MX9303145A - 7-(2-aminoetil)benzotiazolonas. - Google Patents

7-(2-aminoetil)benzotiazolonas.

Info

Publication number
MX9303145A
MX9303145A MX9303145A MX9303145A MX9303145A MX 9303145 A MX9303145 A MX 9303145A MX 9303145 A MX9303145 A MX 9303145A MX 9303145 A MX9303145 A MX 9303145A MX 9303145 A MX9303145 A MX 9303145A
Authority
MX
Mexico
Prior art keywords
independently represent
benzotiazolonas
aminoetil
membered
halogen
Prior art date
Application number
MX9303145A
Other languages
English (en)
Inventor
Roger Victor Bonnert
Roger Charles Brown
David Ranulf Cheshire
Francis Ince
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fisons Plc filed Critical Fisons Plc
Publication of MX9303145A publication Critical patent/MX9303145A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Cosmetics (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Adhesives Or Adhesive Processes (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se describen compuestos de la fórmula (I) en donde: X y Y representan independientemente -S(O)n- ó -O- n representan 0, 1 ó 2, p, q, y r, representa independientemente 2 ó 3, z representa fenilo opcionalmente substituído por halógeno, -OR1, -NO2, ó -NR2R3; ó heterociclo que contiene 5 ó 6 miembros de N, O, ó S y R1, R2 y R3 representan independientemente hidrógeno o alquilo de 1 a 6 átomos de carbono, y derivados farmacéuticamente aceptables de los mismos. También se describen procedimientos para su producción, y composiciones farmacéuticamente y métodos de tratamiento que involucran su uso.
MX9303145A 1992-05-27 1993-05-27 7-(2-aminoetil)benzotiazolonas. MX9303145A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929211172A GB9211172D0 (en) 1992-05-27 1992-05-27 Compounds

Publications (1)

Publication Number Publication Date
MX9303145A true MX9303145A (es) 1994-06-30

Family

ID=10716059

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9303145A MX9303145A (es) 1992-05-27 1993-05-27 7-(2-aminoetil)benzotiazolonas.

Country Status (31)

Country Link
EP (1) EP0649418B1 (es)
JP (1) JP3094452B2 (es)
KR (1) KR100279132B1 (es)
CN (1) CN1036393C (es)
AT (1) ATE172726T1 (es)
AU (1) AU675649B2 (es)
CA (1) CA2136553C (es)
CZ (1) CZ286905B6 (es)
DE (1) DE69321835T2 (es)
DK (1) DK0649418T3 (es)
DZ (1) DZ1694A1 (es)
ES (1) ES2123652T3 (es)
FI (1) FI945538A (es)
GB (1) GB9211172D0 (es)
HU (2) HUT71124A (es)
IL (1) IL105801A (es)
LV (1) LV12443B (es)
MA (1) MA22895A1 (es)
MX (1) MX9303145A (es)
MY (1) MY131193A (es)
NO (1) NO304739B1 (es)
NZ (1) NZ253190A (es)
PH (1) PH31453A (es)
PL (2) PL172904B1 (es)
RU (1) RU2114108C1 (es)
SG (1) SG48068A1 (es)
SK (1) SK281282B6 (es)
TW (1) TW368501B (es)
UA (1) UA27901C2 (es)
WO (1) WO1993024473A1 (es)
ZA (1) ZA933648B (es)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW356468B (en) * 1995-09-15 1999-04-21 Astra Pharma Prod Benzothiazolone compounds useful as beta2-adrenoreceptor and dopamine DA2 receptor agonists process for preparing same and pharmaceutical compositions containing same
GB9526511D0 (en) * 1995-12-23 1996-02-28 Astra Pharma Prod Pharmaceutically active compounds
SE9900693D0 (sv) * 1999-02-26 1999-02-26 Astra Pharma Prod Novel process
SE9902937D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
SE9902938D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
SE9902935D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
SE9902936D0 (sv) * 1999-08-18 1999-08-18 Astra Pharma Prod Pharmaceutical compositions
DE10063957A1 (de) * 2000-12-20 2002-06-27 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und Dopamin-Agonisten
AR040962A1 (es) * 2002-08-09 2005-04-27 Novartis Ag Compuestos derivados de tiazol 1,3-2-ona, composicion farmaceutica y proceso de preparacion del compuesto
GB0218629D0 (en) * 2002-08-09 2002-09-18 Novartis Ag Organic compounds
CA2543858C (en) 2003-11-21 2014-04-15 Theravance, Inc. Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity
GB0426164D0 (en) 2004-11-29 2004-12-29 Novartis Ag Organic compounds
TW200738658A (en) 2005-08-09 2007-10-16 Astrazeneca Ab Novel compounds
TW200738659A (en) * 2005-08-29 2007-10-16 Astrazeneca Ab Novel compounds
TW200745067A (en) 2006-03-14 2007-12-16 Astrazeneca Ab Novel compounds
RU2455295C2 (ru) * 2006-12-20 2012-07-10 АстраЗенека AБ 4-ГИДРОКСИ-2-ОКСО-2,3-ДИГИДРО-1,3-БЕНЗОТИАЗОЛ-7-ИЛЬНЫЕ СОЕДИНЕНИЯ ДЛЯ МОДУЛЯЦИИ β2-АДРЕНОРЕЦЕПТОРНОЙ АКТИВНОСТИ
TW200833670A (en) 2006-12-20 2008-08-16 Astrazeneca Ab Novel compounds 569
GB0702458D0 (en) 2007-02-08 2007-03-21 Astrazeneca Ab Salts 668
GB0704000D0 (en) * 2007-03-01 2007-04-11 Astrazeneca Ab Salts 670
KR20110017456A (ko) 2008-06-18 2011-02-21 아스트라제네카 아베 호흡기 장애의 치료를 위한 베타2-아드레날린성 수용체 효능제로서 작용하는 벤족사지논 유도체
CN102977050B (zh) * 2012-11-20 2015-04-22 浙江工业大学 一种2-苯并噻唑二甲缩醛和2-苯并噻唑甲醛的合成方法
CN106748930B (zh) * 2016-12-05 2019-03-15 三门峡奥科化工有限公司 3-巯基-1-丙醇的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
IE914003A1 (en) * 1990-11-20 1992-05-20 Astra Pharma Prod Biologically Active Amines

