MX357888B - Sales basicas de adicion de nitroxolina y usos de las mismas. - Google Patents

Sales basicas de adicion de nitroxolina y usos de las mismas.

Info

Publication number
MX357888B
MX357888B MX2015012720A MX2015012720A MX357888B MX 357888 B MX357888 B MX 357888B MX 2015012720 A MX2015012720 A MX 2015012720A MX 2015012720 A MX2015012720 A MX 2015012720A MX 357888 B MX357888 B MX 357888B
Authority
MX
Mexico
Prior art keywords
nitroxoline
addition salts
base addition
pharmaceutical compositions
methods
Prior art date
Application number
MX2015012720A
Other languages
English (en)
Spanish (es)
Other versions
MX2015012720A (es
Inventor
Ke Pan
Original Assignee
Asieris Pharmaceutical Tech Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asieris Pharmaceutical Tech Co Ltd filed Critical Asieris Pharmaceutical Tech Co Ltd
Publication of MX2015012720A publication Critical patent/MX2015012720A/es
Publication of MX357888B publication Critical patent/MX357888B/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/24Oxygen atoms attached in position 8

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
MX2015012720A 2013-03-15 2014-03-17 Sales basicas de adicion de nitroxolina y usos de las mismas. MX357888B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361790059P 2013-03-15 2013-03-15
PCT/US2014/030532 WO2014145723A1 (en) 2013-03-15 2014-03-17 Base addition salts of nitroxoline and uses thereof

Publications (2)

Publication Number Publication Date
MX2015012720A MX2015012720A (es) 2016-06-21
MX357888B true MX357888B (es) 2018-07-27

Family

ID=51538074

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015012720A MX357888B (es) 2013-03-15 2014-03-17 Sales basicas de adicion de nitroxolina y usos de las mismas.

Country Status (11)

Country Link
US (1) US9758484B2 (enAn)
EP (1) EP2970128B1 (enAn)
JP (1) JP6273349B2 (enAn)
KR (1) KR20160021077A (enAn)
CN (1) CN105228984B (enAn)
AU (2) AU2014232722B2 (enAn)
BR (1) BR112015022849B1 (enAn)
CA (1) CA2907338C (enAn)
ES (1) ES2766758T3 (enAn)
MX (1) MX357888B (enAn)
WO (1) WO2014145723A1 (enAn)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6869324B2 (ja) 2016-03-31 2021-05-12 チャンスー ヤホン メディテック カンパニー リミテッド ニトロキソリンおよびその類似体と、化学療法剤および免疫療法剤との、がんの治療における、組合せの使用
CA3113463A1 (en) * 2018-09-29 2020-04-02 Jiangsu Yahong Meditech Co., Ltd. Nitroxoline prodrug and use thereof
CN112402388A (zh) 2019-08-05 2021-02-26 江苏亚虹医药科技股份有限公司 一种用于治疗膀胱癌的口服固体制剂及其制备方法
US20230000853A1 (en) * 2019-12-31 2023-01-05 Jiangsu Yahong Meditech Co., Ltd. Pharmaceutical composition containing nitroxoline, nitroxoline tablet, preparation method therefor and use thereof
CN111773193A (zh) * 2020-07-03 2020-10-16 江苏亚虹医药科技有限公司 含硝羟喹啉赖氨酸盐的药物组合物及其制备方法和用途
CN111960998A (zh) * 2020-08-03 2020-11-20 江苏亚虹医药科技有限公司 硝羟喹啉衍生物及其制备方法和用途

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2745834A (en) * 1953-02-09 1956-05-15 Phillips Petroleum Co Stabilization of certain vinyl-pyridines, vinyl quinolines and vinyl-isoquinolines
US2745832A (en) * 1954-03-08 1956-05-15 Nuodex Products Co Inc Metal quinolinolates and methods of making the same
US3872128A (en) 1972-03-08 1975-03-18 Union Carbide Corp Antimicrobial hydroxy quinoline, ethylene-acrylic polymer compositions
JPS5768831A (en) 1980-10-17 1982-04-27 Fuji Photo Film Co Ltd Heat developable photosensitive material
JPS57101835A (en) 1980-12-17 1982-06-24 Fuji Photo Film Co Ltd Thermodevelopable photosensitive material
US4329185A (en) * 1981-01-21 1982-05-11 Dso "Pharmachim" Method for the preparation of a biologically active polyamide net
US5242892A (en) * 1984-07-27 1993-09-07 The Board Of Trustees Of The University Of Illinois Chlorophyll biosynthesis modulators
JPH03284734A (ja) 1990-03-31 1991-12-16 Toshiba Corp 有機非線形光学材料
IT1317735B1 (it) 2000-01-26 2003-07-15 Nicox Sa Sali di agenti antimicrobici.
EP1694652A1 (en) * 2003-12-19 2006-08-30 Rigel Pharmaceuticals, Inc. Stereoisomers and stereoisomeric mixtures of 1-(2,4-pyrimidinediamino)-2-cyclopentanecarboxamide synthetic intermediates
TWI328006B (en) * 2003-12-26 2010-08-01 Nissan Chemical Ind Ltd Crystal form of quinoline compound and process for its production
WO2006117660A2 (en) 2005-05-04 2006-11-09 Clio Pharmaceutical Corporation Method for treating cancer, coronary, inflammatory and macular disease, combining the modulation of zinc- and/or copper dependent proteins
KR101524636B1 (ko) 2005-05-11 2015-06-03 에테하 취리히 원핵 세포로부터의 재조합 n-글리코실화 단백질
EP1892248A1 (en) 2006-08-21 2008-02-27 Eidgenössische Technische Hochschule Zürich Specific and high affinity binding proteins comprising modified SH3 domains of FYN kinase
EP2350012B1 (en) * 2008-10-06 2017-06-28 The Johns Hopkins University Quinoline compounds as inhibitors of angiogenesis, human methionine aminopeptidase, and sirt1, and methods of treating disorders
WO2010136105A2 (en) 2009-05-28 2010-12-02 Merck Patent Gmbh Ammoniumcarboxylates
JP2010070557A (ja) 2009-12-17 2010-04-02 Anacor Pharmaceuticals Inc 加水分解抵抗性ホウ素含有治療薬および使用法
EP2353599A1 (en) 2010-01-28 2011-08-10 University of Ljubljana 8-hydroxyquinolines as inhibitors of cathepsin B
DK2730123T3 (da) * 2011-07-07 2020-03-02 Ericsson Telefon Ab L M Overleveringsbeslutning i betjenende basisstation baseret på en første og anden type mobilitetsmekanisme

