MX347841B - Procedimiento para preparar derivados de antranilamida sustituidos con tetrazoles y polimorfos cristalinos novedosos de estos derivados. - Google Patents
Procedimiento para preparar derivados de antranilamida sustituidos con tetrazoles y polimorfos cristalinos novedosos de estos derivados.Info
- Publication number
- MX347841B MX347841B MX2015009721A MX2015009721A MX347841B MX 347841 B MX347841 B MX 347841B MX 2015009721 A MX2015009721 A MX 2015009721A MX 2015009721 A MX2015009721 A MX 2015009721A MX 347841 B MX347841 B MX 347841B
- Authority
- MX
- Mexico
- Prior art keywords
- derivatives
- novel crystal
- crystal polymorph
- preparing tetrazole
- substituted anthranilamide
- Prior art date
Links
- 239000013078 crystal Substances 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- -1 tetrazole-substituted anthranilamide Chemical class 0.000 title abstract 2
- 239000003905 agrochemical Substances 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/713—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with four or more nitrogen atoms as the only ring hetero atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Dentistry (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pretreatment Of Seeds And Plants (AREA)
- Catching Or Destruction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a un procedimiento para preparar derivados de antranilamida sustituidos con tetrazoles de la fórmula (I). (ver Fórmula) en la que R1, R2, R3, R4, R5 y Z son cada uno según se han definido en la descripción, y a un polimorfo cristalino novedoso de estos derivados y al uso de los mismos en formulaciones agroquímicas.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35492010P | 2010-06-15 | 2010-06-15 | |
| EP10166059 | 2010-06-15 | ||
| PCT/EP2011/059735 WO2011157664A1 (de) | 2010-06-15 | 2011-06-10 | Verfahren zur herstellung von tetrazol-substituierten anthranilsäurediamid-derivaten und neue kristalline modifikation dieser derivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX347841B true MX347841B (es) | 2017-05-16 |
Family
ID=42989671
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2015009721A MX347841B (es) | 2010-06-15 | 2011-06-10 | Procedimiento para preparar derivados de antranilamida sustituidos con tetrazoles y polimorfos cristalinos novedosos de estos derivados. |
| MX2012014775A MX2012014775A (es) | 2010-06-15 | 2011-06-10 | Procedimiento para preparar derivados de antranilamia sustituidos con tetrazoles y polimorfos cristalinos novedosos de estos derivados. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2012014775A MX2012014775A (es) | 2010-06-15 | 2011-06-10 | Procedimiento para preparar derivados de antranilamia sustituidos con tetrazoles y polimorfos cristalinos novedosos de estos derivados. |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US8969572B2 (es) |
| EP (2) | EP2582694B1 (es) |
| JP (3) | JP6199739B2 (es) |
| KR (1) | KR101790305B1 (es) |
| CN (1) | CN103261187B (es) |
| BR (1) | BR112012032244A2 (es) |
| DK (2) | DK2955176T3 (es) |
| ES (2) | ES2660305T3 (es) |
| HR (1) | HRP20151088T1 (es) |
| HU (1) | HUE027943T2 (es) |
| MX (2) | MX347841B (es) |
| PL (1) | PL2582694T3 (es) |
| PT (1) | PT2582694E (es) |
| RS (1) | RS54277B1 (es) |
| SI (1) | SI2582694T1 (es) |
| TW (1) | TWI511668B (es) |
| WO (1) | WO2011157664A1 (es) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011157664A1 (de) * | 2010-06-15 | 2011-12-22 | Bayer Cropscience Ag | Verfahren zur herstellung von tetrazol-substituierten anthranilsäurediamid-derivaten und neue kristalline modifikation dieser derivate |
| BR112012032415A2 (pt) * | 2010-06-18 | 2015-09-15 | Bayer Ip Gmbh | combinações de ingrediente ativo que têm propriedade inseticidas e acaricidas. |
