NO143577C - 2-fenyl-imidazo-isokinolin-derivater med svangerskapsavbrytende virkning - Google Patents

2-fenyl-imidazo-isokinolin-derivater med svangerskapsavbrytende virkning

Info

Publication number
NO143577C
NO143577C NO753853A NO753853A NO143577C NO 143577 C NO143577 C NO 143577C NO 753853 A NO753853 A NO 753853A NO 753853 A NO753853 A NO 753853A NO 143577 C NO143577 C NO 143577C
Authority
NO
Norway
Prior art keywords
isokinoline
imidazo
pregnancy
phenyl
derivatives
Prior art date
Application number
NO753853A
Other languages
English (en)
Norwegian (no)
Other versions
NO143577B (no
NO753853L (de
Inventor
Amedeo Omodei-Sale
Emilio Toia
Giulio Galliani
Leonard J Lerner
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of NO753853L publication Critical patent/NO753853L/no
Publication of NO143577B publication Critical patent/NO143577B/no
Publication of NO143577C publication Critical patent/NO143577C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
NO753853A 1974-11-23 1975-11-17 2-fenyl-imidazo-isokinolin-derivater med svangerskapsavbrytende virkning NO143577C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB50855/74A GB1484615A (en) 1974-11-23 1974-11-23 Tricyclic n-containing derivatives

Publications (3)

Publication Number Publication Date
NO753853L NO753853L (de) 1976-05-25
NO143577B NO143577B (no) 1980-12-01
NO143577C true NO143577C (no) 1981-03-11

Family

ID=10457662

Family Applications (2)

Application Number Title Priority Date Filing Date
NO753854A NO143578C (no) 1974-11-23 1975-11-17 2-fenylpyrazol-isokinolinderivater med svangerskapsavbrytende virkning.
NO753853A NO143577C (no) 1974-11-23 1975-11-17 2-fenyl-imidazo-isokinolin-derivater med svangerskapsavbrytende virkning

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO753854A NO143578C (no) 1974-11-23 1975-11-17 2-fenylpyrazol-isokinolinderivater med svangerskapsavbrytende virkning.

Country Status (25)

Country Link
US (1) US4075342A (de)
JP (1) JPS5516513B2 (de)
AR (2) AR210476A1 (de)
AT (2) AT344176B (de)
BE (1) BE835836A (de)
CA (2) CA1068274A (de)
CH (2) CH614444A5 (de)
DD (2) DD122818A5 (de)
DE (1) DE2551868C2 (de)
DK (2) DK152756C (de)
ES (2) ES442864A1 (de)
FI (2) FI58919C (de)
FR (1) FR2291747A1 (de)
GB (1) GB1484615A (de)
GR (2) GR58293B (de)
IE (1) IE43567B1 (de)
IL (1) IL48389A (de)
IN (2) IN142014B (de)
LU (2) LU73849A1 (de)
NL (1) NL165741C (de)
NO (2) NO143578C (de)
SE (2) SE421619B (de)
SU (3) SU569290A3 (de)
YU (1) YU37328B (de)
ZA (1) ZA756792B (de)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4075343A (en) * 1976-09-13 1978-02-21 Pfizer Inc. Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof
US4313950A (en) * 1978-10-30 1982-02-02 Gruppo Lepetit S.P.A. Antireproductive tricyclic ortho-fused nitrogen containing compounds
GR70248B (de) * 1978-10-30 1982-09-01 Lepetit Spa
EP0012866B1 (de) * 1978-12-21 1983-01-19 Gruppo Lepetit S.P.A. 3H-Naphtho(1,2-d)imidazole, Verfahren zu deren Herstellung, Verbindungen zur Verwendung als entzündungshemmende und antimikrobielle Mittel und sie enthaltende Zusammensetzungen zu dieser Verwendung
US4644002A (en) * 1979-02-09 1987-02-17 Roussel Uclaf Imidazo[2,1-C]quinolines, useful as antiallergic agents
IT1150955B (it) * 1980-06-06 1986-12-17 Lepetit Spa Derivati 3h-naft(1.2-d)-imidazolici il procedimento per la loro preparazione, il loro uso come agenti antiinfiammatori e le composizioni farmaceutiche che li contengono
DE3314843A1 (de) * 1983-04-23 1984-10-25 Beiersdorf Ag, 2000 Hamburg 1-amidino-2,3,3a,8-tetrahydro-1h-pyrazolo (5,1-a)isoindol, verfahren zu dessen herstellung, diese verbindung enthaltende zubereitungen und zwischenprodukte
GB8415540D0 (en) * 1984-06-18 1984-07-25 Fujisawa Pharmaceutical Co Imidazoisoquinoline compounds
EP0607076A1 (de) * 1993-01-15 1994-07-20 Synthelabo 9H-Imidazo 1,2-a benzimidazolderivate mit GABA wirkung
US5948912A (en) * 1995-02-15 1999-09-07 Neurogen Corporation Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
WO1996025411A1 (en) * 1995-02-15 1996-08-22 Neurogen Corporation Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
TW416953B (en) 1996-09-25 2001-01-01 Takeda Chemical Industries Ltd Tricyclic compounds for eliciting a prostaglandin I2 receptor agonistic effect, their production and use
JP4251872B2 (ja) * 2001-04-19 2009-04-08 エーザイ・アール・アンド・ディー・マネジメント株式会社 2−イミノイミダゾール誘導体(2)
JPWO2002098863A1 (ja) * 2001-06-05 2004-09-16 藤沢薬品工業株式会社 縮合イミダゾール誘導体
JP4549970B2 (ja) * 2003-02-19 2010-09-22 エーザイ・アール・アンド・ディー・マネジメント株式会社 環状ベンズアミジン誘導体の製造方法
JP5063351B2 (ja) * 2004-09-17 2012-10-31 エグゼリクシス, インコーポレイテッド ピラゾールキナーゼモジュレーターおよび使用方法
US11142504B2 (en) 2016-03-07 2021-10-12 Northwestern University Substituted heterocycles as c-MYC targeting agents
WO2017155942A2 (en) * 2016-03-07 2017-09-14 Northwestern University Substituted heterocycles as c-myc targeting agents
WO2020257261A1 (en) 2019-06-17 2020-12-24 Northwestern University SUBSTITUTED HETEROCYCLES AS c-MYC TARGETING AGENTS
CN110294758B (zh) * 2019-07-06 2021-10-22 湘潭大学 2-取代5,6-二氢吡唑并[5,1-α]异喹啉、衍生物及其合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1244501A (en) * 1968-03-09 1971-09-02 Aspro Nicholas Ltd Heterocyclic amines
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives

