NO20060910L - Piperidinforbindelser og farmasoytiske sammensetninger som inneholder dem - Google Patents

Piperidinforbindelser og farmasoytiske sammensetninger som inneholder dem

Info

Publication number
NO20060910L
NO20060910L NO20060910A NO20060910A NO20060910L NO 20060910 L NO20060910 L NO 20060910L NO 20060910 A NO20060910 A NO 20060910A NO 20060910 A NO20060910 A NO 20060910A NO 20060910 L NO20060910 L NO 20060910L
Authority
NO
Norway
Prior art keywords
piperidine compound
animal
disclosed
piperidine compounds
piperidine
Prior art date
Application number
NO20060910A
Other languages
English (en)
Norwegian (no)
Inventor
Qun Sun
Xiaoming Zhou
Xin Wen
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Publication of NO20060910L publication Critical patent/NO20060910L/no

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P25/32Alcohol-abuse
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
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    • AHUMAN NECESSITIES
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    • AHUMAN NECESSITIES
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    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Psychology (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Transplantation (AREA)
NO20060910A 2003-07-24 2006-02-24 Piperidinforbindelser og farmasoytiske sammensetninger som inneholder dem NO20060910L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48951503P 2003-07-24 2003-07-24
PCT/US2004/023912 WO2005009987A1 (fr) 2003-07-24 2004-07-23 Composes de piperidine et compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
NO20060910L true NO20060910L (no) 2006-04-04

Family

ID=34102892

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20060910A NO20060910L (no) 2003-07-24 2006-02-24 Piperidinforbindelser og farmasoytiske sammensetninger som inneholder dem

Country Status (29)

Country Link
US (2) US7572812B2 (fr)
EP (2) EP1648878B9 (fr)
JP (1) JP4686456B2 (fr)
KR (2) KR100977242B1 (fr)
CN (2) CN101914088A (fr)
AT (1) ATE430741T1 (fr)
AU (1) AU2004259357B2 (fr)
BR (1) BRPI0412808A (fr)
CA (1) CA2533509C (fr)
CY (1) CY1109273T1 (fr)
DE (1) DE602004020994D1 (fr)
DK (1) DK1648878T3 (fr)
EA (1) EA010852B1 (fr)
ES (1) ES2326979T3 (fr)
GE (1) GEP20094676B (fr)
HK (1) HK1089755A1 (fr)
HR (1) HRP20090404T1 (fr)
IL (3) IL173343A (fr)
IS (1) IS2684B (fr)
MA (1) MA27983A1 (fr)
MX (1) MXPA06000941A (fr)
NO (1) NO20060910L (fr)
NZ (1) NZ545506A (fr)
PL (1) PL1648878T3 (fr)
PT (1) PT1648878E (fr)
SI (1) SI1648878T1 (fr)
UA (1) UA84710C2 (fr)
WO (1) WO2005009987A1 (fr)
ZA (1) ZA200509562B (fr)

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KR100777169B1 (ko) 2001-01-29 2007-11-16 시오노기세이야쿠가부시키가이샤 5-메틸-1-페닐-2-(1h)-피리돈을 활성 성분으로서함유하는 의약 제제
US7157462B2 (en) * 2002-09-24 2007-01-02 Euro-Celtique S.A. Therapeutic agents useful for treating pain
MY142655A (en) * 2003-06-12 2010-12-15 Euro Celtique Sa Therapeutic agents useful for treating pain
DK1867644T3 (da) 2003-07-24 2009-09-21 Euro Celtique Sa Heteroaryl-tetrahydropyridyl-forbindelser, der er anvendelige til behandling eller forebyggelse af smerte
JP2008516973A (ja) 2004-10-15 2008-05-22 タケダ サン ディエゴ インコーポレイテッド キナーゼ阻害剤
WO2006124753A2 (fr) * 2005-05-12 2006-11-23 Amgen Inc. Traitement avec un agent antipyretique, de l'elevation de la temperature corporelle induite par l'antagoniste vr1
DE102005023943A1 (de) 2005-05-20 2006-11-23 Grünenthal GmbH Pentafluorsulfanyl-substituierte Verbindung und deren Verwendung zur Herstellung von Arzneimitteln
US8119655B2 (en) 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors
US20100120717A1 (en) 2006-10-09 2010-05-13 Brown Jason W Kinase inhibitors
MY148657A (en) * 2007-04-27 2013-05-15 Purdue Pharma Lp Trpv1 antagonists and uses thereof
AU2011226773C1 (en) * 2007-04-27 2012-07-26 Purdue Pharma L.P. TRPV1 antagonists and uses thereof
NZ579820A (en) 2007-04-27 2011-01-28 Purdue Pharma Lp Therapeutic agents useful for treating pain
US8084616B2 (en) 2007-10-24 2011-12-27 Abbott Laboratories TRPV1 antagonists
US11969501B2 (en) 2008-04-21 2024-04-30 Dompé Farmaceutici S.P.A. Auris formulations for treating otic diseases and conditions
US9132087B2 (en) 2008-04-21 2015-09-15 Otonomy, Inc. Auris formulations for treating otic diseases and conditions
CN102105133B (zh) 2008-07-21 2015-06-17 奥德纳米有限公司 控制释放型耳结构调节和先天性免疫系统调节组合物以及治疗耳部病症的方法
US8759362B2 (en) * 2008-10-24 2014-06-24 Purdue Pharma L.P. Bicycloheteroaryl compounds and their use as TRPV1 ligands
US8703962B2 (en) * 2008-10-24 2014-04-22 Purdue Pharma L.P. Monocyclic compounds and their use as TRPV1 ligands
WO2010064597A1 (fr) * 2008-12-01 2010-06-10 武田薬品工業株式会社 Dérivé de pipéridine
CN102098080B (zh) * 2009-12-09 2014-07-02 京信通信系统(中国)有限公司 数字微波射频拉远覆盖系统及方法
JP2013514379A (ja) * 2009-12-15 2013-04-25 ニユーロツプ・インコーポレイテツド 神経障害の治療のための化合物
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US20100210686A1 (en) 2010-08-19
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IL204884A (en) 2011-10-31
ATE430741T1 (de) 2009-05-15
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PT1648878E (pt) 2009-07-23
EP1648878B1 (fr) 2009-05-06
EA010852B1 (ru) 2008-12-30
MXPA06000941A (es) 2006-03-30
MA27983A1 (fr) 2006-07-03
BRPI0412808A (pt) 2006-09-26
GEP20094676B (en) 2009-05-10
CN1829708A (zh) 2006-09-06
ZA200509562B (en) 2006-08-30
JP2006528642A (ja) 2006-12-21
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IL173343A0 (en) 2006-06-11
KR100977242B1 (ko) 2010-08-24
AU2004259357B2 (en) 2010-02-18
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US7572812B2 (en) 2009-08-11
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US8349842B2 (en) 2013-01-08
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