MX2016008780A - Derivados de sultam heteroarilo como moduladores del receptor huerfano relacionado con el acido retinoico gamma (ror gamma). - Google Patents
Derivados de sultam heteroarilo como moduladores del receptor huerfano relacionado con el acido retinoico gamma (ror gamma).Info
- Publication number
- MX2016008780A MX2016008780A MX2016008780A MX2016008780A MX2016008780A MX 2016008780 A MX2016008780 A MX 2016008780A MX 2016008780 A MX2016008780 A MX 2016008780A MX 2016008780 A MX2016008780 A MX 2016008780A MX 2016008780 A MX2016008780 A MX 2016008780A
- Authority
- MX
- Mexico
- Prior art keywords
- heteroaryl
- sultam derivatives
- rorc modulators
- rorc
- modulators
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/541—Non-condensed thiazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
Abstract
Los compuestos de la fórmula I o una sal farmacéutica de los mismos, en donde m, n, q, r, A, W, X1, X2, X3, X4, Y, Z, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 y R11 son como se definen en el presente documento. También se describen métodos de preparación de los compuestos y el uso de los compuestos para el tratamiento de enfermedades inflamatorias tales como artritis.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201461925831P | 2014-01-10 | 2014-01-10 | |
PCT/EP2015/050290 WO2015104353A1 (en) | 2014-01-10 | 2015-01-09 | HETEROARYL SULTAM DERIVATIVES AS RORc MODULATORS |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2016008780A true MX2016008780A (es) | 2016-09-08 |
Family
ID=52396653
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2016008780A MX2016008780A (es) | 2014-01-10 | 2015-01-09 | Derivados de sultam heteroarilo como moduladores del receptor huerfano relacionado con el acido retinoico gamma (ror gamma). |
Country Status (9)
Country | Link |
---|---|
US (1) | US20160311817A1 (es) |
EP (1) | EP3092237A1 (es) |
JP (1) | JP2017502070A (es) |
KR (1) | KR20160106165A (es) |
CN (1) | CN105899506A (es) |
CA (1) | CA2933391A1 (es) |
MX (1) | MX2016008780A (es) |
RU (1) | RU2016131356A (es) |
WO (1) | WO2015104353A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2760521T3 (es) | 2014-01-10 | 2020-05-14 | Hoffmann La Roche | Derivados de aril-sultamo como moduladores de RORc |
JP6458041B2 (ja) * | 2014-01-10 | 2019-01-23 | エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft | RORcモジュレーターとしてのアリールスルタム誘導体 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2013064231A1 (en) * | 2011-10-31 | 2013-05-10 | Phenex Pharmaceuticals Ag | SEVEN-MEMBERED SULFONAMIDES AS MODULATORS OF RAR-RELATED ORPHAN RECEPTOR-GAMMA (RORγ, NR1F3) |
US9216988B2 (en) * | 2011-12-22 | 2015-12-22 | Genentech, Inc. | Benzyl sulfonamide derivatives as RORc modulators |
PE20150229A1 (es) * | 2012-05-31 | 2015-03-02 | Phenex Pharmaceuticals Ag | Tiazoles sustituidos por carboxamida o sulfonamida y derivados relacionados como moduladores para el receptor nuclear huerfano rory |
-
2015
- 2015-01-09 WO PCT/EP2015/050290 patent/WO2015104353A1/en active Application Filing
- 2015-01-09 CA CA2933391A patent/CA2933391A1/en not_active Abandoned
- 2015-01-09 CN CN201580004084.9A patent/CN105899506A/zh active Pending
- 2015-01-09 EP EP15701104.0A patent/EP3092237A1/en not_active Withdrawn
- 2015-01-09 RU RU2016131356A patent/RU2016131356A/ru unknown
- 2015-01-09 KR KR1020167021672A patent/KR20160106165A/ko not_active Application Discontinuation
- 2015-01-09 MX MX2016008780A patent/MX2016008780A/es unknown
- 2015-01-09 JP JP2016545914A patent/JP2017502070A/ja active Pending
-
2016
- 2016-07-06 US US15/202,911 patent/US20160311817A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP3092237A1 (en) | 2016-11-16 |
WO2015104353A1 (en) | 2015-07-16 |
CA2933391A1 (en) | 2015-07-16 |
CN105899506A (zh) | 2016-08-24 |
RU2016131356A (ru) | 2018-02-16 |
US20160311817A1 (en) | 2016-10-27 |
KR20160106165A (ko) | 2016-09-09 |
JP2017502070A (ja) | 2017-01-19 |
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