NO142625C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive, nye piperazinderivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive, nye piperazinderivater

Info

Publication number
NO142625C
NO142625C NO770374A NO770374A NO142625C NO 142625 C NO142625 C NO 142625C NO 770374 A NO770374 A NO 770374A NO 770374 A NO770374 A NO 770374A NO 142625 C NO142625 C NO 142625C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
piperazine derivatives
active new
analogy procedure
Prior art date
Application number
NO770374A
Other languages
English (en)
Norwegian (no)
Other versions
NO142625B (no
NO770374L (no
Inventor
Richard Cyrus
Manfred Raschack
Original Assignee
Knoll Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Knoll Ag filed Critical Knoll Ag
Publication of NO770374L publication Critical patent/NO770374L/no
Publication of NO142625B publication Critical patent/NO142625B/no
Publication of NO142625C publication Critical patent/NO142625C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
NO770374A 1976-02-07 1977-02-04 Analogifremgangsmaate ved fremstilling av terapeutisk aktive, nye piperazinderivater NO142625C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19762604845 DE2604845A1 (de) 1976-02-07 1976-02-07 Neue piperazinderivate

Publications (3)

Publication Number Publication Date
NO770374L NO770374L (no) 1977-08-09
NO142625B NO142625B (no) 1980-06-09
NO142625C true NO142625C (no) 1980-09-17

Family

ID=5969327

Family Applications (1)

Application Number Title Priority Date Filing Date
NO770374A NO142625C (no) 1976-02-07 1977-02-04 Analogifremgangsmaate ved fremstilling av terapeutisk aktive, nye piperazinderivater

Country Status (25)

Country Link
US (1) US4079137A (de)
JP (1) JPS52105186A (de)
AT (1) AT355578B (de)
AU (1) AU504526B2 (de)
BE (1) BE850492A (de)
CA (1) CA1094560A (de)
CH (1) CH631448A5 (de)
CS (1) CS201544B2 (de)
DD (1) DD128133A5 (de)
DE (1) DE2604845A1 (de)
DK (1) DK138891C (de)
ES (1) ES455691A1 (de)
FI (1) FI63226C (de)
FR (1) FR2340311A1 (de)
GB (1) GB1550545A (de)
HU (1) HU173483B (de)
IE (1) IE44339B1 (de)
IL (1) IL51316A (de)
LU (1) LU76706A1 (de)
NL (1) NL7700841A (de)
NO (1) NO142625C (de)
PL (1) PL105526B1 (de)
PT (1) PT66154B (de)
SE (1) SE7701187L (de)
ZA (1) ZA77248B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4341698A (en) * 1979-06-21 1982-07-27 Richardson-Merrell Inc. Enkaphalin derivatives
US4483988A (en) * 1980-03-14 1984-11-20 Richardson Merrell Inc. Substituted derivatives of 4-t-alkoxycarbonyl-piperazin-2-ones
US4766125A (en) * 1981-06-23 1988-08-23 Janssen Pharmaceutica N.V. N-aryl-piperazinealkanamides useful for protecting hearts from myocardial injury caused by ischaemia, anoxia or hypoxia
WO2006062917A2 (en) * 2004-12-06 2006-06-15 Sciclone Pharmaceuticals, Inc. Alpha thymosin peptides as cancer vaccine adjuvants
US20080300166A1 (en) * 2007-06-01 2008-12-04 Sciclone Pharmaceuticals, Inc. Treatment of Melanoma with Alpha Thymosin Peptides
EP2240195A4 (de) * 2007-12-12 2011-12-21 Sciclone Pharmaceuticals Inc Melanombehandlung mit alpha-thymosin-peptiden in kombination mit antikörpern gegen mit zytotoxischen t-lymphozyten assoziiertem antigen 4 (ctla4)
CN101945664A (zh) * 2007-12-13 2011-01-12 赛生制药有限公司 用α胸腺肽和激酶抑制剂的组合治疗黑素瘤
JP2011506467A (ja) * 2007-12-14 2011-03-03 サイクローン・ファーマシューティカルズ・インコーポレイテッド 抗悪性腫瘍性熱ショックアポトーシス活性化因子(hsaa)と組み合わせられたアルファチモシンペプチドによる黒色腫の処置の方法
US8829173B2 (en) 2008-09-26 2014-09-09 Tocagen Inc. Recombinant vectors
US8716012B2 (en) * 2009-05-08 2014-05-06 Sciclone Pharmaceuticals, Inc. Alpha thymosin peptides as vaccine enhancers
SG11201702558VA (en) 2014-10-21 2017-05-30 Sciclone Pharmaceuticals Inc Treatment of cancer with immune stimulators

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3472856A (en) * 1967-05-29 1969-10-14 Sterling Drug Inc 1-((thianaphthenyl)-lower-alkyl)-4-substituted-piperazines
US4031216A (en) * 1974-08-12 1977-06-21 Knoll A.G. Chemische Fabriken 3-(3,4-Dialkoxy-benzyl)-3-methyl-piperazines
DE2438725A1 (de) * 1974-08-12 1976-02-26 Knoll Ag Piperazinderivate

Also Published As

Publication number Publication date
IE44339L (en) 1977-08-07
CS201544B2 (en) 1980-11-28
IL51316A0 (en) 1977-03-31
DK138891B (da) 1978-11-13
DE2604845A1 (de) 1977-08-18
HU173483B (hu) 1979-05-28
DK138891C (da) 1979-04-23
LU76706A1 (de) 1977-06-28
SE7701187L (sv) 1977-08-08
BE850492A (fr) 1977-07-18
CH631448A5 (de) 1982-08-13
NL7700841A (nl) 1977-08-09
CA1094560A (en) 1981-01-27
FI770398A (de) 1977-08-08
ATA68177A (de) 1979-08-15
IL51316A (en) 1980-12-31
NO142625B (no) 1980-06-09
GB1550545A (en) 1979-08-15
AT355578B (de) 1980-03-10
DD128133A5 (de) 1977-11-02
AU504526B2 (en) 1979-10-18
NO770374L (no) 1977-08-09
JPS52105186A (en) 1977-09-03
ZA77248B (en) 1977-11-30
DK49077A (da) 1977-08-08
FI63226C (fi) 1983-05-10
FR2340311A1 (fr) 1977-09-02
ES455691A1 (es) 1978-01-01
FR2340311B1 (de) 1980-02-08
AU2195277A (en) 1978-08-10
PT66154A (fr) 1977-03-01
US4079137A (en) 1978-03-14
IE44339B1 (en) 1981-10-21
PT66154B (fr) 1978-07-07
FI63226B (fi) 1983-01-31
PL105526B1 (pl) 1979-10-31

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