NO20066016L - Diamin beta2 adrenergiske receptoragonister - Google Patents

Diamin beta2 adrenergiske receptoragonister

Info

Publication number
NO20066016L
NO20066016L NO20066016A NO20066016A NO20066016L NO 20066016 L NO20066016 L NO 20066016L NO 20066016 A NO20066016 A NO 20066016A NO 20066016 A NO20066016 A NO 20066016A NO 20066016 L NO20066016 L NO 20066016L
Authority
NO
Norway
Prior art keywords
adrenergic receptor
diamine
receptor agonists
beta2 adrenergic
compounds
Prior art date
Application number
NO20066016A
Other languages
English (en)
Norwegian (no)
Inventor
Martin S Linsell
Original Assignee
Theravance Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theravance Inc filed Critical Theravance Inc
Publication of NO20066016L publication Critical patent/NO20066016L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/24—Oxygen atoms attached in position 8
    • C07D215/26—Alcohols; Ethers thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Quinoline Compounds (AREA)
NO20066016A 2004-06-03 2006-12-27 Diamin beta2 adrenergiske receptoragonister NO20066016L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US57656004P 2004-06-03 2004-06-03
PCT/US2005/019549 WO2005121065A2 (en) 2004-06-03 2005-06-02 DIAMINE β2 ADRENERGIC RECEPTOR AGONISTS

Publications (1)

Publication Number Publication Date
NO20066016L true NO20066016L (no) 2007-02-27

Family

ID=35115813

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20066016A NO20066016L (no) 2004-06-03 2006-12-27 Diamin beta2 adrenergiske receptoragonister

Country Status (14)

Country Link
US (2) US20080039495A1 (xx)
EP (1) EP1751086A2 (xx)
JP (1) JP2008501705A (xx)
CN (1) CN1984876A (xx)
AU (1) AU2005252226A1 (xx)
BR (1) BRPI0511695A (xx)
CA (1) CA2569395A1 (xx)
IL (1) IL179631A0 (xx)
MA (1) MA28902B1 (xx)
MX (1) MXPA06013916A (xx)
NO (1) NO20066016L (xx)
RU (1) RU2006146042A (xx)
WO (1) WO2005121065A2 (xx)
ZA (1) ZA200610835B (xx)

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WO2008041914A1 (en) * 2006-10-06 2008-04-10 Astrazeneca Ab 5-(2-AMINO-L-HYDROXYETHYL)-8-HYDROXY-2-OXOQUINOLINE DERIVATIVES AND OTHER COMPOUNDS AS β2 -ADRENERGIC AGONISTS
ES2302447B1 (es) * 2006-10-20 2009-06-12 Laboratorios Almirall S.A. Derivados de 4-(2-amino-1-hidroxietil)fenol como agonistas del receptor beta2 adrenergico.
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SI2379507T1 (sl) 2008-12-30 2014-02-28 Pulmagen Therapeutics (Inflammation) Limited Spojine sulfonamida za zdravljenje respiratornih motenj
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WO2010150014A1 (en) 2009-06-24 2010-12-29 Pulmagen Therapeutics (Inflammation) Limited 5r- 5 -deuterated glitazones for respiratory disease treatment
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WO2011098746A1 (en) 2010-02-09 2011-08-18 Pulmagen Therapeutics (Inflammation) Limited Crystalline acid addition salts of ( 5r) -enanti0mer of pioglitazone
GB201002243D0 (en) 2010-02-10 2010-03-31 Argenta Therapeutics Ltd Respiratory disease treatment
GB201002224D0 (en) 2010-02-10 2010-03-31 Argenta Therapeutics Ltd Respiratory disease treatment
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
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EP2641900A1 (en) 2012-03-20 2013-09-25 Almirall, S.A. Novel polymorphic Crystal forms of 5-(2-{[6-(2,2-difluoro-2-phenylethoxy) hexyl]amino}-1-(R)-hydroxyethyl)-8-hydroxyquinolin-2(1h)-one, heminapadisylate as agonist of the ß2 adrenergic receptor.

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Also Published As

Publication number Publication date
MA28902B1 (fr) 2007-10-01
WO2005121065A3 (en) 2006-02-09
US20050272769A1 (en) 2005-12-08
EP1751086A2 (en) 2007-02-14
ZA200610835B (en) 2007-11-28
WO2005121065A2 (en) 2005-12-22
BRPI0511695A (pt) 2008-01-08
US20080039495A1 (en) 2008-02-14
MXPA06013916A (es) 2007-03-07
RU2006146042A (ru) 2008-07-20
IL179631A0 (en) 2007-05-15
US7402673B2 (en) 2008-07-22
AU2005252226A1 (en) 2005-12-22
JP2008501705A (ja) 2008-01-24
CN1984876A (zh) 2007-06-20
CA2569395A1 (en) 2005-12-22

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