FI874547A0 - 4,5-dihydro och 4,5,6,7 -tetrahydropyrazolo (1,5-a) pyrimidiner. - Google Patents

4,5-dihydro och 4,5,6,7 -tetrahydropyrazolo (1,5-a) pyrimidiner.

Info

Publication number
FI874547A0
FI874547A0 FI874547A FI874547A FI874547A0 FI 874547 A0 FI874547 A0 FI 874547A0 FI 874547 A FI874547 A FI 874547A FI 874547 A FI874547 A FI 874547A FI 874547 A0 FI874547 A0 FI 874547A0
Authority
FI
Finland
Prior art keywords
pyrimidiner
tetrahydropyrazolo
och
dihydro
dihydro och
Prior art date
Application number
FI874547A
Other languages
English (en)
Other versions
FI874547A (fi
FI87459B (fi
FI87459C (fi
Inventor
Shin Shyong Tseng
John Paul Dusza
Joseph William Epstein
Herbert Joseph Brabander
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/919,730 external-priority patent/US4847256A/en
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of FI874547A0 publication Critical patent/FI874547A0/fi
Publication of FI874547A publication Critical patent/FI874547A/fi
Priority to FI904198A priority Critical patent/FI89487C/fi
Publication of FI87459B publication Critical patent/FI87459B/fi
Application granted granted Critical
Publication of FI87459C publication Critical patent/FI87459C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI874547A 1986-10-16 1987-10-15 Foerfarande foer framstaellning av terapeutiskt anvaendbara 4,5-dihydro- och 4,5,6,7-tetrahydropyratzolo/1,5-a/pyrimidinderivater FI87459C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI904198A FI89487C (fi) 1986-10-16 1990-08-24 Foerfarande foer framstaellning av terapeutiskt aktiva 4-/(substituerad)alkylkarbonyl/-4,5-dihydro- och -4,5,6,7-tetrahydro-7-/(substituerad)fenyl/pyrazolo-/1,5-a/pyrimidin-3-karbonitriler

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US91973186A 1986-10-16 1986-10-16
US06/919,730 US4847256A (en) 1986-10-16 1986-10-16 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines
US91973186 1986-10-16
US91973086 1986-10-16

Publications (4)

Publication Number Publication Date
FI874547A0 true FI874547A0 (fi) 1987-10-15
FI874547A FI874547A (fi) 1988-04-17
FI87459B FI87459B (fi) 1992-09-30
FI87459C FI87459C (fi) 1993-01-11

Family

ID=27129779

Family Applications (1)

Application Number Title Priority Date Filing Date
FI874547A FI87459C (fi) 1986-10-16 1987-10-15 Foerfarande foer framstaellning av terapeutiskt anvaendbara 4,5-dihydro- och 4,5,6,7-tetrahydropyratzolo/1,5-a/pyrimidinderivater

Country Status (10)

