DE602005021110D1 - Verfahren zur herstellung von n-piperidino-1,5-diphenylpyrazol-3-carboxamid-derivaten - Google Patents
Verfahren zur herstellung von n-piperidino-1,5-diphenylpyrazol-3-carboxamid-derivatenInfo
- Publication number
- DE602005021110D1 DE602005021110D1 DE602005021110T DE602005021110T DE602005021110D1 DE 602005021110 D1 DE602005021110 D1 DE 602005021110D1 DE 602005021110 T DE602005021110 T DE 602005021110T DE 602005021110 T DE602005021110 T DE 602005021110T DE 602005021110 D1 DE602005021110 D1 DE 602005021110D1
- Authority
- DE
- Germany
- Prior art keywords
- diphenylpyrazole
- piperidino
- preparing
- carboxamide derivatives
- carboxamide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0408111A FR2873372B1 (fr) | 2004-07-22 | 2004-07-22 | Procede de preparation de derives n-piperidino-1,5- diphenylpyrazole-3-carboxamide |
| PCT/FR2005/001850 WO2006021652A1 (fr) | 2004-07-22 | 2005-07-20 | Procede de preparation de derives n-piperidino-1,5-diphenylpyrazole-3-carboxamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE602005021110D1 true DE602005021110D1 (de) | 2010-06-17 |
Family
ID=34949586
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE602005021110T Active DE602005021110D1 (de) | 2004-07-22 | 2005-07-20 | Verfahren zur herstellung von n-piperidino-1,5-diphenylpyrazol-3-carboxamid-derivaten |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US7462632B2 (de) |
| EP (1) | EP1773783B1 (de) |
| JP (1) | JP4879175B2 (de) |
| KR (1) | KR20070036050A (de) |
| CN (1) | CN100537543C (de) |
| AR (1) | AR049995A1 (de) |
| AT (1) | ATE466843T1 (de) |
| AU (1) | AU2005276350A1 (de) |
| BR (1) | BRPI0510399A (de) |
| CA (1) | CA2564223A1 (de) |
| DE (1) | DE602005021110D1 (de) |
| FR (1) | FR2873372B1 (de) |
| IL (1) | IL179107A0 (de) |
| MA (1) | MA28576B1 (de) |
| MX (1) | MXPA06012954A (de) |
| NO (1) | NO20071008L (de) |
| RU (1) | RU2329252C1 (de) |
| TW (1) | TW200609223A (de) |
| UY (1) | UY29023A1 (de) |
| WO (1) | WO2006021652A1 (de) |
| ZA (1) | ZA200609639B (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1816125A1 (de) * | 2006-02-02 | 2007-08-08 | Ranbaxy Laboratories, Ltd. | Kristalline Formen eines CB1-Cannabinoidrezeptorantagonisten und deren Herstellungsverfahren |
| US20100076022A1 (en) * | 2006-09-01 | 2010-03-25 | Hetero Drugs Limited | Novel polymorphs of rimonabant |
| EP2061783A2 (de) * | 2006-09-11 | 2009-05-27 | Hetero Drugs Limited | Verbessertes verfahren für rimonabant |
| WO2008035023A1 (en) * | 2006-09-19 | 2008-03-27 | Cipla Limited | Polymorphs of rimonabant |
| EP1944297A1 (de) * | 2007-01-09 | 2008-07-16 | Miklós Vértessy | Festes und kristallines Rimonabant, Herstellungsverfahren dafür und pharmazeutische Zusammensetzung davon |
| EP1947090A1 (de) * | 2007-01-17 | 2008-07-23 | Laboratorios del Dr. Esteve S.A. | Verfahren zur Herstellung von N-piperidino-1,5-diphenylpyrazol-3-carboxamid-Derivaten |
| WO2008088900A2 (en) * | 2007-01-18 | 2008-07-24 | Teva Pharmaceutical Industries Ltd. | Polymorphic forms of rimonabant base and processes for preparation thereof |
| WO2008102367A1 (en) * | 2007-02-19 | 2008-08-28 | Darmesh Mahendrabhai Shah | Process for preparation of pyrazole derivatives |
| FR2913018A1 (fr) * | 2007-02-23 | 2008-08-29 | Sanofi Aventis Sa | Solution solide amorphe contenant un derive de pyrazole-3-carboxamide sous forme amorphe et des excipients stabilisateurs |