Also Published As

Publication number Publication date
YU292775A (en) 1983-04-27
SE421620B (sv) 1982-01-18
GB1484615A (en) 1977-09-01
NO143578B (no) 1980-12-01
SU582764A3 (ru) 1977-11-30
DD122819A5 (de) 1976-11-05
DE2551868A1 (de) 1976-08-12
DE2551868C2 (de) 1982-07-15
NO143577B (no) 1980-12-01
BE835836A (fr) 1976-03-16
GR58292B (en) 1977-09-20
DD122818A5 (de) 1976-11-05
ATA884575A (de) 1977-11-15
IN141710B (de) 1977-04-09
GR58293B (en) 1977-09-20
CA1068274A (en) 1979-12-18
IE43567B1 (en) 1981-04-08
FI58919B (fi) 1981-01-30
AU8620475A (en) 1977-05-05
SE7513138L (sv) 1976-05-24
FR2291747A1 (fr) 1976-06-18
DK522275A (da) 1976-05-24
SE421619B (sv) 1982-01-18
IL48389A (en) 1979-01-31
ZA756792B (en) 1976-10-27
LU73850A1 (de) 1976-06-11
ATA884675A (de) 1978-03-15
NL165741C (nl) 1981-05-15
NO753854L (de) 1976-05-25
SU569290A3 (ru) 1977-08-15
FI753046A (de) 1976-05-24
LU73849A1 (de) 1976-06-11
JPS5175098A (de) 1976-06-29
FI58918C (fi) 1981-05-11
FI753045A (de) 1976-05-24
FR2291747B1 (de) 1978-11-17
JPS5516513B2 (de) 1980-05-02
ES442863A1 (es) 1977-08-16
DK152756C (da) 1988-09-26
CA1068273A (en) 1979-12-18
FI58918B (fi) 1981-01-30
NL7512848A (nl) 1976-05-25
AT344176B (de) 1978-07-10
CH614208A5 (de) 1979-11-15
SU578883A3 (ru) 1977-10-30
IE43567L (en) 1976-05-23
YU37328B (en) 1984-08-31
AR210476A1 (es) 1977-08-15
NO753853L (de) 1976-05-25
IL48389A0 (en) 1975-12-31
DK152756B (da) 1988-05-09
SE7513137L (sv) 1976-05-24
DK522175A (da) 1976-05-24
NO143578C (no) 1981-03-11
IN142014B (de) 1977-05-21
NL165741B (nl) 1980-12-15
FI58919C (fi) 1981-05-11
US4075342A (en) 1978-02-21
CH614444A5 (de) 1979-11-30
ES442864A1 (es) 1977-08-16
AR209459A1 (es) 1977-04-29
AT346332B (de) 1978-11-10

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