Also Published As

Publication number Publication date
WO1993024473A1 (en) 1993-12-09
PH31453A (en) 1998-11-03
DK0649418T3 (da) 1999-07-12
AU675649B2 (en) 1997-02-13
MY131193A (en) 2007-07-31
NO944509D0 (no) 1994-11-24
SK143394A3 (en) 1995-06-07
CA2136553C (en) 2000-08-15
ZA933648B (en) 1993-11-25
NZ253190A (en) 1995-12-21
CN1085899A (zh) 1994-04-27
CN1036393C (zh) 1997-11-12
NO944509L (no) 1994-11-24
HU9403387D0 (en) 1995-02-28
LV12443B (en) 2000-06-20
CZ286905B6 (en) 2000-08-16
CA2136553A1 (en) 1993-12-09
SG48068A1 (en) 1998-04-17
IL105801A (en) 1997-01-10
UA27901C2 (uk) 2000-10-16
IL105801A0 (en) 1993-09-22
PL172807B1 (pl) 1997-11-28
ES2123652T3 (es) 1999-01-16
FI945538A0 (fi) 1994-11-25
GB9211172D0 (en) 1992-07-08
RU2114108C1 (ru) 1998-06-27
DZ1694A1 (fr) 2002-02-17
DE69321835D1 (de) 1998-12-03
FI945538A (fi) 1994-11-25
AU4334393A (en) 1993-12-30
KR100279132B1 (ko) 2001-01-15
LV12443A (en) 2000-03-20
HUT71124A (en) 1995-11-28
TW368501B (en) 1999-09-01
HU211947A9 (en) 1996-01-29
RU94046093A (ru) 1996-09-27
EP0649418A1 (en) 1995-04-26
DE69321835T2 (de) 1999-05-12
NO304739B1 (no) 1999-02-08
PL172904B1 (pl) 1997-12-31
MA22895A1 (fr) 1993-12-31
JPH08503923A (ja) 1996-04-30
SK281282B6 (sk) 2001-02-12
JP3094452B2 (ja) 2000-10-03
CZ291694A3 (en) 1995-03-15
EP0649418B1 (en) 1998-10-28
ATE172726T1 (de) 1998-11-15

Similar Documents

Publication Publication Date Title
ES2123652T3 (es) 7-(2-aminoetil)-benzotiazolonas.
HUP0101999A2 (hu) 4-Hidroxi-kinolin-3-karboxamid- és -hidrazid-származékok, ezeket tartalmazó gyógyászati készítmények, valamint e vegyületek alkalmazása
DK0683789T3 (da) N-alkyl-2-substituerede ATP-analoger
FI913478A0 (fi) Diazinderivat.
NO882036D0 (no) Fremgangsmaate for fremstilling av terapeutisk aktive heterocykliske ketoner.
NO304379B1 (no) 11,21-bisfenyl-19-norpregnan-derivater, anvendelse derav og farmas°ytiske preparater inneholdende slike derivater
DK0587088T3 (da) Substituerede cyclohexan-derivater, fremgangsmåde til deres fremstilling og anvendelsen af forbindelserne til behandling af sygdomme
ATE170852T1 (de) Benzolsulfonamid-derivate zur behandlung der blaseninstabilität
DK0446141T3 (da) Imidazo(1,2-c)quinazolinderivater og fremgangsmåde til fremstilling deraf samt farmaceutiske midler indeholdende dem
DE69330601D1 (de) Serotoninergische ergolin derivate
DK283984D0 (da) Benzodiazepinderivater og fremgangsmaade til fremstilling deraf
DE69619088D1 (de) Quinoxalin-Derivate zur Behandlung von Tinnitus
ATE1585T1 (de) Clavulansaeurederivate, ihre herstellung und sie enthaltende pharmazeutische praeparate.

Legal Events

Date Code Title Description
FG Grant or registration
GB Transfer or rights
PD Change of proprietorship

Owner name: ASTRAZENECA AB

MM Annulment or lapse due to non-payment of fees