NO20072756L - 4-(4-(imidazol)-4-yl)-pyrimidin-2-ylamino)benzamider som CDK-inhibitorer - Google Patents

4-(4-(imidazol)-4-yl)-pyrimidin-2-ylamino)benzamider som CDK-inhibitorer

Info

Publication number
NO20072756L
NO20072756L NO20072756A NO20072756A NO20072756L NO 20072756 L NO20072756 L NO 20072756L NO 20072756 A NO20072756 A NO 20072756A NO 20072756 A NO20072756 A NO 20072756A NO 20072756 L NO20072756 L NO 20072756L
Authority
NO
Norway
Prior art keywords
benzamides
ylamino
imidazol
pyrimidin
cdk inhibitors
Prior art date
Application number
NO20072756A
Other languages
English (en)
Inventor
Maurice Raymond Verscho Finlay
Clifford David Jones
Clive Green
David Michael Andrews
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35645682&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20072756(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0427699A external-priority patent/GB0427699D0/en
Priority claimed from GB0515740A external-priority patent/GB0515740D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20072756L publication Critical patent/NO20072756L/no

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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Vascular Medicine (AREA)
  • Transplantation (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Forbindelser med formel (I): (I) hvor variable grupper er som definert heri og hvor farmasøytisk akseptable salter og in vivo hydrolyserbare estere er beskrevet. Også beskrevet er prosesser for deres fremstilling og anvendelse av dem som medikamenter, spesielt medikamenter for å produsere en cellecyklus-hemmende (anti-celle-proliferasjon) effekt hos et varmblodig dyr, så som mennesker. ?? ?? ?? ?? 1
NO20072756A 2004-12-17 2007-05-30 4-(4-(imidazol)-4-yl)-pyrimidin-2-ylamino)benzamider som CDK-inhibitorer NO20072756L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0427699A GB0427699D0 (en) 2004-12-17 2004-12-17 Chemical compounds
GB0515740A GB0515740D0 (en) 2005-07-30 2005-07-30 Chemical compounds
PCT/GB2005/004865 WO2006064251A1 (en) 2004-12-17 2005-12-15 4- (4- (imidazol-4-yl) pyrimidin-2-ylamino) benzamides as cdk inhibitors

Publications (1)

Publication Number Publication Date
NO20072756L true NO20072756L (no) 2007-08-30

Family

ID=35645682

Family Applications (1)

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NO20072756A NO20072756L (no) 2004-12-17 2007-05-30 4-(4-(imidazol)-4-yl)-pyrimidin-2-ylamino)benzamider som CDK-inhibitorer

Country Status (15)

Country Link
US (1) US20090099160A1 (no)
EP (1) EP1828183A1 (no)
JP (1) JP2008524191A (no)
KR (1) KR20070091018A (no)
AR (1) AR052170A1 (no)
AU (1) AU2005315392B2 (no)
BR (1) BRPI0517426A (no)
CA (1) CA2589793A1 (no)
IL (1) IL183526A0 (no)
MX (1) MX2007007272A (no)
NO (1) NO20072756L (no)
NZ (1) NZ555474A (no)
TW (1) TW200635924A (no)
UY (1) UY29277A1 (no)
WO (1) WO2006064251A1 (no)

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AU2005315392B2 (en) 2010-03-11
BRPI0517426A (pt) 2008-10-07
NZ555474A (en) 2010-10-29
WO2006064251A1 (en) 2006-06-22
CA2589793A1 (en) 2006-06-22
TW200635924A (en) 2006-10-16
EP1828183A1 (en) 2007-09-05
US20090099160A1 (en) 2009-04-16
IL183526A0 (en) 2007-09-20
UY29277A1 (es) 2006-07-31
AU2005315392A1 (en) 2006-06-22
AR052170A1 (es) 2007-03-07
MX2007007272A (es) 2007-07-11
JP2008524191A (ja) 2008-07-10
KR20070091018A (ko) 2007-09-06

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