NO171067C - Analogifremgangsmaate for fremstilling av terapeutisk aktive 4,5-dihydro- og 4,5,6,7-tetrahydro-pyrazolo (1,5-a)pyrimidiner - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive 4,5-dihydro- og 4,5,6,7-tetrahydro-pyrazolo (1,5-a)pyrimidiner

Info

Publication number
NO171067C
NO171067C NO874302A NO874302A NO171067C NO 171067 C NO171067 C NO 171067C NO 874302 A NO874302 A NO 874302A NO 874302 A NO874302 A NO 874302A NO 171067 C NO171067 C NO 171067C
Authority
NO
Norway
Prior art keywords
pyrazolo
pyrimidines
tetrahydro
dihydro
preparation
Prior art date
Application number
NO874302A
Other languages
English (en)
Norwegian (no)
Other versions
NO171067B (no
NO874302L (no
NO874302D0 (no
Inventor
Shin Shyong Tseng
John Paul Dusza
Joseph William Epstein
Herbert Joseph Brabander
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/919,730 external-priority patent/US4847256A/en
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of NO874302D0 publication Critical patent/NO874302D0/no
Publication of NO874302L publication Critical patent/NO874302L/no
Priority to NO903284A priority Critical patent/NO171213C/no
Publication of NO171067B publication Critical patent/NO171067B/no
Publication of NO171067C publication Critical patent/NO171067C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO874302A 1986-10-16 1987-10-15 Analogifremgangsmaate for fremstilling av terapeutisk aktive 4,5-dihydro- og 4,5,6,7-tetrahydro-pyrazolo (1,5-a)pyrimidiner NO171067C (no)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NO903284A NO171213C (no) 1986-10-16 1990-07-24 Pyrazolo(1,5-a)pyrimidiner, saerlig egnet for anvendelse som mellomprodukt

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US91973186A 1986-10-16 1986-10-16
US06/919,730 US4847256A (en) 1986-10-16 1986-10-16 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines

Publications (4)

Publication Number Publication Date
NO874302D0 NO874302D0 (no) 1987-10-15
NO874302L NO874302L (no) 1988-04-18
NO171067B NO171067B (no) 1992-10-12
NO171067C true NO171067C (no) 1993-01-20

Family

ID=27129779

Family Applications (1)

Application Number Title Priority Date Filing Date
NO874302A NO171067C (no) 1986-10-16 1987-10-15 Analogifremgangsmaate for fremstilling av terapeutisk aktive 4,5-dihydro- og 4,5,6,7-tetrahydro-pyrazolo (1,5-a)pyrimidiner

Country Status (10)

Country Link
EP (1) EP0264773A1 (de)
KR (1) KR880005132A (de)
AU (1) AU601498B2 (de)
DK (1) DK539087A (de)
FI (1) FI87459C (de)
HU (1) HU203103B (de)
IL (1) IL84214A (de)
NO (1) NO171067C (de)
NZ (1) NZ222179A (de)
PT (1) PT85936B (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4963553A (en) * 1986-10-16 1990-10-16 American Cyanamid Co. 4-[(substituted) alkylcarbonyl]-4,5-dihydro- and -4,5,6,7-tetrahydro-7-[(substituted)phenyl]pyrazolo[1,5-a]pyrimidines
US5126340A (en) * 1986-10-16 1992-06-30 American Cyanamid Company 4-[(substituted)alkylcarbonyl]-4,5-dihydro and -4,5,6,7-tetrahydro-7-[(substituted)-phenyl]pyrazolo[1,5-a]pyrimidine-3-carbonitriles
US5219857A (en) * 1986-10-16 1993-06-15 American Cyanamid Company Method of treating cognitive and related neural behavioral problems
DE68911951T2 (de) * 1988-02-22 1994-06-01 American Cyanamid Co 5-(Substituierte Amino)-8-(phenyl oder substituierte phenyl)-3H,6H-1,4,5a,8a-tetraazaacenaphthylen-3-one.
US4963552A (en) * 1989-08-28 1990-10-16 American Cyanamid Company 1-substitute-1,2-dihydro-4-((substituted)phenyl)imidazo-[1,5-a]pyrimidine-8-carbonitriles
DE4133957A1 (de) * 1991-10-14 1993-04-15 Wella Ag Haarfaerbemittel mit einem gehalt an aminopyrazolderivaten sowie neue pyrazolderivate
SG47588A1 (en) * 1992-03-26 1998-04-17 American Cyanamid Co An improved process for the synthesis of 5-[(substituted) amino] -8- [phenyl or substituted-phenyl]-3H, 6H-1, 4, 5A, 8A-tetraazaacenaphtylen-3- ones
GB0016787D0 (en) 2000-07-07 2000-08-30 Pfizer Ltd Compounds useful in therapy
DE10153344A1 (de) * 2001-10-29 2003-05-15 Gruenenthal Gmbh Verwendung von substituierten Pyrazolopyrimidinen als Liganden von Nucleosid-Transport-Proteinen und/oder von Purinorezeptoren
BR0208244A (pt) 2001-03-14 2004-03-02 Gr Nenthal Gmbh Pirazolo-e tiazolopirinidinas substituìdas
ES2222813B1 (es) * 2003-07-24 2005-12-16 Ferrer Internacional, S.A. N-(3-(3-sustituidas-pirazolo(1,5-a)pirimidin-7-il)-fenil)-sulfonamidas y composiciones y metodos relacionados.
TWI252851B (en) * 2003-07-24 2006-04-11 Ferrer Int 7-substituted 3-nitro-pyrazolo[1,5-a]pyrimidines and compositions and methods related thereto
WO2006033795A2 (en) * 2004-09-17 2006-03-30 Wyeth Substituted pyrazolo [1, 5-a] pyrimidines for inhibiting abnormal cell growth
WO2006033796A1 (en) * 2004-09-17 2006-03-30 Wyeth SUBSTITUTED PYRAZOLO [1,5-a] PYRIMIDINES AND PROCESS FOR MAKING SAME

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4236005A (en) * 1979-07-02 1980-11-25 American Cyanamid Company Imidazo[1,5-a]pyrimidines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents
US4521422A (en) * 1983-06-23 1985-06-04 American Cyanamid Company Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones
NZ208554A (en) * 1983-06-23 1987-06-30 American Cyanamid Co (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions

Also Published As

Publication number Publication date
DK539087D0 (da) 1987-10-15
IL84214A (en) 1993-05-13
AU601498B2 (en) 1990-09-13
HUT47276A (en) 1989-02-28
EP0264773A1 (de) 1988-04-27
IL84214A0 (en) 1988-03-31
NO171067B (no) 1992-10-12
FI87459C (fi) 1993-01-11
PT85936B (pt) 1990-07-31
KR880005132A (ko) 1988-06-28
FI874547A0 (fi) 1987-10-15
DK539087A (da) 1988-04-17
NO874302L (no) 1988-04-18
HU203103B (en) 1991-05-28
PT85936A (en) 1987-11-01
NZ222179A (en) 1991-01-29
NO874302D0 (no) 1987-10-15
FI874547A (fi) 1988-04-17
FI87459B (fi) 1992-09-30
AU7980087A (en) 1988-04-21

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