Also Published As

Publication number Publication date
MX2015012720A (es) 2016-06-21
EP2970128A1 (en) 2016-01-20
CA2907338A1 (en) 2014-09-18
AU2014232722B2 (en) 2017-03-09
CN105228984B (zh) 2018-03-23
JP6273349B2 (ja) 2018-01-31
JP2016514705A (ja) 2016-05-23
AU2014232722A1 (en) 2015-09-24
US9758484B2 (en) 2017-09-12
CA2907338C (en) 2019-09-17
KR20160021077A (ko) 2016-02-24
BR112015022849A2 (pt) 2017-12-26
AU2017200820A1 (en) 2017-03-02
BR112015022849B1 (pt) 2020-02-18
ES2766758T3 (es) 2020-06-15
EP2970128A4 (en) 2016-11-30
EP2970128B1 (en) 2019-12-04
CN105228984A (zh) 2016-01-06
WO2014145723A1 (en) 2014-09-18
US20160031819A1 (en) 2016-02-04
HK1214589A1 (zh) 2016-07-29

Similar Documents

Publication Publication Date Title
PH12017501956A1 (en) Compositions of obeticholic acid and methods of use
MX2021007268A (es) Formas solidas de acido {[5-(3-clorofenil)-3-hidroxipiridin-2-carb onil]amino}acetico, composiciones, y usos de las mismas.
IN2015DN01156A (enAn)
MX392026B (es) Compuestos heterocíclicos como inmunomoduladores.
MX2015012502A (es) Inhibidores de proteina cinasa dependiente de adn.
SG10201909545XA (en) Bile acid derivatives as fxr/tgr5 agonists and methods of use thereof
MD4800B1 (ro) Compuşi de aminopirimidinil ca inhibitori de JAK
IN2014DN09434A (enAn)
MX2016002544A (es) Compuestos utiles como inmunomoduladores.
PH12016500105A1 (en) Sulfonamides as modulators of sodium channels
MX2015010125A (es) Derivados de piridazinona-amidas.
MX363457B (es) Compuestos de sulfonamida heterociclica sustituida utiles como moduladores del canal del receptor de potencial transitorio a1 (trpa1).
WO2014028600A3 (en) 3-AMINOCYCLOALKYL COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF
IN2014KN02601A (enAn)
MY181602A (en) Isochromene derivatives as phosphoinositide 3-kinases inhibitors
EA201591406A1 (ru) C-19 модифицированные тритерпеноиды с ингибиторной активностью созревания вич
NZ719169A (en) Heteroaryl butanoic acid derivatives as lta4h inhibitors
MX357888B (es) Sales basicas de adicion de nitroxolina y usos de las mismas.
MX2018001733A (es) Compuestos heterocíclicos de fumagillol y métodos de elaboración y uso de los mismos.
EA032271B9 (ru) Вещества, фармацевтическая композиция и методы применения при лечении воспалительных заболеваний
MD20170011A2 (ro) Compuşi imidazopiridazinici
WO2016029136A8 (en) 3-amidobenzamides and uses thereof for increasing cellular levels of a3g
MX2013002208A (es) Derivados de sulfonilpiperazina que interactuan con la proteina reguladora de glucocinasa para el tratamiento de diabetes.
EA201591704A1 (ru) Новые устойчивые соли пентадекапептида, способ их получения, их применение в производстве фармацевтических составов и их применение в терапии
WO2019040105A3 (en) COMPOUNDS, SALTS THEREOF AND METHODS FOR THE TREATMENT OF DISEASES

Legal Events

Date Code Title Description
FG Grant or registration