Country Link
EP (1) EP0264773A1 (fi)
KR (1) KR880005132A (fi)
AU (1) AU601498B2 (fi)
DK (1) DK539087A (fi)
FI (1) FI87459C (fi)
HU (1) HU203103B (fi)
IL (1) IL84214A (fi)
NO (1) NO171067C (fi)
NZ (1) NZ222179A (fi)
PT (1) PT85936B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5126340A (en) * 1986-10-16 1992-06-30 American Cyanamid Company 4-[(substituted)alkylcarbonyl]-4,5-dihydro and -4,5,6,7-tetrahydro-7-[(substituted)-phenyl]pyrazolo[1,5-a]pyrimidine-3-carbonitriles
US5219857A (en) * 1986-10-16 1993-06-15 American Cyanamid Company Method of treating cognitive and related neural behavioral problems
US4963553A (en) * 1986-10-16 1990-10-16 American Cyanamid Co. 4-[(substituted) alkylcarbonyl]-4,5-dihydro- and -4,5,6,7-tetrahydro-7-[(substituted)phenyl]pyrazolo[1,5-a]pyrimidines
EP0329940B1 (en) * 1988-02-22 1994-01-05 American Cyanamid Company 5-(substituted)amino)-8- (phenyl or substituted phenyl)-3H,6H-1,2,5,a,8 a-tetraazaacenaphthylen-3-ones
US4963552A (en) * 1989-08-28 1990-10-16 American Cyanamid Company 1-substitute-1,2-dihydro-4-((substituted)phenyl)imidazo-[1,5-a]pyrimidine-8-carbonitriles
DE4133957A1 (de) * 1991-10-14 1993-04-15 Wella Ag Haarfaerbemittel mit einem gehalt an aminopyrazolderivaten sowie neue pyrazolderivate
EP0562236A1 (en) * 1992-03-26 1993-09-29 American Cyanamid Company Process for the synthesis of 5-[(substituted)-amino]-8-[phenyl or substiutued-phenyl]-3H, 6H-1, 4, 5A, 8A-tetraazaacephthylen-3-ones
GB0016787D0 (en) 2000-07-07 2000-08-30 Pfizer Ltd Compounds useful in therapy
DE10153344A1 (de) * 2001-10-29 2003-05-15 Gruenenthal Gmbh Verwendung von substituierten Pyrazolopyrimidinen als Liganden von Nucleosid-Transport-Proteinen und/oder von Purinorezeptoren
EP1368355B1 (de) 2001-03-14 2006-06-07 Grünenthal GmbH Substituierte pyrazolo- und thiazolopyrimidine als analgetika
ES2222813B1 (es) * 2003-07-24 2005-12-16 Ferrer Internacional, S.A. N-(3-(3-sustituidas-pirazolo(1,5-a)pirimidin-7-il)-fenil)-sulfonamidas y composiciones y metodos relacionados.
TWI252851B (en) * 2003-07-24 2006-04-11 Ferrer Int 7-substituted 3-nitro-pyrazolo[1,5-a]pyrimidines and compositions and methods related thereto
WO2006033795A2 (en) * 2004-09-17 2006-03-30 Wyeth Substituted pyrazolo [1, 5-a] pyrimidines for inhibiting abnormal cell growth
WO2006033796A1 (en) * 2004-09-17 2006-03-30 Wyeth SUBSTITUTED PYRAZOLO [1,5-a] PYRIMIDINES AND PROCESS FOR MAKING SAME

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4236005A (en) * 1979-07-02 1980-11-25 American Cyanamid Company Imidazo[1,5-a]pyrimidines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents
US4521422A (en) * 1983-06-23 1985-06-04 American Cyanamid Company Aryl and heteroaryl[7-(aryl and heteroaryl)pyrazolo[1,5-a]pyrimidin-3-yl]methanones
NZ208554A (en) * 1983-06-23 1987-06-30 American Cyanamid Co (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions

Also Published As

Publication number Publication date
DK539087D0 (da) 1987-10-15
AU7980087A (en) 1988-04-21
DK539087A (da) 1988-04-17
AU601498B2 (en) 1990-09-13
NZ222179A (en) 1991-01-29
NO874302D0 (no) 1987-10-15
NO171067B (no) 1992-10-12
KR880005132A (ko) 1988-06-28
FI874547A (fi) 1988-04-17
HU203103B (en) 1991-05-28
FI87459B (fi) 1992-09-30
PT85936A (en) 1987-11-01
FI87459C (fi) 1993-01-11
HUT47276A (en) 1989-02-28
PT85936B (pt) 1990-07-31
NO874302L (no) 1988-04-18
EP0264773A1 (en) 1988-04-27
IL84214A0 (en) 1988-03-31
IL84214A (en) 1993-05-13
NO171067C (no) 1993-01-20

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Legal Events

Date Code Title Description
MM Patent lapsed
MM Patent lapsed

Owner name: AMERICAN CYANAMID COMPANY