NL8503424A - Indoolverbindingen; werkwijze voor het bereiden daarvan; farmaceutische preparaten. - Google Patents

Indoolverbindingen; werkwijze voor het bereiden daarvan; farmaceutische preparaten. Download PDF

Info

Publication number
NL8503424A
NL8503424A NL8503424A NL8503424A NL8503424A NL 8503424 A NL8503424 A NL 8503424A NL 8503424 A NL8503424 A NL 8503424A NL 8503424 A NL8503424 A NL 8503424A NL 8503424 A NL8503424 A NL 8503424A
Authority
NL
Netherlands
Prior art keywords
group
indole
general formula
compound
hydrogen atom
Prior art date
Application number
NL8503424A
Other languages
English (en)
Dutch (nl)
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NL8503424A publication Critical patent/NL8503424A/nl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
NL8503424A 1984-12-13 1985-12-12 Indoolverbindingen; werkwijze voor het bereiden daarvan; farmaceutische preparaten. NL8503424A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8431426 1984-12-13
GB848431426A GB8431426D0 (en) 1984-12-13 1984-12-13 Chemical compounds

Publications (1)

Publication Number Publication Date
NL8503424A true NL8503424A (nl) 1986-07-01

Family

ID=10571103

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8503424A NL8503424A (nl) 1984-12-13 1985-12-12 Indoolverbindingen; werkwijze voor het bereiden daarvan; farmaceutische preparaten.

Country Status (11)

Country Link
JP (1) JPS61151172A (it)
AU (1) AU579687B2 (it)
BE (1) BE903846A (it)
CH (1) CH667454A5 (it)
DE (1) DE3543982A1 (it)
FR (1) FR2574793B1 (it)
GB (2) GB8431426D0 (it)
IT (1) IT1182089B (it)
NL (1) NL8503424A (it)
SE (1) SE8505887L (it)
ZA (1) ZA859520B (it)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds
GB8607824D0 (en) * 1986-03-27 1986-04-30 Glaxo Group Ltd Chemical compounds
GB8614287D0 (en) * 1986-06-12 1986-07-16 Glaxo Group Ltd Chemical compounds
US4894386A (en) * 1987-04-15 1990-01-16 Ici Americas Inc. Aliphatic carboxamides
GB8719167D0 (en) * 1987-08-13 1987-09-23 Glaxo Group Ltd Chemical compounds
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
PT97888B (pt) * 1990-06-07 1998-12-31 Zeneca Ltd Processo para a preparacao de compostos heterociclicos derivados de indol e de composicoes farmaceuticas que os contem
GB9209882D0 (en) * 1992-05-07 1992-06-24 Glaxo Lab Sa Compositions
GB9211277D0 (en) 1992-05-28 1992-07-15 Glaxo Group Inc Pharmaceutical compositions
GB9216009D0 (en) * 1992-07-28 1992-09-09 Almirall Lab New indol derivatives
ES2056025B1 (es) * 1992-10-08 1995-05-01 Almirall Lab Nuevos derivados de indol.
FR2707639B1 (fr) * 1993-06-30 1995-10-13 Pf Medicament Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.
CA2508290C (en) 2002-12-20 2017-02-28 Ciba Specialty Chemicals Holding Inc. Synthesis of amines and intermediates for the synthesis thereof
WO2005118551A2 (en) 2004-05-28 2005-12-15 Ligand Pharmaceuticals Inc. Thrombopoietin activity modulating compounds and methods
EP1805155B1 (en) * 2004-10-25 2010-11-03 Ligand Pharmaceuticals, Inc. Thrombopoietin activity modulating compounds and methods
JP5164972B2 (ja) 2007-03-29 2013-03-21 第一三共株式会社 cPLA2阻害活性を有するインドール誘導体およびその用途並びに製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA795239B (en) * 1978-10-12 1980-11-26 Glaxo Group Ltd Heterocyclic compounds
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
BE903778A (fr) * 1984-12-04 1986-06-03 Glaxo Group Ltd Derives d'indoles.
GB8530507D0 (en) * 1985-12-11 1986-01-22 Glaxo Group Plc Chemical compounds

Also Published As

Publication number Publication date
GB2168347A (en) 1986-06-18
AU579687B2 (en) 1988-12-01
BE903846A (fr) 1986-06-12
GB8431426D0 (en) 1985-01-23
IT1182089B (it) 1987-09-30
SE8505887D0 (sv) 1985-12-12
CH667454A5 (fr) 1988-10-14
GB8530591D0 (en) 1986-01-22
AU5115185A (en) 1986-06-19
DE3543982A1 (de) 1986-06-19
JPS61151172A (ja) 1986-07-09
ZA859520B (en) 1986-08-27
FR2574793A1 (fr) 1986-06-20
GB2168347B (en) 1988-02-03
IT8548921A0 (it) 1985-12-12
FR2574793B1 (fr) 1988-10-14
SE8505887L (sv) 1986-06-14

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