| UA111593C2 (uk) * | 2010-07-07 | 2016-05-25 | Баєр Інтеллекчуел Проперті Гмбх | Аміди антранілової кислоти у комбінації з фунгіцидами |
| JP5926253B2 (ja) * | 2010-07-09 | 2016-05-25 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | 有害生物駆除剤としてのアントラニルアミド誘導体 |
| EP2812310A1 (de) * | 2012-02-07 | 2014-12-17 | Bayer Intellectual Property GmbH | Verfahren zur herstellung von substituierten anthranilsäure-derivaten |
| EP2649879A1 (en) | 2012-04-10 | 2013-10-16 | Basf Se | Pesticidal mixtures containing fluxapyroxad |
| WO2013156331A1 (en) | 2012-04-16 | 2013-10-24 | Basf Se | Synergistic compositions comprising pyraclostrobin and an insecticidal compound |
| KR102191469B1 (ko) * | 2013-02-06 | 2020-12-16 | 바이엘 애니멀 헬스 게엠베하 | 해충 방제제로서의 할로겐-치환된 피라졸 유도체 |
| US11297837B2 (en) | 2016-02-19 | 2022-04-12 | Basf Se | Pesticidally activi mixtures comprising anthranilamide compounds |
| TWI679197B (zh) * | 2016-05-05 | 2019-12-11 | 瑞士商伊蘭科動物健康公司 | 雜芳基-1,2,4-三唑及雜芳基-三唑化合物 |
| WO2019123194A1 (en) | 2017-12-20 | 2019-06-27 | Pi Industries Ltd. | Anthranilamides, their use as insecticide and processes for preparing the same. |
| EP3728256B1 (en) | 2017-12-20 | 2024-10-02 | PI Industries Ltd. | Pyrazolopyridine-diamides, their use as insecticide and processes for preparing the same |
| KR102811706B1 (ko) | 2018-01-30 | 2025-05-22 | 피아이 인더스트리스 엘티디. | 새로운 안트라닐아미드, 살충제로서 그의 용도 및 그의 제조 방법 |
| KR102760014B1 (ko) * | 2018-05-21 | 2025-01-24 | 피아이 인더스트리스 엘티디. | 안트라닐산 디아미드의 새로운 제조 방법 |
| CN112469687B (zh) | 2018-07-20 | 2023-10-13 | Pi工业有限公司 | 制备邻甲酰胺基苯甲酰胺类化合物的新方法 |
| CA3129876A1 (en) | 2019-02-18 | 2020-08-27 | Pi Industries Ltd. | A process for preparing anthranilic diamides and intermediates thereof |
| KR102841700B1 (ko) | 2019-02-22 | 2025-08-01 | 피아이 인더스트리스 엘티디. | 안트라닐산 디아미드 화합물 및 그의 중간체의 합성 방법 |
| TWI878337B (zh) * | 2019-08-19 | 2025-04-01 | 美商富曼西公司 | 用於製備3-鹵代-4,5-二氫-1h-吡唑的羧酸衍生物的方法 |
| EP3964506A1 (de) | 2020-09-04 | 2022-03-09 | Bayer Aktiengesellschaft | Verfahren zur herstellung eines tetrazol-substituierten anthranilsäurediamid-derivates |
| CN116670115A (zh) | 2020-09-17 | 2023-08-29 | 皮埃企业有限公司 | 制备邻胺苯甲酸/邻胺苯甲酰胺化合物及其中间产物的方法 |
| AR123593A1 (es) | 2020-09-26 | 2022-12-21 | Pi Industries Ltd | Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos |
| JP2024528002A (ja) | 2021-07-27 | 2024-07-26 | シンジェンタ クロップ プロテクション アクチェンゲゼルシャフト | ジアミド耐性有害生物の防除のための方法及びそのための化合物 |
| WO2023012081A1 (en) | 2021-08-05 | 2023-02-09 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests & compounds therefor |
| MX2024002008A (es) | 2021-08-19 | 2024-03-05 | Syngenta Crop Protection Ag | Metodo para controlar plagas resistentes a diamidas y compuestos para el mismo. |
| WO2023110710A1 (en) | 2021-12-13 | 2023-06-22 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests & compounds therefor |
| EP4197333A1 (en) | 2021-12-15 | 2023-06-21 | Syngenta Crop Protection AG | Method for controlling diamide resistant pests & compounds therefor |
| WO2024133426A1 (en) | 2022-12-21 | 2024-06-27 | Syngenta Crop Protection Ag | Method for controlling diamide resistant pests and compounds therefor |
| WO2025134143A1 (en) | 2023-12-19 | 2025-06-26 | Pi Industries Ltd. | A method for the synthesis of substituted anthranilic amide compounds, intermediates and salts thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR043048A1 (es) | 2002-08-30 | 2005-07-13 | Syngenta Participations Ag | Derivados de 4-(3,3-dihalo- aliloxi) fenol con propiedades pesticidas |
| AU2004267094A1 (en) * | 2003-08-20 | 2005-03-03 | Vertex Pharmaceuticals Incorporated | (4 -amino -1,2, 5-oxadiazol-4-yl) -hetxiroaromatic compounds useful as protein kinase inhibitors |