| WO2009109222A1 (en) * | 2008-03-04 | 2009-09-11 | Maprimed, S. A. | Process for the preparation of rimonabant |
| WO2010079241A1 (es) | 2009-01-12 | 2010-07-15 | Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion | Uso de antagonistas y/o agonistas inversos de los receptores cb1 para la preparación de medicamentos que incrementen la excitabilidad de las motoneuronas |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2713225B1 (fr) * | 1993-12-02 | 1996-03-01 | Sanofi Sa | N-pipéridino-3-pyrazolecarboxamide substitué. |
| FR2714057B1 (fr) * | 1993-12-17 | 1996-03-08 | Sanofi Elf | Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant. |
| JP4314339B2 (ja) * | 2002-08-22 | 2009-08-12 | 三井化学アグロ株式会社 | ニコチンアミドラゾン誘導体 |
-
2004
- 2004-07-22 FR FR0408111A patent/FR2873372B1/fr not_active Expired - Fee Related
-
2005
- 2005-07-19 UY UY29023A patent/UY29023A1/es not_active Application Discontinuation
- 2005-07-19 AR ARP050102971A patent/AR049995A1/es unknown
- 2005-07-20 WO PCT/FR2005/001850 patent/WO2006021652A1/fr active Application Filing
- 2005-07-20 AT AT05790868T patent/ATE466843T1/de not_active IP Right Cessation
- 2005-07-20 DE DE602005021110T patent/DE602005021110D1/de active Active
- 2005-07-20 MX MXPA06012954A patent/MXPA06012954A/es not_active Application Discontinuation
- 2005-07-20 RU RU2006141239/04A patent/RU2329252C1/ru not_active IP Right Cessation
- 2005-07-20 BR BRPI0510399-1A patent/BRPI0510399A/pt not_active IP Right Cessation
- 2005-07-20 EP EP05790868A patent/EP1773783B1/de active Active
- 2005-07-20 JP JP2007521985A patent/JP4879175B2/ja not_active Expired - Fee Related
- 2005-07-20 ZA ZA200609639A patent/ZA200609639B/xx unknown
- 2005-07-20 AU AU2005276350A patent/AU2005276350A1/en not_active Abandoned
- 2005-07-20 CN CNB2005800163474A patent/CN100537543C/zh not_active Expired - Fee Related
- 2005-07-20 KR KR1020067024365A patent/KR20070036050A/ko not_active Application Discontinuation
- 2005-07-20 CA CA002564223A patent/CA2564223A1/fr not_active Abandoned
- 2005-07-21 TW TW094124731A patent/TW200609223A/zh unknown
-
2006
- 2006-11-07 IL IL179107A patent/IL179107A0/en unknown
- 2006-11-10 MA MA29444A patent/MA28576B1/fr unknown
- 2006-11-14 US US11/559,566 patent/US7462632B2/en not_active Expired - Fee Related
-
2007
- 2007-02-21 NO NO20071008A patent/NO20071008L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2008506756A (ja) | 2008-03-06 |
| US20080119653A1 (en) | 2008-05-22 |
| AU2005276350A1 (en) | 2006-03-02 |
| UY29023A1 (es) | 2006-02-24 |
| IL179107A0 (en) | 2007-03-08 |
| JP4879175B2 (ja) | 2012-02-22 |
| ATE466843T1 (de) | 2010-05-15 |
| FR2873372A1 (fr) | 2006-01-27 |
| FR2873372B1 (fr) | 2006-09-08 |
| EP1773783A1 (de) | 2007-04-18 |
| BRPI0510399A (pt) | 2007-11-13 |
| MA28576B1 (fr) | 2007-05-02 |
| RU2329252C1 (ru) | 2008-07-20 |
| CN100537543C (zh) | 2009-09-09 |
| ZA200609639B (en) | 2008-08-27 |
| NO20071008L (no) | 2007-02-21 |
| WO2006021652A1 (fr) | 2006-03-02 |
| US7462632B2 (en) | 2008-12-09 |
| MXPA06012954A (es) | 2007-02-12 |
| CN1956963A (zh) | 2007-05-02 |
| AR049995A1 (es) | 2006-09-20 |
| EP1773783B1 (de) | 2010-05-05 |
| KR20070036050A (ko) | 2007-04-02 |
| TW200609223A (en) | 2006-03-16 |
| CA2564223A1 (fr) | 2006-03-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |