MXPA04011858A - Quinuclidinas sustituidas en la posicion 3 y su uso. - Google Patents
Quinuclidinas sustituidas en la posicion 3 y su uso.Info
- Publication number
- MXPA04011858A MXPA04011858A MXPA04011858A MXPA04011858A MXPA04011858A MX PA04011858 A MXPA04011858 A MX PA04011858A MX PA04011858 A MXPA04011858 A MX PA04011858A MX PA04011858 A MXPA04011858 A MX PA04011858A MX PA04011858 A MXPA04011858 A MX PA04011858A
- Authority
- MX
- Mexico
- Prior art keywords
- alkyl
- independently
- represent hydrogen
- amino
- halo
- Prior art date
Links
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- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Reproductive Health (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Gynecology & Obstetrics (AREA)
- Pulmonology (AREA)
- Obesity (AREA)
- Virology (AREA)
- Nutrition Science (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- AIDS & HIV (AREA)
- Child & Adolescent Psychology (AREA)
- Urology & Nephrology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200200834 | 2002-05-30 | ||
| PCT/DK2003/000354 WO2003101987A1 (en) | 2002-05-30 | 2003-05-27 | 3-substituted quinuclidines and their use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA04011858A true MXPA04011858A (es) | 2005-03-31 |
Family
ID=29594980
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA04011858A MXPA04011858A (es) | 2002-05-30 | 2003-05-27 | Quinuclidinas sustituidas en la posicion 3 y su uso. |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US7332507B2 (https=) |
| EP (1) | EP1513839B1 (https=) |
| JP (1) | JP2005530814A (https=) |
| CN (1) | CN1656093A (https=) |
| AT (1) | ATE334129T1 (https=) |
| AU (1) | AU2003227522A1 (https=) |
| CA (1) | CA2482639A1 (https=) |
| DE (1) | DE60307102T2 (https=) |
| MX (1) | MXPA04011858A (https=) |
| NZ (1) | NZ536197A (https=) |
| WO (1) | WO2003101987A1 (https=) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA05003317A (es) | 2002-09-25 | 2005-07-05 | Memory Pharm Corp | Indazoles, benzotiazoles y benzoisotiazoles asi como preparacion y usos de los mismos. |
| DE602004010299T2 (de) | 2003-12-22 | 2008-09-18 | Memory Pharmaceuticals Corp. | Indole, 1h-indazole, 1,2-benzisoxazole und 1,2-benzisothiazole und deren herstellung und anwendungen |
| NZ550534A (en) | 2004-03-25 | 2009-07-31 | Memory Pharm Corp | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| WO2006001894A1 (en) | 2004-04-22 | 2006-01-05 | Memory Pharmaceutical Corporation | Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
| JP2007538011A (ja) | 2004-05-07 | 2007-12-27 | メモリー・ファーマシューティカルズ・コーポレイション | １ｈ−インダゾール、ベンゾチアゾール、１，２−ベンゾイソキサゾール、１，２−ベンゾイソチアゾール、およびクロモン、ならびにそれらの調製および使用 |
| AR050253A1 (es) | 2004-06-24 | 2006-10-11 | Smithkline Beecham Corp | Compuesto derivado de indazol carboxamida, composicion que lo comprende y su uso para la preparacion de un medicamento |
| RU2418797C2 (ru) | 2004-12-22 | 2011-05-20 | Мемори Фармасьютиклз Корпорейшн | Лиганды никотинового рецептора альфа-7, их получение и применение |
| US8063071B2 (en) | 2007-10-31 | 2011-11-22 | GlaxoSmithKline, LLC | Chemical compounds |
| PE20081889A1 (es) | 2007-03-23 | 2009-03-05 | Smithkline Beecham Corp | Indol carboxamidas como inhibidores de ikk2 |
