NL8200828A - N-acyl-polypeptiden en werkwijzen voor het bereiden en toepassen van deze polypeptiden. - Google Patents

N-acyl-polypeptiden en werkwijzen voor het bereiden en toepassen van deze polypeptiden. Download PDF

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Publication number
NL8200828A
NL8200828A NL8200828A NL8200828A NL8200828A NL 8200828 A NL8200828 A NL 8200828A NL 8200828 A NL8200828 A NL 8200828A NL 8200828 A NL8200828 A NL 8200828A NL 8200828 A NL8200828 A NL 8200828A
Authority
NL
Netherlands
Prior art keywords
group
carbon atoms
acyl
formula
hydrogen atom
Prior art date
Application number
NL8200828A
Other languages
English (en)
Dutch (nl)
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1531/81A external-priority patent/CH647246A5/de
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of NL8200828A publication Critical patent/NL8200828A/nl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/26—Containing cys-cys disulfide bridge between nonadjacent cysteine residues

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Medicinal Chemistry (AREA)
  • Zoology (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NL8200828A 1981-03-06 1982-03-02 N-acyl-polypeptiden en werkwijzen voor het bereiden en toepassen van deze polypeptiden. NL8200828A (nl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH1531/81A CH647246A5 (en) 1981-03-06 1981-03-06 Polypeptide derivatives, their preparation and pharmaceutical products which contain these polypeptide derivatives
CH153181 1981-03-06
CH572381 1981-09-04
CH572381 1981-09-04

Publications (1)

Publication Number Publication Date
NL8200828A true NL8200828A (nl) 1982-10-01

Family

ID=25687920

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8200828A NL8200828A (nl) 1981-03-06 1982-03-02 N-acyl-polypeptiden en werkwijzen voor het bereiden en toepassen van deze polypeptiden.

Country Status (16)

Country Link
US (1) US4435385A (cs)
AU (1) AU8116482A (cs)
CA (1) CA1188682A (cs)
DE (1) DE3207311A1 (cs)
DK (1) DK81082A (cs)
ES (2) ES510167A0 (cs)
FI (1) FI820689L (cs)
FR (1) FR2501199B1 (cs)
GB (1) GB2095261B (cs)
GR (1) GR78227B (cs)
IL (1) IL65167A (cs)
IT (1) IT1189229B (cs)
NL (1) NL8200828A (cs)
NZ (1) NZ199911A (cs)
PT (1) PT74526B (cs)
SE (1) SE8201339L (cs)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH655505B (cs) * 1982-08-24 1986-04-30
CA1249397A (en) * 1984-03-07 1989-01-24 Fadia E. Ali Process for preparing des-proline vasopressin antagonists
US4684620A (en) * 1984-09-04 1987-08-04 Gibson-Stephens Neuropharmaceuticals, Inc. Cyclic polypeptides having mu-receptor specificity
GB8423431D0 (en) * 1984-09-17 1984-10-24 Sandoz Ltd Organic compounds
US4725577A (en) * 1985-04-25 1988-02-16 Administrators Of The Tulane Educational Fund Biologically active lysine containing octapeptides
US4650787A (en) * 1985-04-25 1987-03-17 Schally Andrew Victor Biologically active octapeptides
US4904642A (en) * 1985-09-12 1990-02-27 The Administrators Of The Tulane Educational Fund Therapeutic somatostatin analogs
GR862206B (en) * 1985-09-12 1986-12-31 Univ Tulane Therapeutic somatostatin analogs
JPH085913B2 (ja) * 1985-09-12 1996-01-24 ザ・アドミニストレ−タ−ズ・オブ・ザ・ツ−レイン・エデユケイシヨナル・フアンド 治療用ソマトスタチン同族体
US4853371A (en) * 1986-06-17 1989-08-01 The Administrators Of The Tulane Educational Fund Therapeutic somatostatin analogs
US4871717A (en) * 1987-01-07 1989-10-03 Administrators Of The Tulane Educational Fund Peptides
US4798821A (en) * 1987-03-02 1989-01-17 Merck & Co., Inc. Antihypertensive therapy for diabetics
US5073541A (en) * 1987-11-18 1991-12-17 Administrators Of The Tulane Educational Fund Treatment of small cell lung cancer with somatostatin analogs
US5019647A (en) * 1988-05-24 1991-05-28 Merck & Co., Inc. Gastrin releasing peptide antagonist
US5028692A (en) * 1989-04-25 1991-07-02 Merck & Co., Inc. Gastrin releasing peptide antagonist
EP0457888B1 (en) * 1989-12-08 1996-07-10 The Administrators of The Tulane Educational Fund Octapeptide analogs of somatostatin having threonine at the sixth position
US5504069A (en) * 1993-02-11 1996-04-02 Biomeasure, Inc. Inhibition of trauma-induced tumor growth
US5597894A (en) * 1995-06-05 1997-01-28 The Louisiana State University Medical Center Foundation Multi-tyrosinated somatostatin analogs
US6262229B1 (en) 1996-12-04 2001-07-17 Biomeasure Incorporated Somatostatin antagonists
US7026289B2 (en) 1997-05-13 2006-04-11 Societe De Conseils De Recherches Et D'applications Scientifiques, Sas Method and compositions for treating hyperlipidemia and other conditions
AU8019898A (en) * 1997-05-13 1998-12-08 Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) Somatostatin and somatostatin agonists for treating insulin insensitivity and syndrome
US6004928A (en) * 1997-05-13 1999-12-21 Biomeasure, Incorporated Method of treating hyperlipidemia
WO1998051331A1 (en) 1997-05-13 1998-11-19 Societe De Conseils De Recherches Et D'applications Scientifiques S.A. (S.C.R.A.S.) Somatostatin and somatostatin agonists for decreasing body weight
US5968903A (en) * 1998-05-07 1999-10-19 Biomeasure, Incorporated Inhibition of H. pylori proliferation
US6750199B2 (en) * 2000-07-17 2004-06-15 Micrologix Biotech Inc. Antimicrobial sulfonamide derivatives of lipopeptide antibiotics
KR100743212B1 (ko) 2001-06-08 2007-07-26 소시에떼 더 콘세이유 더 레세르세 에 다플리까띠옹 시엔띠피끄, 에스.아.에스. 소마토스타틴-도파민 키메라 유사체
CA2523197C (en) 2003-04-22 2016-05-24 Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. Peptide vectors
WO2014197938A1 (en) 2013-06-13 2014-12-18 Antisense Therapeutics Ltd Combination therapy

