NL8102099A - 2-guanidinothiazool-derivaten met farmacologische werking. - Google Patents

2-guanidinothiazool-derivaten met farmacologische werking. Download PDF

Info

Publication number
NL8102099A
NL8102099A NL8102099A NL8102099A NL8102099A NL 8102099 A NL8102099 A NL 8102099A NL 8102099 A NL8102099 A NL 8102099A NL 8102099 A NL8102099 A NL 8102099A NL 8102099 A NL8102099 A NL 8102099A
Authority
NL
Netherlands
Prior art keywords
guanidino
group
thiazole
formula
derivatives according
Prior art date
Application number
NL8102099A
Other languages
English (en)
Dutch (nl)
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of NL8102099A publication Critical patent/NL8102099A/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NL8102099A 1980-04-29 1981-04-28 2-guanidinothiazool-derivaten met farmacologische werking. NL8102099A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14494680A 1980-04-29 1980-04-29
US14494680 1980-04-29

Publications (1)

Publication Number Publication Date
NL8102099A true NL8102099A (nl) 1981-11-16

Family

ID=22510873

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8102099A NL8102099A (nl) 1980-04-29 1981-04-28 2-guanidinothiazool-derivaten met farmacologische werking.

Country Status (16)

Country Link
JP (1) JPS574977A (ja)
AR (1) AR231538A1 (ja)
AU (1) AU540239B2 (ja)
BE (1) BE888602A (ja)
CH (1) CH646964A5 (ja)
DE (1) DE3116890A1 (ja)
DK (1) DK188881A (ja)
ES (1) ES8206501A1 (ja)
FR (1) FR2481280A1 (ja)
GB (1) GB2076397B (ja)
IE (1) IE51151B1 (ja)
IL (1) IL62747A (ja)
IT (1) IT1146750B (ja)
NL (1) NL8102099A (ja)
NZ (1) NZ196923A (ja)
SE (1) SE452462B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2531705B1 (fr) * 1982-08-13 1986-12-05 Sanofi Sa Amidobenzamides, leurs sels, procede pour leur preparation et compositions pharmaceutiques les renfermant
US4501747A (en) * 1982-05-10 1985-02-26 Sanofi Certain amide derivatives of 2-guanidino-thiazoles and compositions containing same
JPS59104370A (ja) * 1982-12-03 1984-06-16 Kotobuki Seiyaku Kk チアゾ−ル誘導体及びその製造方法
GB2138803B (en) * 1983-04-26 1986-06-18 Shionogi & Co 2-guanidino-4-hydroxymethylthiazole and derivatives thereof
US4680300A (en) * 1985-01-10 1987-07-14 Syntex (U.S.A.) Inc. Anti-inflammatory guanidines
US4837316A (en) * 1985-08-29 1989-06-06 Fujirebio Kabushiki Kaisha Alkylamide derivatives with H2 -receptor antagonistic and cytoprotective action
EP0385525B1 (en) * 1989-03-03 1994-04-13 Akzo Nv Aminoethylthiazole and aminoethyloxazole derivatives.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4165378A (en) * 1977-04-20 1979-08-21 Ici Americas Inc. Guanidine derivatives of imidazoles and thiazoles
ZA782129B (en) * 1977-04-20 1979-03-28 Ici Ltd Hertocyclic derivatives
EP0003640B1 (en) * 1978-01-18 1982-01-27 Imperial Chemical Industries Plc Antisecretory guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them
ATE6156T1 (de) * 1978-10-16 1984-02-15 Imperial Chemical Industries Plc Verzweigtkettige heterozyklische guanidinderivate mit antisekretorischer wirkung, verfahren zu ihrer herstellung, zwischenprodukte und die genannten derivate enthaltende pharmazeutische zusammensetzungen.
US4309435A (en) * 1978-10-16 1982-01-05 Imperial Chemical Industries Ltd. Antisecretory guanidine derivatives and pharmaceutical compositions containing them
EP0014057B1 (en) * 1979-01-18 1985-01-02 Imperial Chemical Industries Plc Guanidine derivatives, processes for their manufacture and pharmaceutical compositions containing them
PH16099A (en) * 1979-03-06 1983-06-24 Yamanouchi Pharma Co Ltd Guanidinothiazole compounds,process for preparing them and medical composition containing them
GR71929B (ja) * 1979-11-13 1983-08-19 Ici Ltd
JPS5754177A (ja) * 1980-09-19 1982-03-31 Teikoku Hormone Mfg Co Ltd Chikanchiazoorujudotai
JPS57102852A (en) * 1980-12-19 1982-06-26 Shionogi & Co Ltd Dicarboxylic acid diamide

Also Published As

Publication number Publication date
SE8102683L (sv) 1981-10-30
IT8167585A0 (it) 1981-04-29
ES501736A0 (es) 1982-08-16
JPS574977A (en) 1982-01-11
NZ196923A (en) 1983-12-16
DK188881A (da) 1981-10-30
IL62747A0 (en) 1981-06-29
JPH027952B2 (ja) 1990-02-21
FR2481280A1 (fr) 1981-10-30
BE888602A (fr) 1981-10-28
GB2076397B (en) 1984-02-08
AU540239B2 (en) 1984-11-08
AR231538A1 (es) 1984-12-28
AU6996681A (en) 1981-11-05
IE51151B1 (en) 1986-10-15
GB2076397A (en) 1981-12-02
IT1146750B (it) 1986-11-19
ES8206501A1 (es) 1982-08-16
IE810956L (en) 1981-10-29
IL62747A (en) 1984-10-31
FR2481280B1 (ja) 1983-10-28
DE3116890A1 (de) 1982-03-04
CH646964A5 (de) 1984-12-28
SE452462B (sv) 1987-11-30

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BV The patent application has lapsed