| BRPI0515221A (pt) | 2004-08-17 | 2008-07-15 | Du Pont | composto, composição para controlar uma peste invertebrada, composições spray e de isca, dispositivo de armadilha, métodos para controlar uma peste invertebrada e métodos de controle |
| DE102006032168A1 (de) | 2006-06-13 | 2007-12-20 | Bayer Cropscience Ag | Anthranilsäurediamid-Derivate mit heteroaromatischen Substituenten |
| CN101466702B (zh) * | 2006-06-13 | 2014-04-02 | 拜尔农作物科学股份公司 | 具有杂芳族和杂环族取代基的邻氨基苯甲酰二胺衍生物 |
| PE20110838A1 (es) | 2008-12-18 | 2011-11-19 | Bayer Cropscience Ag | Amidas del acido antranilico sustituidas con tetrazol como plaguicidas |
| WO2011157664A1 (de) * | 2010-06-15 | 2011-12-22 | Bayer Cropscience Ag | Verfahren zur herstellung von tetrazol-substituierten anthranilsäurediamid-derivaten und neue kristalline modifikation dieser derivate |
-
2011
- 2011-06-10 WO PCT/EP2011/059735 patent/WO2011157664A1/de not_active Ceased
- 2011-06-10 CN CN201180039525.0A patent/CN103261187B/zh active Active
- 2011-06-10 EP EP11726391.3A patent/EP2582694B1/de active Active
- 2011-06-10 DK DK15171321.1T patent/DK2955176T3/en active
- 2011-06-10 MX MX2015009721A patent/MX347841B/es unknown
- 2011-06-10 JP JP2013514665A patent/JP6199739B2/ja active Active
- 2011-06-10 EP EP15171321.1A patent/EP2955176B1/de active Active
- 2011-06-10 MX MX2012014775A patent/MX2012014775A/es active IP Right Grant
- 2011-06-10 HR HRP20151088TT patent/HRP20151088T1/hr unknown
- 2011-06-10 PL PL11726391T patent/PL2582694T3/pl unknown
- 2011-06-10 HU HUE11726391A patent/HUE027943T2/en unknown
- 2011-06-10 SI SI201130627T patent/SI2582694T1/sl unknown
- 2011-06-10 PT PT117263913T patent/PT2582694E/pt unknown
- 2011-06-10 BR BR112012032244A patent/BR112012032244A2/pt not_active Application Discontinuation
- 2011-06-10 RS RS20150651A patent/RS54277B1/sr unknown
- 2011-06-10 ES ES15171321.1T patent/ES2660305T3/es active Active
- 2011-06-10 ES ES11726391.3T patent/ES2547314T3/es active Active
- 2011-06-10 DK DK11726391.3T patent/DK2582694T3/en active
- 2011-06-10 KR KR1020137000731A patent/KR101790305B1/ko active Active
- 2011-06-14 US US13/159,961 patent/US8969572B2/en active Active
- 2011-06-14 TW TW100120623A patent/TWI511668B/zh active
-
2014
- 2014-09-22 US US14/492,264 patent/US9056861B2/en active Active
-
2015
- 2015-11-11 JP JP2015221282A patent/JP6170118B2/ja active Active
-
2016
- 2016-07-20 JP JP2016142220A patent/JP6254646B2/ja active Active
Also Published As
| Publication number | Publication date |
|---|---|
| JP6170118B2 (ja) | 2017-07-26 |
| DK2955176T3 (en) | 2018-03-12 |
| WO2011157664A1 (de) | 2011-12-22 |
| ES2660305T3 (es) | 2018-03-21 |
| US20150025116A1 (en) | 2015-01-22 |
| PT2582694E (pt) | 2015-10-15 |
| EP2582694A1 (de) | 2013-04-24 |
| MX2012014775A (es) | 2013-01-29 |
| CN103261187A (zh) | 2013-08-21 |
| RS54277B1 (sr) | 2016-02-29 |
| DK2582694T3 (en) | 2015-10-26 |
| HUE027943T2 (en) | 2016-11-28 |
| KR101790305B1 (ko) | 2017-10-25 |
| PL2582694T3 (pl) | 2015-12-31 |
| EP2955176B1 (de) | 2017-12-06 |
| JP6199739B2 (ja) | 2017-09-20 |
| BR112012032244A2 (pt) | 2016-09-27 |
| CN103261187B (zh) | 2016-08-03 |
| JP2013530175A (ja) | 2013-07-25 |
| JP2017008062A (ja) | 2017-01-12 |
| KR20130112860A (ko) | 2013-10-14 |
| TWI511668B (zh) | 2015-12-11 |
| US9056861B2 (en) | 2015-06-16 |
| EP2582694B1 (de) | 2015-07-22 |
| JP2016065076A (ja) | 2016-04-28 |
| SI2582694T1 (sl) | 2015-11-30 |
| TW201212820A (en) | 2012-04-01 |
| EP2955176A1 (de) | 2015-12-16 |
| HRP20151088T1 (hr) | 2015-11-20 |
| ES2547314T3 (es) | 2015-10-05 |
| US20120101133A1 (en) | 2012-04-26 |
| US8969572B2 (en) | 2015-03-03 |
| JP6254646B2 (ja) | 2017-12-27 |
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