NO20065889L - 3-`4-{6-substituert alkanoyl)pyridin-3-yf}-3-fenyl!-5-(1 H-1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midler. - Google Patents

3-`4-{6-substituert alkanoyl)pyridin-3-yf}-3-fenyl!-5-(1 H-1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midler.

Info

Publication number
NO20065889L
NO20065889L NO20065889A NO20065889A NO20065889L NO 20065889 L NO20065889 L NO 20065889L NO 20065889 A NO20065889 A NO 20065889A NO 20065889 A NO20065889 A NO 20065889A NO 20065889 L NO20065889 L NO 20065889L
Authority
NO
Norway
Prior art keywords
oner
oxazolidin
triazol
ylmethyl
pyridin
Prior art date
Application number
NO20065889A
Other languages
English (en)
Inventor
Michael Barry Gravenstock
Folkert Beck
Frei Zhou
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0411593A external-priority patent/GB0411593D0/en
Priority claimed from GB0500054A external-priority patent/GB0500054D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20065889L publication Critical patent/NO20065889L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Forbindelser med formel I samt farmasøytisk akseptable salter og prodrugs derav er beskrevet, hvor R1, R2, R3 og R4 er som definert heri. Det er også beskrevet fremgangsmåter for fremstilling av forbindelser med formel I samt fremgangsmåter for anvendelse av forbindelser med formel I for behandling av bakterielle infeksjoner.
NO20065889A 2004-05-25 2006-12-19 3-`4-{6-substituert alkanoyl)pyridin-3-yf}-3-fenyl!-5-(1 H-1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midler. NO20065889L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0411593A GB0411593D0 (en) 2004-05-25 2004-05-25 Chemical compounds
GB0500054A GB0500054D0 (en) 2005-01-05 2005-01-05 Chemical compounds
PCT/GB2005/002051 WO2005116022A1 (en) 2004-05-25 2005-05-24 3- `4- {6-substituted alkanoyl) pyridin-3-yl} -3-phenyl! -5- (1h-1, 2, 3-triazol-1-ylmethyl) -1, 3-oxazolidin-2-ones as antibacterial agents

Publications (1)

Publication Number Publication Date
NO20065889L true NO20065889L (no) 2007-02-20

Family

ID=34968778

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20065889A NO20065889L (no) 2004-05-25 2006-12-19 3-`4-{6-substituert alkanoyl)pyridin-3-yf}-3-fenyl!-5-(1 H-1,2,3-triazol-1-ylmetyl)-1,3-oksazolidin-2-oner som antibakterielle midler.

Country Status (10)

Country Link
US (1) US20080021012A1 (no)
EP (1) EP1753754A1 (no)
JP (1) JP2008500317A (no)
AU (1) AU2005247668A1 (no)
BR (1) BRPI0511526A (no)
CA (1) CA2566963A1 (no)
IL (1) IL179349A0 (no)
MX (1) MXPA06013537A (no)
NO (1) NO20065889L (no)
WO (1) WO2005116022A1 (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100854211B1 (ko) 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
WO2010042887A2 (en) 2008-10-10 2010-04-15 Trius Therapeutics Methods for preparing oxazolidinones and compositions containing them
PE20120585A1 (es) 2009-02-03 2012-06-13 Trius Therapeutics Forma cristalina del fosfato de dihidrogeno r)-3-(4-(2-(2-metiltetrazol-5-il) piridin-5-il)-3-fluorofensil)-5-hidroximetil oxazolidin-2-ona
US8580767B2 (en) * 2009-05-28 2013-11-12 Trius Therapeutics, Inc. Oxazolidinone containing dimer compounds, compositions and methods to make and use
KR101561964B1 (ko) 2013-11-15 2015-10-20 한국과학기술연구원 옥사졸리디논 화합물 및 이를 포함하는 c형 간염 예방 또는 치료용 약학 조성물
EP3436434B1 (en) 2016-03-31 2020-07-08 Oncternal Therapeutics, Inc. Indoline analogs and uses thereof
AU2021292747A1 (en) 2020-06-18 2023-02-23 Akagera Medicines, Inc. Oxazolidinone compounds, liposome compositions comprising oxazolidinone compounds and methods of use thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0009803D0 (en) * 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
HUP0301562A2 (hu) * 2000-06-05 2003-12-29 Dong A Pharm. Co., Ltd. Új oxazolidinonszármazékok és eljárás ezek előállítására, ezeket tartalmazó gyógyszerkészítmények
KR20040087329A (ko) * 2002-02-28 2004-10-13 아스트라제네카 아베 3-시클릴-5-(질소-함유 5-원 고리) 메틸-옥사졸리디논유도체 및 그의 항균제로서의 용도

Also Published As

Publication number Publication date
BRPI0511526A (pt) 2007-12-26
IL179349A0 (en) 2007-03-08
AU2005247668A1 (en) 2005-12-08
CA2566963A1 (en) 2005-12-08
US20080021012A1 (en) 2008-01-24
EP1753754A1 (en) 2007-02-21
JP2008500317A (ja) 2008-01-10
WO2005116022A1 (en) 2005-12-08
MXPA06013537A (es) 2007-01-26

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