MX2021001761A - Formulaciones de ag10. - Google Patents

Formulaciones de ag10.

Info

Publication number
MX2021001761A
MX2021001761A MX2021001761A MX2021001761A MX2021001761A MX 2021001761 A MX2021001761 A MX 2021001761A MX 2021001761 A MX2021001761 A MX 2021001761A MX 2021001761 A MX2021001761 A MX 2021001761A MX 2021001761 A MX2021001761 A MX 2021001761A
Authority
MX
Mexico
Prior art keywords
formulations
pharmaceutically acceptable
acceptable salt
disintegrants
lubricants
Prior art date
Application number
MX2021001761A
Other languages
English (en)
Inventor
Mark Michael Menning
Jesper Jernelius
Original Assignee
Eidos Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eidos Therapeutics Inc filed Critical Eidos Therapeutics Inc
Publication of MX2021001761A publication Critical patent/MX2021001761A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente divulgación proporciona formulaciones de tableta de alta carga de AG10 o una sal farmacéuticamente aceptable del mismo. En algunos aspectos, en este documento se proporcionan formulaciones de tableta de alta carga de AG10 o una sal farmacéuticamente aceptable del mismo que incluyen al menos el 40% o más de AG10 en peso y al menos un excipiente farmacéutico seleccionado de uno o más rellenos, uno o más aglutinantes, uno o más desintegrantes, y uno o más lubricantes.
MX2021001761A 2018-08-17 2019-08-16 Formulaciones de ag10. MX2021001761A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862765154P 2018-08-17 2018-08-17
PCT/US2019/046789 WO2020037189A1 (en) 2018-08-17 2019-08-16 Formulations of ag10

Publications (1)

Publication Number Publication Date
MX2021001761A true MX2021001761A (es) 2021-04-19

Family

ID=69524257

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021001761A MX2021001761A (es) 2018-08-17 2019-08-16 Formulaciones de ag10.

Country Status (17)

Country Link
US (2) US11260047B2 (es)
EP (1) EP3836920A4 (es)
JP (2) JP7469293B2 (es)
KR (1) KR20210046708A (es)
CN (1) CN112804998A (es)
AU (1) AU2019321583A1 (es)
BR (1) BR112020026493A2 (es)
CA (1) CA3104695A1 (es)
CL (1) CL2021000289A1 (es)
EA (1) EA202190561A1 (es)
IL (1) IL280906A (es)
MA (1) MA53238A (es)
MX (1) MX2021001761A (es)
SG (1) SG11202101393PA (es)
TW (1) TWI834708B (es)
UA (1) UA128256C2 (es)
WO (1) WO2020037189A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL268683B2 (en) 2017-02-17 2023-04-01 Eidos Therapeutics Inc Processes for the preparation of ag-10, its intermediates and salts
JP2021518381A (ja) 2018-03-23 2021-08-02 エイドス セラピューティクス，インコーポレイティド Ａｇ１０を使用するｔｔｒアミロイドーシスの治療方法
KR20210046708A (ko) 2018-08-17 2021-04-28 에이도스 테라퓨틱스, 인코포레이티드 Ag10의 제형
WO2023052652A1 (en) 2021-10-01 2023-04-06 Sandoz Ag Crystalline form of acoramidis hydrochloride

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IL268683B2 (en) 2017-02-17 2023-04-01 Eidos Therapeutics Inc Processes for the preparation of ag-10, its intermediates and salts
JP2021518381A (ja) 2018-03-23 2021-08-02 エイドス セラピューティクス，インコーポレイティド Ａｇ１０を使用するｔｔｒアミロイドーシスの治療方法
KR20210046708A (ko) 2018-08-17 2021-04-28 에이도스 테라퓨틱스, 인코포레이티드 Ag10의 제형

Also Published As

Publication number Publication date
SG11202101393PA (en) 2021-03-30
IL280906A (en) 2021-04-29
JP2021534189A (ja) 2021-12-09
JP2024083460A (ja) 2024-06-21
MA53238A (fr) 2022-04-13
TWI834708B (zh) 2024-03-11
WO2020037189A1 (en) 2020-02-20
KR20210046708A (ko) 2021-04-28
EP3836920A1 (en) 2021-06-23
TW202021583A (zh) 2020-06-16
US12005043B2 (en) 2024-06-11
US11260047B2 (en) 2022-03-01
CN112804998A (zh) 2021-05-14
AU2019321583A1 (en) 2021-01-21
US20200054607A1 (en) 2020-02-20
JP7469293B2 (ja) 2024-04-16
UA128256C2 (uk) 2024-05-22
US20220313661A1 (en) 2022-10-06
BR112020026493A2 (pt) 2021-03-23
CL2021000289A1 (es) 2021-08-27
CA3104695A1 (en) 2020-02-20
EP3836920A4 (en) 2022-04-13
EA202190561A1 (ru) 2021-05-26

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