MX360857B - Régimen de dosificación para inhibidores de janus quinasa (jak). - Google Patents

Régimen de dosificación para inhibidores de janus quinasa (jak).

Info

Publication number
MX360857B
MX360857B MX2015000871A MX2015000871A MX360857B MX 360857 B MX360857 B MX 360857B MX 2015000871 A MX2015000871 A MX 2015000871A MX 2015000871 A MX2015000871 A MX 2015000871A MX 360857 B MX360857 B MX 360857B
Authority
MX
Mexico
Prior art keywords
jak
janus
mammal
dosage regime
quinasa
Prior art date
Application number
MX2015000871A
Other languages
English (en)
Spanish (es)
Other versions
MX2015000871A (es
Inventor
Andrea J Gonzales
Sallie B Cosgrove
Phyllis B Malpas
Michael Rolf Stegemann
Wendy Turner Collard
Original Assignee
Zoetis Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48901189&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX360857(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Zoetis Llc filed Critical Zoetis Llc
Publication of MX2015000871A publication Critical patent/MX2015000871A/es
Publication of MX360857B publication Critical patent/MX360857B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
MX2015000871A 2012-07-20 2013-07-18 Régimen de dosificación para inhibidores de janus quinasa (jak). MX360857B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261674289P 2012-07-20 2012-07-20
US201361815803P 2013-04-25 2013-04-25
PCT/US2013/051015 WO2014015107A1 (en) 2012-07-20 2013-07-18 Dosing regimen for janus kinase (jak) inhibitors

Publications (2)

Publication Number Publication Date
MX2015000871A MX2015000871A (es) 2015-05-07
MX360857B true MX360857B (es) 2018-11-20

Family

ID=48901189

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015000871A MX360857B (es) 2012-07-20 2013-07-18 Régimen de dosificación para inhibidores de janus quinasa (jak).

Country Status (25)

Country Link
US (1) US9522151B2 (https=)
EP (1) EP2874630B1 (https=)
JP (2) JP6022063B2 (https=)
KR (2) KR20150028299A (https=)
CN (2) CN104470525A (https=)
AU (1) AU2013292547B2 (https=)
BR (1) BR112015000808A2 (https=)
CA (1) CA2878867C (https=)
CY (1) CY1121436T1 (https=)
DK (1) DK2874630T3 (https=)
ES (1) ES2707627T3 (https=)
HK (2) HK1209314A1 (https=)
HR (1) HRP20182088T1 (https=)
HU (1) HUE042771T2 (https=)
IN (1) IN2015DN00370A (https=)
LT (1) LT2874630T (https=)
MX (1) MX360857B (https=)
NZ (1) NZ703152A (https=)
PL (1) PL2874630T3 (https=)
PT (1) PT2874630T (https=)
RS (1) RS58242B1 (https=)
SI (1) SI2874630T1 (https=)
SM (1) SMT201900044T1 (https=)
WO (1) WO2014015107A1 (https=)
ZA (1) ZA201500134B (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CU24275B1 (es) 2013-02-22 2017-10-05 Pfizer Derivados de cicloalquilo pirrolo [2,3-d] pirimidina-4-il amino útiles como inhibidores de quinasas janus relacionadas y composiciones farmacéuticas que contienen tales compuestos
EP3180344B1 (en) 2014-08-12 2019-09-18 Pfizer Inc Pyrrolo[2,3-d]pyrimidine derivatives useful for inhibiting janus kinase
US11780848B2 (en) 2015-10-16 2023-10-10 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1- carboxamide and solid state forms thereof
EP3362455A1 (en) 2015-10-16 2018-08-22 AbbVie Inc. PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF
US11365198B2 (en) 2015-10-16 2022-06-21 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
US12365689B2 (en) 2015-10-16 2025-07-22 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
US10550126B2 (en) 2015-10-16 2020-02-04 Abbvie Inc. Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-A]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof
WO2017143014A1 (en) * 2016-02-16 2017-08-24 Brian Kim Jak inhibitors and uses thereof
CN107098908B (zh) * 2016-02-23 2021-01-08 欣凯医药科技(上海)有限公司 一种吡咯并嘧啶类化合物的制备方法和应用
KR102195348B1 (ko) 2018-11-15 2020-12-24 에이치케이이노엔 주식회사 단백질 키나제 억제제로서의 신규 화합물 및 이를 포함하는 약제학적 조성물
WO2020155931A1 (zh) 2019-01-30 2020-08-06 格格巫（珠海）生物科技有限公司 一种jak抑制剂及其制备方法
US11992490B2 (en) 2019-10-16 2024-05-28 Incyte Corporation Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP)
CN117242080A (zh) 2020-12-18 2023-12-15 勃林格殷格翰动物保健美国公司 含硼吡唑化合物、包括其的组合物、其方法和用途
EP4310085A4 (en) * 2021-03-16 2025-09-24 Hk Inno N Corp NOVEL SALTS OF HETEROCYCLIC COMPOUND AS PROTEIN KINASE INHIBITOR AND USES THEREOF
CN117136059A (zh) * 2021-04-22 2023-11-28 深圳微芯生物科技股份有限公司 包含jak3/jak1/tbk1选择性抑制剂的药物组合物及其医药用途
WO2024259429A2 (en) * 2023-06-16 2024-12-19 The University Of Chicago Methods and compositions for pharmaceutically relevant interactions

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9911365A (pt) * 1998-06-19 2001-03-13 Pfizer Prod Inc Compostos pirrolo[2,3-d]pirimidina
JP4884570B2 (ja) * 2008-08-20 2012-02-29 ファイザー・インク ピロロ［２，３−ｄ］ピリミジン化合物

Also Published As

Publication number Publication date
HK1209314A1 (en) 2016-04-01
CY1121436T1 (el) 2020-05-29
PL2874630T3 (pl) 2019-04-30
AU2013292547A1 (en) 2015-01-22
AU2013292547B2 (en) 2017-05-04
ZA201500134B (en) 2016-08-31
RS58242B1 (sr) 2019-03-29
WO2014015107A1 (en) 2014-01-23
US9522151B2 (en) 2016-12-20
JP6022063B2 (ja) 2016-11-09
NZ703152A (en) 2016-03-31
US20150126535A1 (en) 2015-05-07
KR20170034949A (ko) 2017-03-29
SI2874630T1 (sl) 2019-04-30
ES2707627T3 (es) 2019-04-04
IN2015DN00370A (https=) 2015-06-12
PT2874630T (pt) 2019-01-31
DK2874630T3 (en) 2019-01-28
JP2015522620A (ja) 2015-08-06
BR112015000808A2 (pt) 2017-06-27
HK1252083A1 (zh) 2019-05-17
SMT201900044T1 (it) 2019-02-28
HRP20182088T1 (hr) 2019-02-08
HUE042771T2 (hu) 2019-07-29
EP2874630A1 (en) 2015-05-27
CA2878867C (en) 2018-01-09
CN108354938A (zh) 2018-08-03
MX2015000871A (es) 2015-05-07
CN104470525A (zh) 2015-03-25
CA2878867A1 (en) 2014-01-23
EP2874630B1 (en) 2018-12-05
JP2017019816A (ja) 2017-01-26
LT2874630T (lt) 2019-02-11
KR20150028299A (ko) 2015-03-13

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