NL8105529A - Werkwijze voor het bereiden van buspirone. - Google Patents

Werkwijze voor het bereiden van buspirone. Download PDF

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Publication number
NL8105529A
NL8105529A NL8105529A NL8105529A NL8105529A NL 8105529 A NL8105529 A NL 8105529A NL 8105529 A NL8105529 A NL 8105529A NL 8105529 A NL8105529 A NL 8105529A NL 8105529 A NL8105529 A NL 8105529A
Authority
NL
Netherlands
Prior art keywords
formula
azaspiro
dione
decane
labeled
Prior art date
Application number
NL8105529A
Other languages
English (en)
Dutch (nl)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of NL8105529A publication Critical patent/NL8105529A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/20—Spiro-condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
NL8105529A 1980-12-11 1981-12-08 Werkwijze voor het bereiden van buspirone. NL8105529A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21521480A 1980-12-11 1980-12-11
US21521480 1980-12-11

Publications (1)

Publication Number Publication Date
NL8105529A true NL8105529A (nl) 1982-07-01

Family

ID=22802113

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8105529A NL8105529A (nl) 1980-12-11 1981-12-08 Werkwijze voor het bereiden van buspirone.

Country Status (18)

Country Link
JP (1) JPS57122082A (cs)
AT (1) AT380686B (cs)
AU (1) AU528067B2 (cs)
BE (1) BE891446A (cs)
CA (1) CA1172255A (cs)
CH (1) CH647518A5 (cs)
DE (1) DE3149011A1 (cs)
DK (1) DK154560C (cs)
FI (1) FI73993C (cs)
FR (1) FR2496105B1 (cs)
GB (1) GB2089341B (cs)
GR (1) GR76331B (cs)
IE (1) IE51948B1 (cs)
IT (1) IT1172073B (cs)
LU (1) LU83833A1 (cs)
NL (1) NL8105529A (cs)
SE (1) SE444438B (cs)
YU (1) YU42432B (cs)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU212301B (en) * 1989-04-28 1996-05-28 Alkaloida Vegyeszeti Gyar Process for producing buspirone
US5484788A (en) * 1993-03-26 1996-01-16 Beth Israel Hospital Association Buspirone as a systemic immunosuppressant
US5631017A (en) * 1993-03-26 1997-05-20 Beth Israel Deaconess Medical Center, Inc. Topical application of buspirone for treatment of pathological conditions associated with immune responses
KR950014099A (ko) * 1993-11-10 1995-06-15 장기하 N-(2-피리미딜)피페라지닐 부틸아미드의 제조방법
US5637314A (en) * 1995-06-07 1997-06-10 Beth Israel Deaconess Medical Center, Inc. Topical and systemic application of buspirone or derivatives thereof for treating atopic dermatitis

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE759371A (fr) * 1969-11-24 1971-05-24 Bristol Myers Co Azaspirodecanediones heterocycliques et procedes pour leur preparation
DE2341925A1 (de) * 1973-08-20 1975-03-06 Thomae Gmbh Dr K Neue pyrimidinderivate und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
GR76331B (cs) 1984-08-04
IT1172073B (it) 1987-06-18
CA1172255A (en) 1984-08-07
DE3149011C2 (cs) 1988-08-25
CH647518A5 (de) 1985-01-31
AT380686B (de) 1986-06-25
DK154560C (da) 1989-04-17
FI813937L (fi) 1982-06-12
IE51948B1 (en) 1987-04-29
SE444438B (sv) 1986-04-14
DE3149011A1 (de) 1982-07-15
IT8149718A0 (it) 1981-11-16
GB2089341A (en) 1982-06-23
IE812897L (en) 1982-06-11
FR2496105A1 (fr) 1982-06-18
JPS57122082A (en) 1982-07-29
LU83833A1 (fr) 1982-07-07
FR2496105B1 (fr) 1985-12-13
GB2089341B (en) 1984-09-19
JPH0113476B2 (cs) 1989-03-06
YU243681A (en) 1984-02-29
FI73993B (fi) 1987-08-31
ATA529581A (de) 1985-11-15
DK154560B (da) 1988-11-28
FI73993C (fi) 1987-12-10
AU528067B2 (en) 1983-04-14
DK548081A (da) 1982-06-12
YU42432B (en) 1988-08-31
BE891446A (fr) 1982-06-11
SE8107446L (sv) 1982-06-12
AU7604181A (en) 1982-07-15

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Legal Events

Date Code Title Description
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
A85 Still pending on 85-01-01
BC A request for examination has been filed
BN A decision not to publish the application has become irrevocable