NO20071008L - Fremgangsmate for fremstilling av N-piperidino-1,5-difenylpyrazol-3-karboksamidderivater - Google Patents
Fremgangsmate for fremstilling av N-piperidino-1,5-difenylpyrazol-3-karboksamidderivaterInfo
- Publication number
- NO20071008L NO20071008L NO20071008A NO20071008A NO20071008L NO 20071008 L NO20071008 L NO 20071008L NO 20071008 A NO20071008 A NO 20071008A NO 20071008 A NO20071008 A NO 20071008A NO 20071008 L NO20071008 L NO 20071008L
- Authority
- NO
- Norway
- Prior art keywords
- diphenylpyrazole
- piperidino
- preparation
- carboxamide derivatives
- hydrogen atom
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Abstract
Det er beskrevet en fremgangsmåte for fremstilling av en forbindelse av formel (I), hvori: R1 betyr et hydrogenatom eller halogenatom eller en (C1-C4)alkylgruppe; R2, R3, R4, R5, R6 og R7 betyr uavhengig av hverandre, et hydrogenatom eller halogenatom eller en (C1-C4)alkyl, (C1-C4)alkoksy eller trifluorometylgruppe, så vel som salter derav.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0408111A FR2873372B1 (fr) | 2004-07-22 | 2004-07-22 | Procede de preparation de derives n-piperidino-1,5- diphenylpyrazole-3-carboxamide |
PCT/FR2005/001850 WO2006021652A1 (fr) | 2004-07-22 | 2005-07-20 | Procede de preparation de derives n-piperidino-1,5-diphenylpyrazole-3-carboxamide |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20071008L true NO20071008L (no) | 2007-02-21 |
Family
ID=34949586
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20071008A NO20071008L (no) | 2004-07-22 | 2007-02-21 | Fremgangsmate for fremstilling av N-piperidino-1,5-difenylpyrazol-3-karboksamidderivater |
Country Status (21)
Country | Link |
---|---|
US (1) | US7462632B2 (no) |
EP (1) | EP1773783B1 (no) |
JP (1) | JP4879175B2 (no) |
KR (1) | KR20070036050A (no) |
CN (1) | CN100537543C (no) |
AR (1) | AR049995A1 (no) |
AT (1) | ATE466843T1 (no) |
AU (1) | AU2005276350A1 (no) |
BR (1) | BRPI0510399A (no) |
CA (1) | CA2564223A1 (no) |
DE (1) | DE602005021110D1 (no) |
FR (1) | FR2873372B1 (no) |
IL (1) | IL179107A0 (no) |
MA (1) | MA28576B1 (no) |
MX (1) | MXPA06012954A (no) |
NO (1) | NO20071008L (no) |
RU (1) | RU2329252C1 (no) |
TW (1) | TW200609223A (no) |
UY (1) | UY29023A1 (no) |
WO (1) | WO2006021652A1 (no) |
ZA (1) | ZA200609639B (no) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1816125A1 (en) * | 2006-02-02 | 2007-08-08 | Ranbaxy Laboratories, Ltd. | Novel crystalline forms of an antagonist of CB1 cannabinoid receptor and preparation method thereof |
WO2008026219A2 (en) * | 2006-09-01 | 2008-03-06 | Hetero Drugs Limited | Novel polymorphs of rimonabant |
US20100076197A1 (en) * | 2006-09-11 | 2010-03-25 | Hetero Drugs Limited | Process for rimonabant |
WO2008035023A1 (en) * | 2006-09-19 | 2008-03-27 | Cipla Limited | Polymorphs of rimonabant |
EP1944297A1 (en) * | 2007-01-09 | 2008-07-16 | Miklós Vértessy | Solid and crystalline rimonabant and processes for preparation, and pharmaceutical composition thereof |
EP1947090A1 (en) * | 2007-01-17 | 2008-07-23 | Laboratorios del Dr. Esteve S.A. | Method for preparing N-piperidino-1,5-diphenylpyrazole-3-carboxamide and derivatives |
WO2008088900A2 (en) * | 2007-01-18 | 2008-07-24 | Teva Pharmaceutical Industries Ltd. | Polymorphic forms of rimonabant base and processes for preparation thereof |
WO2008102367A1 (en) * | 2007-02-19 | 2008-08-28 | Darmesh Mahendrabhai Shah | Process for preparation of pyrazole derivatives |