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904594A (en) 1973-07-02 1975-09-09 Salk Inst For Biological Studi Somatostatin and acylated des-(ala' 1', gly' 2') derivatives thereof
DE2608336A1 (de) * 1975-03-11 1976-09-30 Sandoz Ag Neue organische verbindungen, ihre herstellung und verwendung
NL7902932A (nl) * 1978-04-24 1979-10-26 American Home Prod Aan somatostatine structureel verwante peptiden.
US4225472A (en) * 1979-05-29 1980-09-30 American Home Products Corporation Truncated somatostatin analogs
DE19375086I2 (de) * 1979-11-27 2003-01-09 Novartis Ag Polypeptide Verfahren zu ihrer Herstellung pharmazeutische Zusammensetzungen die diese Polypeptide enthalten und ihre Verwendung
US4282143A (en) * 1980-06-13 1981-08-04 American Home Products Corporation Octapeptides lowering growth hormone

Also Published As

Publication number Publication date
DK81082A (da) 1982-09-07
IT8247937A1 (it) 1983-09-05
CA1188682A (en) 1985-06-11
ES8503642A1 (es) 1985-03-01
DE3207311A1 (de) 1982-12-02
IL65167A (en) 1985-06-30
ES8400082A1 (es) 1983-10-16
SE8201339L (sv) 1982-09-07
IT1189229B (it) 1988-01-28
IT8247937A0 (it) 1982-03-05
FI820689A7 (fi) 1982-09-07
FR2501199B1 (fr) 1986-02-21
AU8116482A (en) 1982-09-09
GR78227B (cs) 1984-09-26
FI820689L (fi) 1982-09-07
NZ199911A (en) 1985-05-31
PT74526B (en) 1984-10-09
US4435385A (en) 1984-03-06
GB2095261B (en) 1984-08-15
GB2095261A (en) 1982-09-29
ES522916A0 (es) 1985-03-01
ES510167A0 (es) 1983-10-16
PT74526A (en) 1982-04-01
FR2501199A1 (fr) 1982-09-10
IL65167A0 (en) 1982-05-31

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BV The patent application has lapsed