MXPA03004250A - Compuesto de lactama. - Google Patents

Compuesto de lactama.

Info

Publication number
MXPA03004250A
MXPA03004250A MXPA03004250A MXPA03004250A MXPA03004250A MX PA03004250 A MXPA03004250 A MX PA03004250A MX PA03004250 A MXPA03004250 A MX PA03004250A MX PA03004250 A MXPA03004250 A MX PA03004250A MX PA03004250 A MXPA03004250 A MX PA03004250A
Authority
MX
Mexico
Prior art keywords
lactam compound
lactam
compound
Prior art date
Application number
MXPA03004250A
Other languages
English (en)
Spanish (es)
Inventor
David Mitchell
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MXPA03004250A publication Critical patent/MXPA03004250A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrrole Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
MXPA03004250A 2000-11-17 2001-11-02 Compuesto de lactama. MXPA03004250A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24965600P 2000-11-17 2000-11-17
PCT/US2001/027795 WO2002040451A2 (en) 2000-11-17 2001-11-02 Lactam compound

Publications (1)

Publication Number Publication Date
MXPA03004250A true MXPA03004250A (es) 2003-09-22

Family

ID=22944436

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03004250A MXPA03004250A (es) 2000-11-17 2001-11-02 Compuesto de lactama.

Country Status (33)

Country Link
US (1) US20040248878A1 (OSRAM)
EP (1) EP1353910B1 (OSRAM)
JP (1) JP4116431B2 (OSRAM)
KR (1) KR20030045194A (OSRAM)
CN (2) CN101624372A (OSRAM)
AR (1) AR031356A1 (OSRAM)
AT (1) ATE362919T1 (OSRAM)
AU (2) AU2432102A (OSRAM)
BR (1) BR0115424A (OSRAM)
CA (1) CA2425497C (OSRAM)
CY (1) CY1106682T1 (OSRAM)
CZ (1) CZ20031340A3 (OSRAM)
DE (1) DE60128587T2 (OSRAM)
DK (1) DK1353910T3 (OSRAM)
DZ (1) DZ3454A1 (OSRAM)
EA (1) EA006919B1 (OSRAM)
EC (1) ECSP034598A (OSRAM)
ES (1) ES2286162T3 (OSRAM)
HR (1) HRP20030385A2 (OSRAM)
HU (1) HUP0301862A3 (OSRAM)
IL (1) IL155275A0 (OSRAM)
MX (1) MXPA03004250A (OSRAM)
MY (1) MY141607A (OSRAM)
NO (1) NO325217B1 (OSRAM)
PE (1) PE20020798A1 (OSRAM)
PL (1) PL211018B1 (OSRAM)
PT (1) PT1353910E (OSRAM)
SK (1) SK287794B6 (OSRAM)
SV (1) SV2003000741A (OSRAM)
TW (1) TWI235151B (OSRAM)
UA (1) UA77165C2 (OSRAM)
WO (1) WO2002040451A2 (OSRAM)
ZA (1) ZA200303411B (OSRAM)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA74849C2 (en) * 2000-11-17 2006-02-15 Lilly Co Eli Lactam
CA2509413C (en) 2002-12-20 2012-05-01 Glaxo Group Limited Benzazepine derivatives for the treatment of neurological disorders
DE602004009295T2 (de) 2003-01-14 2008-07-03 Arena Pharmaceuticals, Inc., San Diego 1,2,3-trisubstituierte aryl- und heteroarylderivate als modulatoren des metabolismus zur vorbeugung und behandlung von metabolismus-bedingten krankheiten wie diabetes oder hyperglykämie
AR045047A1 (es) 2003-07-11 2005-10-12 Arena Pharm Inc Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos
RU2404968C2 (ru) 2005-04-08 2010-11-27 Дайити Санкио Компани, Лимитед Пиридилдиметилсульфоновое производное
EP1985615A4 (en) 2006-01-31 2011-12-14 Api Corp PROCESS FOR THE PREPARATION OF BENZAZEPINONE
TW200920362A (en) 2007-09-11 2009-05-16 Daiichi Sankyo Co Ltd Alkylsulfone derivatives
FR2932800B1 (fr) * 2008-06-20 2015-02-20 Servier Lab Nouveau procede de synthese de la 7,8-dimethoxy-1,3-dihydro- 2h-3-benzazepin-2-one, et application a la synthese de l'ivabradine et de ses sels d'addition a un acide pharmaceutiquement acceptable
PH12013500547A1 (en) 2010-09-22 2013-06-10 Arena Pharm Inc Modulators of the gpr119 receptor and the treatment of disorders related thereto
KR101899014B1 (ko) 2012-01-06 2018-09-17 삼성전자주식회사 비엘디씨 모터의 제어 장치 및 그 방법
CN102690231B (zh) * 2012-04-11 2014-07-09 南京友杰医药科技有限公司 治疗阿尔茨海默病潜在药物司马西特的合成方法
EP2987496B1 (en) 2013-04-19 2018-08-08 National University Corporation Okayama University Treatment agent for cognitive disorders, induced by amyloid -protein, therapeutic agent for alzheimer's disease, and treatment method and pathological analysis method related to these
ES2995737T3 (en) 2015-01-06 2025-02-11 Arena Pharm Inc Compound for use in treating conditions related to the s1p1 receptor
MA42807A (fr) 2015-06-22 2018-07-25 Arena Pharm Inc Sel l-arginine cristallin d'acide (r)-2-(7-(4-cyclopentyl-3-(trifluorométhyl)benzyloxy)-1,2,3,4-tétrahydrocyclo-penta[b]indol-3-yl)acétique (composé 1) pour une utilisation dans des troubles associés au récepteur de s1p1
WO2018151873A1 (en) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of primary biliary cholangitis
EP3801459B1 (en) 2018-06-06 2024-08-07 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the s1p1 receptor
EP4126952A1 (en) 2020-03-26 2023-02-08 Seagen Inc. Methods of treating multiple myeloma

