MX2012002842A - Metodo para fabricar derivado de acido 4-(5-metilpiridin-2.iloamin o) piperidin-1-carboxilico. - Google Patents
Metodo para fabricar derivado de acido 4-(5-metilpiridin-2.iloamin o) piperidin-1-carboxilico.Info
- Publication number
- MX2012002842A MX2012002842A MX2012002842A MX2012002842A MX2012002842A MX 2012002842 A MX2012002842 A MX 2012002842A MX 2012002842 A MX2012002842 A MX 2012002842A MX 2012002842 A MX2012002842 A MX 2012002842A MX 2012002842 A MX2012002842 A MX 2012002842A
- Authority
- MX
- Mexico
- Prior art keywords
- reaction
- ylamino
- iron core
- bearing
- useful process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Motor Or Generator Frames (AREA)
Abstract
Es establece un método novedoso para fabricar 5-metil-2- (piperidin-4-ilamino) piridina. Este método puede usarse como un método de fabricación industrial para producir un derivado de ácido 4-(5-metilpiridin-2-ilamino)piperidin-1-carboxílico representado por la fórmula general, (ver fórmulas) en donde R representa un grupo alquilo lineal o ramificado que tiene 1 hasta 6 átomos de carbono o un grupo aralquilo que tiene 7 hasta 12 átomos de carbono en una solución de reacción que tiene un hidrocarburo monociclico aromático como un medio de reacción, en presencia de triacetoxiborohidruro de sodio como un agente reductor, o después de agregar borohidruro de sodio y ácido acético a la solución de reacción con anticipación.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2009207408 | 2009-09-08 | ||
| PCT/JP2010/005489 WO2011030537A1 (ja) | 2009-09-08 | 2010-09-07 | ４－（５－メチルピリジン－２－イルアミノ）ピペリジン－１－カルボン酸誘導体の製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2012002842A true MX2012002842A (es) | 2012-04-19 |
Family
ID=43732217
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2012002842A MX2012002842A (es) | 2009-09-08 | 2010-09-07 | Metodo para fabricar derivado de acido 4-(5-metilpiridin-2.iloamin o) piperidin-1-carboxilico. |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20120142932A1 (es) |
| EP (1) | EP2476677A1 (es) |
| JP (1) | JPWO2011030537A1 (es) |
| KR (1) | KR20120069710A (es) |
| CN (1) | CN102498108A (es) |
| BR (1) | BR112012003324A2 (es) |
| CA (1) | CA2773464A1 (es) |
| MX (1) | MX2012002842A (es) |
| TW (1) | TW201114758A (es) |
| WO (1) | WO2011030537A1 (es) |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EG12406A (en) * | 1976-08-12 | 1979-03-31 | Janssen Pharmaceutica Nv | Process for preparing of novel n-aryl-n-(1-l-4-piperidinyl)-arylacetamides |
| GB0030303D0 (en) * | 2000-12-13 | 2001-01-24 | Lilly Co Eli | Compounds |
| CN1326853C (zh) * | 2001-10-09 | 2007-07-18 | 杏林制药株式会社 | 4－(2－呋喃甲酰)氨基哌啶、其合成中间体、其制备方法及其作为药物的用途 |
| UA82711C2 (en) * | 2003-09-12 | 2008-05-12 | Эли Лилли Энд Компани | Substituted 2-carbonylamino-6-piperidinaminopyridines and substituted 1-carbonylamino-3-piperidinaminobenzenes as 5-ht1f agonists |
| GB0508318D0 (en) | 2005-04-25 | 2005-06-01 | Novartis Ag | Organic compounds |
| JP2008539220A (ja) * | 2005-04-26 | 2008-11-13 | ファイザー・リミテッド | バソプレシンアンタゴニストとしてのトリアゾール誘導体 |
| MX2009007644A (es) | 2007-01-16 | 2009-07-27 | Purdue Pharma Lp | Compuestos de piperidina heterociclicos sustituidos y usos de los mismos. |
-
2010
- 2010-09-07 EP EP10815137A patent/EP2476677A1/en not_active Withdrawn
- 2010-09-07 CA CA2773464A patent/CA2773464A1/en not_active Abandoned
- 2010-09-07 CN CN2010800406299A patent/CN102498108A/zh active Pending
- 2010-09-07 MX MX2012002842A patent/MX2012002842A/es unknown
- 2010-09-07 KR KR1020127008853A patent/KR20120069710A/ko not_active Application Discontinuation
- 2010-09-07 WO PCT/JP2010/005489 patent/WO2011030537A1/ja active Application Filing
- 2010-09-07 BR BRBR112012003324-7A patent/BR112012003324A2/pt not_active IP Right Cessation
- 2010-09-07 US US13/386,698 patent/US20120142932A1/en not_active Abandoned
- 2010-09-07 JP JP2011530746A patent/JPWO2011030537A1/ja active Pending
- 2010-09-08 TW TW099130282A patent/TW201114758A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPWO2011030537A1 (ja) | 2013-02-04 |
| WO2011030537A1 (ja) | 2011-03-17 |
| EP2476677A1 (en) | 2012-07-18 |
| TW201114758A (en) | 2011-05-01 |
| CA2773464A1 (en) | 2011-03-17 |
| BR112012003324A2 (pt) | 2015-09-01 |
| US20120142932A1 (en) | 2012-06-07 |
| CN102498108A (zh) | 2012-06-13 |
| KR20120069710A (ko) | 2012-06-28 |
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