NO20062661L - Beta-laktamer for behandling av CNS lidelser - Google Patents

Beta-laktamer for behandling av CNS lidelser

Info

Publication number
NO20062661L
NO20062661L NO20062661A NO20062661A NO20062661L NO 20062661 L NO20062661 L NO 20062661L NO 20062661 A NO20062661 A NO 20062661A NO 20062661 A NO20062661 A NO 20062661A NO 20062661 L NO20062661 L NO 20062661L
Authority
NO
Norway
Prior art keywords
cyano
hydroxy
halogen
alkyl
represents hydrogen
Prior art date
Application number
NO20062661A
Other languages
English (en)
Norwegian (no)
Inventor
Romano Di Fabio
Giuseppe Alvaro
Riccardo Giovannini
Maria Elvira Tranquillini
Alfredo Paio
Lucia Mattio
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20062661L publication Critical patent/NO20062661L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Addiction (AREA)
  • Anesthesiology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
NO20062661A 2003-11-12 2006-06-09 Beta-laktamer for behandling av CNS lidelser NO20062661L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0326407.4A GB0326407D0 (en) 2003-11-12 2003-11-12 Chemical compounds
PCT/EP2004/012772 WO2005049600A1 (en) 2003-11-12 2004-11-10 Beta-lactams for treatment of cns disorders

Publications (1)

Publication Number Publication Date
NO20062661L true NO20062661L (no) 2006-06-09

Family

ID=29726427

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20062661A NO20062661L (no) 2003-11-12 2006-06-09 Beta-laktamer for behandling av CNS lidelser

Country Status (28)

Country Link
US (1) US20080262041A1 (ru)
EP (1) EP1689737B1 (ru)
JP (1) JP2007510692A (ru)
KR (1) KR20060118477A (ru)
CN (1) CN1878764A (ru)
AR (1) AR046233A1 (ru)
AT (1) ATE401321T1 (ru)
AU (1) AU2004291296B2 (ru)
BR (1) BRPI0416285A (ru)
CA (1) CA2546007A1 (ru)
CY (1) CY1108404T1 (ru)
DE (1) DE602004015144D1 (ru)
DK (1) DK1689737T3 (ru)
ES (1) ES2310295T3 (ru)
GB (1) GB0326407D0 (ru)
HK (1) HK1094698A1 (ru)
HR (1) HRP20080501T3 (ru)
IL (1) IL175279A0 (ru)
IS (1) IS8477A (ru)
MA (1) MA28156A1 (ru)
MY (1) MY138378A (ru)
NO (1) NO20062661L (ru)
PL (1) PL1689737T3 (ru)
PT (1) PT1689737E (ru)
RU (1) RU2006120417A (ru)
SI (1) SI1689737T1 (ru)
TW (1) TW200528439A (ru)
WO (1) WO2005049600A1 (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101410372A (zh) 2006-01-24 2009-04-15 拜欧希格诺有限公司 新内酰胺类
AU2015200142B2 (en) * 2006-01-24 2016-07-07 Unilever Plc Novel lactams

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL262366A (ru) * 1960-03-14
FR2676055B1 (fr) * 1991-05-03 1993-09-03 Sanofi Elf Composes polycycliques amines et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant.
CA2083891A1 (en) * 1991-12-03 1993-06-04 Angus Murray Macleod Heterocyclic compounds, compositions containing them and their use in therapy
GB9200535D0 (en) * 1992-01-10 1992-02-26 Fujisawa Pharmaceutical Co New compound
US5824690A (en) * 1993-05-06 1998-10-20 Hoechst Marion Roussel Inc. Substituted pyrrolidin-3-yl-alkyl-piperidines
GB9317104D0 (en) * 1993-08-17 1993-09-29 Zeneca Ltd Therapeutic heterocycles
GB9322643D0 (en) * 1993-11-03 1993-12-22 Zeneca Ltd Lactam derivatives
ATE177095T1 (de) * 1994-08-25 1999-03-15 Merrell Pharma Inc Substituierte piperidine für die behandlung von allergischen krankheiten
US5780466A (en) * 1995-01-30 1998-07-14 Sanofi Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present
TW332201B (en) * 1995-04-06 1998-05-21 Janssen Pharmaceutica Nv 1,3-Dihydro-1-(phenylalkyl)-2H-imidazol-2-one derivatives
US6211199B1 (en) * 1995-11-17 2001-04-03 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases
FR2779429B1 (fr) * 1998-06-03 2000-07-13 Synthelabo Derives d'oxindole, leurs preparations et leurs applications en therapeutique
US6204265B1 (en) * 1998-12-23 2001-03-20 Schering Corporation Substituted oximes and hydrazones as neurokinin antagonists
GB0114867D0 (en) * 2001-06-18 2001-08-08 Merck Sharp & Dohme Therapeutic agents
GB0412865D0 (en) * 2004-06-09 2004-07-14 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
CA2546007A1 (en) 2005-06-02
DE602004015144D1 (de) 2008-08-28
BRPI0416285A (pt) 2007-01-23
AU2004291296A1 (en) 2005-06-02
JP2007510692A (ja) 2007-04-26
KR20060118477A (ko) 2006-11-23
AR046233A1 (es) 2005-11-30
HK1094698A1 (en) 2007-04-04
GB0326407D0 (en) 2003-12-17
AU2004291296B2 (en) 2011-04-07
MY138378A (en) 2009-05-29
EP1689737B1 (en) 2008-07-16
SI1689737T1 (sl) 2008-12-31
IS8477A (is) 2006-05-22
TW200528439A (en) 2005-09-01
IL175279A0 (en) 2006-09-05
ATE401321T1 (de) 2008-08-15
CN1878764A (zh) 2006-12-13
CY1108404T1 (el) 2014-02-12
PT1689737E (pt) 2008-10-24
EP1689737A1 (en) 2006-08-16
DK1689737T3 (da) 2008-10-27
ES2310295T3 (es) 2009-01-01
WO2005049600A1 (en) 2005-06-02
HRP20080501T3 (en) 2008-11-30
RU2006120417A (ru) 2007-12-27
US20080262041A1 (en) 2008-10-23
PL1689737T3 (pl) 2008-12-31
MA28156A1 (fr) 2006-09-01

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