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3812952B2 (ja) * 1996-12-23 2006-08-23 エラン ファーマシューティカルズ,インコーポレイテッド シクロアルキル、ラクタム、ラクトンおよびその関連化合物およびその医薬組成物、並びに該化合物を用いたβ−アミロイドペプチドの放出および/またはその合成を阻害する方法
WO1999067219A1 (en) * 1998-06-22 1999-12-29 Elan Pharmaceuticals, Inc. Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
AU1569501A (en) * 1999-11-09 2001-06-06 Eli Lilly And Company Beta-aminoacid compounds useful for inhibiting beta-amyloid peptide release and/or its synthesis

Also Published As

Publication number Publication date
EP1353910A2 (en) 2003-10-22
PE20020798A1 (es) 2002-09-06
CN1575282A (zh) 2005-02-02
AU2432102A (en) 2002-05-27
EA006919B1 (ru) 2006-04-28
DE60128587D1 (de) 2007-07-05
HRP20030385A2 (en) 2003-08-31
CY1106682T1 (el) 2012-05-23
DK1353910T3 (da) 2007-09-10
US20040248878A1 (en) 2004-12-09
WO2002040451A2 (en) 2002-05-23
CA2425497A1 (en) 2002-05-23
NO20032215D0 (no) 2003-05-15
AU2002224321B2 (en) 2006-10-19
BR0115424A (pt) 2003-10-21
PL211018B1 (pl) 2012-03-30
CA2425497C (en) 2010-08-17
HUP0301862A2 (hu) 2003-09-29
CN100516047C (zh) 2009-07-22
MY141607A (en) 2010-05-31
DE60128587T2 (de) 2008-01-31
ATE362919T1 (de) 2007-06-15
KR20030045194A (ko) 2003-06-09
NO325217B1 (no) 2008-02-25
EP1353910B1 (en) 2007-05-23
PT1353910E (pt) 2007-08-20
SK5432003A3 (en) 2004-09-08
NO20032215L (no) 2003-07-16
DZ3454A1 (fr) 2002-05-23
ZA200303411B (en) 2004-08-02
EA200300579A1 (ru) 2003-12-25
PL360991A1 (en) 2004-09-20
IL155275A0 (en) 2003-11-23
AR031356A1 (es) 2003-09-17
CZ20031340A3 (cs) 2004-06-16
ECSP034598A (es) 2003-06-25
JP2004521084A (ja) 2004-07-15
SK287794B6 (sk) 2011-10-04
WO2002040451A3 (en) 2003-08-28
JP4116431B2 (ja) 2008-07-09
UA77165C2 (en) 2006-11-15
ES2286162T3 (es) 2007-12-01
CN101624372A (zh) 2010-01-13
HUP0301862A3 (en) 2007-09-28
SV2003000741A (es) 2003-01-13
TWI235151B (en) 2005-07-01

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