MX376118B - Formulaciones inyectables fisiológicamente balanceadas de fosnetupitant. - Google Patents

Formulaciones inyectables fisiológicamente balanceadas de fosnetupitant.

Info

Publication number
MX376118B
MX376118B MX2018015036A MX2018015036A MX376118B MX 376118 B MX376118 B MX 376118B MX 2018015036 A MX2018015036 A MX 2018015036A MX 2018015036 A MX2018015036 A MX 2018015036A MX 376118 B MX376118 B MX 376118B
Authority
MX
Mexico
Prior art keywords
fosnetupitant
physiologically balanced
injectable formulations
balanced injectable
formulations
Prior art date
Application number
MX2018015036A
Other languages
English (en)
Spanish (es)
Other versions
MX2018015036A (es
Inventor
Alessio Venturini
Roberta Cannella
Original Assignee
Helsinn Healthcare Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=59055193&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX376118(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Helsinn Healthcare Sa filed Critical Helsinn Healthcare Sa
Publication of MX2018015036A publication Critical patent/MX2018015036A/es
Publication of MX376118B publication Critical patent/MX376118B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/473Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2018015036A 2016-06-06 2017-06-01 Formulaciones inyectables fisiológicamente balanceadas de fosnetupitant. MX376118B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662345942P 2016-06-06 2016-06-06
PCT/EP2017/063268 WO2017211663A1 (en) 2016-06-06 2017-06-01 Physiologically balanced injectable formulations of fosnetupitant

Publications (2)

Publication Number Publication Date
MX2018015036A MX2018015036A (es) 2019-04-11
MX376118B true MX376118B (es) 2025-03-07

Family

ID=59055193

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018015036A MX376118B (es) 2016-06-06 2017-06-01 Formulaciones inyectables fisiológicamente balanceadas de fosnetupitant.

Country Status (36)

Country Link
US (4) US10624911B2 (enExample)
EP (2) EP3435980B1 (enExample)
JP (2) JP6936817B2 (enExample)
KR (1) KR102459416B1 (enExample)
CN (1) CN109310627B (enExample)
AR (1) AR108676A1 (enExample)
AU (1) AU2017276588B2 (enExample)
BR (1) BR112018074655B1 (enExample)
CA (1) CA3025837C (enExample)
CL (1) CL2018003338A1 (enExample)
CO (1) CO2018011686A2 (enExample)
CY (1) CY1122755T1 (enExample)
DK (1) DK3435980T3 (enExample)
EA (1) EA036605B1 (enExample)
EC (1) ECSP19000169A (enExample)
ES (1) ES2771226T3 (enExample)
HR (1) HRP20200196T1 (enExample)
IL (1) IL263126B (enExample)
JO (1) JOP20170137B1 (enExample)
LT (1) LT3435980T (enExample)
MA (1) MA44513B1 (enExample)
MD (1) MD3435980T2 (enExample)
MX (1) MX376118B (enExample)
MY (1) MY194081A (enExample)
PE (1) PE20190347A1 (enExample)
PH (1) PH12018502524B1 (enExample)
PL (1) PL3435980T3 (enExample)
PT (1) PT3435980T (enExample)
RS (1) RS59852B1 (enExample)
SG (1) SG11201809708PA (enExample)
SI (1) SI3435980T1 (enExample)
TW (1) TWI725191B (enExample)
UA (1) UA122285C2 (enExample)
UY (1) UY37273A (enExample)
WO (1) WO2017211663A1 (enExample)
ZA (1) ZA201807932B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11654154B2 (en) 2019-01-29 2023-05-23 Navinta Iii Inc Process for preparing injectable Fosaprepitant Dimeglumine compositions having improved storage stability
US12097197B2 (en) 2021-12-21 2024-09-24 Slayback Pharma Llc Stable liquid compositions of netupitant and palonosetron
JP7783403B2 (ja) * 2022-03-23 2025-12-09 大鵬薬品工業株式会社 ホスネツピタント又はその医薬上許容される塩の安定化製剤およびその製造方法
WO2025036703A1 (en) * 2023-08-13 2025-02-20 Helsinn Healthcare Sa Fosnetupitant for administration via intravenous bolus
WO2025056094A1 (zh) * 2023-09-15 2025-03-20 广州帝奇医药技术有限公司 一种冻干制剂和注射液及其制备方法
CN119185243A (zh) * 2024-11-28 2024-12-27 山东齐都药业有限公司 福奈妥匹坦帕洛诺司琼口服掩味颗粒剂及其制备方法与应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL111960A (en) 1993-12-17 1999-12-22 Merck & Co Inc Morpholines and thiomorpholines their preparation and pharmaceutical compositions containing them
KR100286412B1 (ko) 1993-12-29 2001-04-16 더블유. 지. 콜 치환된 모르폴린 유도체, 이의 제조방법 및 이를 포함하는 약제학적 조성물
IL112778A0 (en) 1994-03-04 1995-05-26 Merck & Co Inc Substituted heterocycles, their preparation and pharmaceutical compositions containing them
JO2735B1 (en) * 2003-01-30 2013-09-15 هيلسين هيلث كير أس ايه. Liquid pharmaceutical formations of balloonosterone
US20060167072A1 (en) * 2004-01-30 2006-07-27 Helsinn Healthcare Sa Liquid pharmaceutical formulations of palonosetron
US20100048607A1 (en) * 2008-08-25 2010-02-25 Chandrashekhar Kocherlakota Formulations comprising palonosetron
US8426450B1 (en) 2011-11-29 2013-04-23 Helsinn Healthcare Sa Substituted 4-phenyl pyridines having anti-emetic effect
EP2866797B1 (en) * 2012-07-06 2020-04-29 Pharmathen S.A. Stable injectable pharmaceutical composition of neurokinin 1 receptor antagonist and process for preparation thereof

