MX357352B - Uso de derivados poliaminoisoprenilo en un tratamiento antibiotico o antiseptico. - Google Patents

Uso de derivados poliaminoisoprenilo en un tratamiento antibiotico o antiseptico.

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Publication number
MX357352B
MX357352B MX2013009721A MX2013009721A MX357352B MX 357352 B MX357352 B MX 357352B MX 2013009721 A MX2013009721 A MX 2013009721A MX 2013009721 A MX2013009721 A MX 2013009721A MX 357352 B MX357352 B MX 357352B
Authority
MX
Mexico
Prior art keywords
antibiotic
antiseptic treatment
polyaminoisoprenilo
derivatives
polyaminoisoprenylderivatives
Prior art date
Application number
MX2013009721A
Other languages
English (en)
Other versions
MX2013009721A (es
Inventor
Bolla Jean-Michel
Michel Brunel Jean
Lorenzi Vannina
Berti Liliane
Pierre Félix Casanova Joseph
Original Assignee
Univ Aix Marseille
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Aix Marseille filed Critical Univ Aix Marseille
Publication of MX2013009721A publication Critical patent/MX2013009721A/es
Publication of MX357352B publication Critical patent/MX357352B/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/20—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton
    • C07C211/22—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton containing at least two amino groups bound to the carbon skeleton
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    • A01N33/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic nitrogen compounds
    • A01N33/02—Amines; Quaternary ammonium compounds
    • A—HUMAN NECESSITIES
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    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
    • A—HUMAN NECESSITIES
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    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • A—HUMAN NECESSITIES
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    • A01N43/84—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms six-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,4
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A61K31/431—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems containing further heterocyclic rings, e.g. ticarcillin, azlocillin, oxacillin
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/145—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/15—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
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  • Wood Science & Technology (AREA)
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  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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Abstract

La presente invención se relaciona con el uso de derivados de poliaminoisoprenilo en un tratamiento antibiótico o antiséptico de bacterias que incluyen aquellas que presentan resistencia a múltiples fármacos (MDR), en particular como inhibidores de bomba de descarga. También se relaciona con derivados novedosos de poliaminoisoprenilo, las composiciones que comprenden los mismos, el proceso para preparar los mismos, y el uso de los mismos en tratamiento antibiótico o antiséptico.
MX2013009721A 2011-02-23 2012-02-23 Uso de derivados poliaminoisoprenilo en un tratamiento antibiotico o antiseptico. MX357352B (es)

Applications Claiming Priority (2)

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EP11305193 2011-02-23
PCT/EP2012/053113 WO2012113891A1 (en) 2011-02-23 2012-02-23 Use of polyaminoisoprenyl derivatives in antibiotic or antiseptic treatment

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MX357352B true MX357352B (es) 2018-07-05

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JP (1) JP2014513670A (es)
CN (1) CN103492358A (es)
BR (1) BR112013021518A2 (es)
CA (1) CA2827578A1 (es)
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MX (1) MX357352B (es)
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WO2017125912A1 (en) * 2016-01-21 2017-07-27 Dexcel Pharma Technologies Ltd. Methods for treating helicobacter infection
KR101749687B1 (ko) 2016-04-25 2017-06-21 경북대학교 산학협력단 7,10-에폭시옥타데카-7,9-다이에노산을 유효성분으로 포함하는 항균 조성물
US10695314B2 (en) 2016-04-25 2020-06-30 Kyungpook National University Industry-Academic Cooperation Foundation Antimicrobial composition containing 7,10-epoxyoctadeca-7,9-dienoic acid as active ingredient
KR101792239B1 (ko) 2016-11-01 2017-10-31 경북대학교 산학협력단 7,10-에폭시옥타데카-7,9-다이에노산 및 항생제를 유효성분으로 포함하는 항균 조성물
AR111430A1 (es) * 2017-05-01 2019-07-10 Sumitomo Chemical Co Método para controlar la enfermedad de plantas resistente a múltiples fármacos de tipo eflujo

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US3429970A (en) 1961-02-02 1969-02-25 Hoffmann La Roche Method of hindering the metamorphosis and reproduction of arthropodes
US3808339A (en) * 1969-07-22 1974-04-30 Scm Corp Insect repellent compositions and process containing n-(dialkylaminoalkoxy)alkyl terpenylamine
JPS55129255A (en) * 1979-03-28 1980-10-06 Kuraray Co Ltd Farnesylacetamide compounds or their salts
JPS55129275A (en) * 1979-03-28 1980-10-06 Kuraray Co Ltd Farnesylacetic acid amide bearing piperazine ring or its salt
JPS57192340A (en) * 1981-05-18 1982-11-26 Nisshin Flour Milling Co Ltd Isoprenylamine derivative
JPS59101448A (ja) 1982-11-30 1984-06-12 Eisai Co Ltd ポリプレニルカルボン酸アミドおよびその製造方法ならびにそれを含有する医薬
JPS60123451A (ja) * 1983-12-07 1985-07-02 Eisai Co Ltd ポリプレニル系化合物およびその製造方法ならびにそれを含有する医薬
JPS63307849A (ja) 1987-06-09 1988-12-15 Yamanouchi Pharmaceut Co Ltd スペルミン誘導体
JPH0418056A (ja) * 1990-05-09 1992-01-22 Sanwa Kagaku Kenkyusho Co Ltd ポリイソプレン化合物及びその塩、これ等の製法並びにこれ等を有効成分とする消化性潰瘍治療剤
US6951961B2 (en) 2002-05-17 2005-10-04 Marina Nikolaevna Protopopova Methods of use and compositions for the diagnosis and treatment of infectious disease
US20040033986A1 (en) 2002-05-17 2004-02-19 Protopopova Marina Nikolaevna Anti tubercular drug: compositions and methods
EP2184061A1 (en) 2008-11-07 2010-05-12 Universite de Corse Genariol as bacterial efflux pump inhibitor

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WO2012113891A1 (en) 2012-08-30
MX2013009721A (es) 2014-01-31
PL2678307T3 (pl) 2018-11-30
US10562842B2 (en) 2020-02-18
US20140128335A1 (en) 2014-05-08
US20170015617A1 (en) 2017-01-19
CN103492358A (zh) 2014-01-01
BR112013021518A2 (pt) 2020-09-29
CA2827578A1 (en) 2012-08-30
EP2678307B1 (en) 2018-04-04
ES2675356T3 (es) 2018-07-10
JP2014513670A (ja) 2014-06-05
US9464032B2 (en) 2016-10-11
EP2678307A1 (en) 2014-01-01
ZA201307058B (en) 2015-08-26

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