| WO2010102968A1 (en) | 2009-03-10 | 2010-09-16 | Glaxo Group Limited | Indole derivatives as ikk2 inhibitors |
| CN110845492B (zh) * | 2018-08-21 | 2022-05-13 | 鲁南制药集团股份有限公司 | 一种异丙托溴铵一水合物 |
| CN110845491B (zh) * | 2018-08-21 | 2022-05-13 | 鲁南制药集团股份有限公司 | 一种异丙托溴铵晶体 |
| CN113121522A (zh) * | 2019-12-30 | 2021-07-16 | 武汉先路医药科技股份有限公司 | 一种异丙托溴铵晶体及其制备方法 |
| CN114306331B (zh) * | 2020-10-10 | 2023-07-18 | 远大生命科学(武汉)有限公司 | 戊乙奎醚在治疗或预防视力损伤性眼部疾病中的用途 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4009565A1 (de) * | 1990-03-24 | 1991-09-26 | Merck Patent Gmbh | Indolderivate |
| SE9201478D0 (sv) | 1992-05-11 | 1992-05-11 | Kabi Pharmacia Ab | Heteroaromatic quinuclidinenes, their use and preparation |
| SE9904176D0 (sv) | 1999-11-18 | 1999-11-18 | Astra Ab | New use |
| DE10045112A1 (de) * | 2000-09-11 | 2002-03-21 | Merck Patent Gmbh | Verwendung von Indolderivaten zur Behandlung von Erkrankungen des zentralen Nervensystems |
| AU2001296193B2 (en) * | 2000-10-20 | 2006-04-27 | Biovitrum Ab | 2-, 3-, 4-, or 5-substituted-N1-(benzensulfonyl)indoles and their use in therapy |
| US6884807B2 (en) | 2000-12-01 | 2005-04-26 | Neurosearch, A/S | 3-substituted quinuclidines and their use as nicotinic agonists |
| DE10121217A1 (de) * | 2001-04-30 | 2002-10-31 | Merck Patent Gmbh | 6H-Oxazolo[4,5-e]indol-Derivate als nikotinische Acetylcholinrezeptor Liganden und/oder serotonerge Liganden |
| DE10121215A1 (de) * | 2001-04-30 | 2002-10-31 | Merck Patent Gmbh | Dihydro-imidazo[4,5-e]indol- und 7H-Pyrrolo[3,2-f]chinoxalin Derivate als nikotinische Acetylcholinrezeptor Liganden und/oder serotonerge Liganden |
-
2003
- 2003-05-27 AU AU2003227522A patent/AU2003227522A1/en not_active Abandoned
- 2003-05-27 CN CNA038123258A patent/CN1656093A/zh active Pending
- 2003-05-27 DE DE60307102T patent/DE60307102T2/de not_active Expired - Lifetime
- 2003-05-27 CA CA002482639A patent/CA2482639A1/en not_active Abandoned
- 2003-05-27 US US10/512,570 patent/US7332507B2/en not_active Expired - Fee Related
- 2003-05-27 JP JP2004509678A patent/JP2005530814A/ja not_active Withdrawn
- 2003-05-27 AT AT03724901T patent/ATE334129T1/de not_active IP Right Cessation
- 2003-05-27 MX MXPA04011858A patent/MXPA04011858A/es active IP Right Grant
- 2003-05-27 EP EP03724901A patent/EP1513839B1/en not_active Expired - Lifetime
- 2003-05-27 WO PCT/DK2003/000354 patent/WO2003101987A1/en not_active Ceased
- 2003-05-27 NZ NZ536197A patent/NZ536197A/en not_active IP Right Cessation
-
2007
- 2007-12-20 US US12/004,022 patent/US20080132704A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| DE60307102T2 (de) | 2006-12-07 |
| AU2003227522A1 (en) | 2003-12-19 |
| EP1513839B1 (en) | 2006-07-26 |
| WO2003101987A1 (en) | 2003-12-11 |
| US20050176756A1 (en) | 2005-08-11 |
| CN1656093A (zh) | 2005-08-17 |
| EP1513839A1 (en) | 2005-03-16 |
| US20080132704A1 (en) | 2008-06-05 |
| JP2005530814A (ja) | 2005-10-13 |
| CA2482639A1 (en) | 2003-12-11 |
| DE60307102D1 (de) | 2006-09-07 |
| NZ536197A (en) | 2006-08-31 |
| ATE334129T1 (de) | 2006-08-15 |
| US7332507B2 (en) | 2008-02-19 |
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| FG | Grant or registration |