FR2913018A1 (fr) * | 2007-02-23 | 2008-08-29 | Sanofi Aventis Sa | Solution solide amorphe contenant un derive de pyrazole-3-carboxamide sous forme amorphe et des excipients stabilisateurs |
WO2009109222A1 (en) * | 2008-03-04 | 2009-09-11 | Maprimed, S. A. | Process for the preparation of rimonabant |
WO2010079241A1 (es) | 2009-01-12 | 2010-07-15 | Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion | Uso de antagonistas y/o agonistas inversos de los receptores cb1 para la preparación de medicamentos que incrementen la excitabilidad de las motoneuronas |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2713225B1 (fr) * | 1993-12-02 | 1996-03-01 | Sanofi Sa | N-pipéridino-3-pyrazolecarboxamide substitué. |
FR2714057B1 (fr) * | 1993-12-17 | 1996-03-08 | Sanofi Elf | Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant. |
JP4314339B2 (ja) * | 2002-08-22 | 2009-08-12 | 三井化学アグロ株式会社 | ニコチンアミドラゾン誘導体 |
-
2004
- 2004-07-22 FR FR0408111A patent/FR2873372B1/fr not_active Expired - Fee Related
-
2005
- 2005-07-19 AR ARP050102971A patent/AR049995A1/es unknown
- 2005-07-19 UY UY29023A patent/UY29023A1/es not_active Application Discontinuation
- 2005-07-20 ZA ZA200609639A patent/ZA200609639B/xx unknown
- 2005-07-20 KR KR1020067024365A patent/KR20070036050A/ko not_active Application Discontinuation
- 2005-07-20 MX MXPA06012954A patent/MXPA06012954A/es not_active Application Discontinuation
- 2005-07-20 JP JP2007521985A patent/JP4879175B2/ja not_active Expired - Fee Related
- 2005-07-20 WO PCT/FR2005/001850 patent/WO2006021652A1/fr active Application Filing
- 2005-07-20 CN CNB2005800163474A patent/CN100537543C/zh not_active Expired - Fee Related
- 2005-07-20 EP EP05790868A patent/EP1773783B1/fr active Active
- 2005-07-20 BR BRPI0510399-1A patent/BRPI0510399A/pt not_active IP Right Cessation
- 2005-07-20 DE DE602005021110T patent/DE602005021110D1/de active Active
- 2005-07-20 AT AT05790868T patent/ATE466843T1/de not_active IP Right Cessation
- 2005-07-20 AU AU2005276350A patent/AU2005276350A1/en not_active Abandoned
- 2005-07-20 CA CA002564223A patent/CA2564223A1/fr not_active Abandoned
- 2005-07-20 RU RU2006141239/04A patent/RU2329252C1/ru not_active IP Right Cessation
- 2005-07-21 TW TW094124731A patent/TW200609223A/zh unknown
-
2006
- 2006-11-07 IL IL179107A patent/IL179107A0/en unknown
- 2006-11-10 MA MA29444A patent/MA28576B1/fr unknown
- 2006-11-14 US US11/559,566 patent/US7462632B2/en not_active Expired - Fee Related
-
2007
- 2007-02-21 NO NO20071008A patent/NO20071008L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP1773783A1 (fr) | 2007-04-18 |
CN1956963A (zh) | 2007-05-02 |
AR049995A1 (es) | 2006-09-20 |
JP4879175B2 (ja) | 2012-02-22 |
TW200609223A (en) | 2006-03-16 |
FR2873372B1 (fr) | 2006-09-08 |
MXPA06012954A (es) | 2007-02-12 |
WO2006021652A1 (fr) | 2006-03-02 |
RU2329252C1 (ru) | 2008-07-20 |
DE602005021110D1 (de) | 2010-06-17 |
MA28576B1 (fr) | 2007-05-02 |
CN100537543C (zh) | 2009-09-09 |
US20080119653A1 (en) | 2008-05-22 |
US7462632B2 (en) | 2008-12-09 |
EP1773783B1 (fr) | 2010-05-05 |
CA2564223A1 (fr) | 2006-03-02 |
AU2005276350A1 (en) | 2006-03-02 |
ZA200609639B (en) | 2008-08-27 |
FR2873372A1 (fr) | 2006-01-27 |
BRPI0510399A (pt) | 2007-11-13 |
JP2008506756A (ja) | 2008-03-06 |
IL179107A0 (en) | 2007-03-08 |
UY29023A1 (es) | 2006-02-24 |
ATE466843T1 (de) | 2010-05-15 |
KR20070036050A (ko) | 2007-04-02 |
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Legal Events
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FC2A | Withdrawal, rejection or dismissal of laid open patent application |