時商依思特拉私人有限責任公司 化合物及其用於緩解絕經相關症狀的用途

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2565115A (en) * 1948-10-28 1951-08-21 Squibb & Sons Inc Method of obtaining a conjugated estrogen preparation
US2720483A (en) * 1951-02-21 1955-10-11 Olin Mathieson Method of obtaining a conjugatedestrogen preparation
US5210081A (en) * 1992-02-26 1993-05-11 American Home Products Corporation Alkali metal 8,9-dehydroestrone sulfate esters
US5759577A (en) * 1995-01-17 1998-06-02 American Home Products Corporation Controlled release of steroids from sugar coatings
US5547948A (en) * 1995-01-17 1996-08-20 American Home Products Corporation Controlled release of steroids from sugar coatings
US5998402A (en) * 1996-04-19 1999-12-07 American Home Products Corporation 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
US6479535B1 (en) * 1998-05-15 2002-11-12 Wyeth 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations
JP4790178B2 (ja) * 1999-07-06 2011-10-12 アンドルシェルシュ・インコーポレイテッド 体重増加の処置方法および/または抑制方法
AR029538A1 (es) * 2000-07-06 2003-07-02 Wyeth Corp Composiciones farmaceuticas de agentes estrogenicos
MXPA04011634A (es) * 2002-06-13 2005-07-05 Wyeth Corp Regimenes de tratamiento con bazedoxifeno.
WO2005100314A1 (en) * 2004-04-07 2005-10-27 Wyeth Crystalline polymorph of bazedoxifene acetate
AR048527A1 (es) * 2004-04-07 2006-05-03 Wyeth Corp Variedades cristalinas de acetato de bazedoxifeno
RU2400227C2 (ru) * 2004-04-08 2010-09-27 Вайет Состав, содержащий твердую дисперсию базедоксифен ацетата
CA2561004A1 (en) * 2004-04-08 2005-10-27 Wyeth Bazedoxifene ascorbate as selective estrogen receptor modulator

Also Published As

Publication number Publication date
ECSP078057A (es) 2008-01-23
NI200700331A (es) 2009-02-16
WO2007002823A3 (en) 2007-08-09
PE20070188A1 (es) 2007-03-16
CN101252921A (zh) 2008-08-27
TW200738283A (en) 2007-10-16
CR9597A (es) 2008-03-06
CA2613102A1 (en) 2007-01-04
AU2006263638A1 (en) 2007-01-04
KR20080031037A (ko) 2008-04-07
AR054806A1 (es) 2007-07-18
RU2395286C2 (ru) 2010-07-27
BRPI0612586A2 (pt) 2010-11-23
WO2007002823A2 (en) 2007-01-04
PA8684501A1 (es) 2007-01-17
IL188223A0 (en) 2008-03-20
EP1898888A2 (en) 2008-03-19
RU2007148071A (ru) 2009-08-10
JP2008545012A (ja) 2008-12-11
US20070003623A1 (en) 2007-01-04

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