Also Published As

Publication number Publication date
CL2018003338A1 (es) 2019-02-22
EA201892837A1 (ru) 2019-06-28
RS59852B1 (sr) 2020-02-28
BR112018074655A2 (pt) 2019-03-06
LT3435980T (lt) 2020-02-25
CN109310627B (zh) 2021-12-14
EP3435980A1 (en) 2019-02-06
MY194081A (en) 2022-11-11
SI3435980T1 (sl) 2020-03-31
US12208109B2 (en) 2025-01-28
PL3435980T3 (pl) 2020-05-18
US11529362B2 (en) 2022-12-20
PT3435980T (pt) 2020-02-21
US20230172953A1 (en) 2023-06-08
WO2017211663A1 (en) 2017-12-14
DK3435980T3 (da) 2020-02-24
MD3435980T2 (ro) 2020-03-31
IL263126B (en) 2021-04-29
SG11201809708PA (en) 2018-11-29
JOP20170137B1 (ar) 2021-08-17
NZ747865A (en) 2024-05-31
KR20190015276A (ko) 2019-02-13
EP3435980B1 (en) 2019-11-13
PE20190347A1 (es) 2019-03-07
IL263126A (en) 2018-12-31
TW201801727A (zh) 2018-01-16
UA122285C2 (uk) 2020-10-12
JP2019521102A (ja) 2019-07-25
CY1122755T1 (el) 2021-03-12
KR102459416B1 (ko) 2022-10-27
CO2018011686A2 (es) 2019-02-08
JP6936817B2 (ja) 2021-09-22
PH12018502524A1 (en) 2019-10-14
US10624911B2 (en) 2020-04-21
ES2771226T3 (es) 2020-07-06
BR112018074655B1 (pt) 2024-02-15
UY37273A (es) 2018-01-31
EP3626231A1 (en) 2020-03-25
CN109310627A (zh) 2019-02-05
MX2018015036A (es) 2019-04-11
MA44513B1 (fr) 2020-02-28
AU2017276588A1 (en) 2018-11-22
ZA201807932B (en) 2019-08-28
HRP20200196T1 (hr) 2020-05-01
CA3025837C (en) 2024-02-13
CA3025837A1 (en) 2017-12-14
TWI725191B (zh) 2021-04-21
AU2017276588B2 (en) 2022-06-02
PH12018502524B1 (en) 2022-04-27
JP2021183639A (ja) 2021-12-02
US20170348335A1 (en) 2017-12-07
US20250235473A1 (en) 2025-07-24
EA036605B1 (ru) 2020-11-27
JP7223084B2 (ja) 2023-02-15
ECSP19000169A (es) 2019-01-31
US20200206249A1 (en) 2020-07-02
AR108676A1 (es) 2018-09-12

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