MX2012002031A - Moleculas pequeñas que contienen boro como agentes antiprotozoarios. - Google Patents

Moleculas pequeñas que contienen boro como agentes antiprotozoarios.

Info

Publication number
MX2012002031A
MX2012002031A MX2012002031A MX2012002031A MX2012002031A MX 2012002031 A MX2012002031 A MX 2012002031A MX 2012002031 A MX2012002031 A MX 2012002031A MX 2012002031 A MX2012002031 A MX 2012002031A MX 2012002031 A MX2012002031 A MX 2012002031A
Authority
MX
Mexico
Prior art keywords
boron
small molecules
containing small
antiprotozoal agents
compounds
Prior art date
Application number
MX2012002031A
Other languages
English (en)
Inventor
Jacob J Plattner
Yong-Kang Zhang
Yasheen Zhou
Huchen Zhou
Dazhong Ding
Original Assignee
Anacor Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals Inc filed Critical Anacor Pharmaceuticals Inc
Publication of MX2012002031A publication Critical patent/MX2012002031A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06—Antimalarials

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención proporciona los nuevos compuestos de la siguiente fórmula, (ver fórmula) útiles para tratar infecciones por protozoarios, las composiciones farmacéuticas que contienen tales compuestos, así como las combinaciones de estos compuestos con al menos un agente terapéuticamente efectivo adicional.
MX2012002031A 2009-08-19 2010-08-16 Moleculas pequeñas que contienen boro como agentes antiprotozoarios. MX2012002031A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23529609P 2009-08-19 2009-08-19
PCT/US2010/045639 WO2011022337A1 (en) 2009-08-19 2010-08-16 Boron-containing small molecules as antiprotozoal agents

Publications (1)

Publication Number Publication Date
MX2012002031A true MX2012002031A (es) 2012-07-04

Family

ID=43383496

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012002031A MX2012002031A (es) 2009-08-19 2010-08-16 Moleculas pequeñas que contienen boro como agentes antiprotozoarios.

Country Status (4)

Country Link
US (1) US20110207701A1 (es)
IL (1) IL218163A0 (es)
MX (1) MX2012002031A (es)
WO (1) WO2011022337A1 (es)

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WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
WO2011116348A1 (en) * 2010-03-19 2011-09-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agent
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US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
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EP3086644A1 (en) 2013-12-23 2016-11-02 Syngenta Participations AG Benzoxaborole fungicides
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AR103397A1 (es) * 2015-01-13 2017-05-10 Syngenta Participations Ag Oxoborazoles microbicidas
US10633399B2 (en) * 2015-08-17 2020-04-28 Channel Therapeutics, Inc. Functionalized aminobenzoboroxoles
CN106467557B (zh) * 2015-08-18 2019-05-03 北京海美桐医药科技有限公司 他瓦硼罗的一种制备方法
TW201735792A (zh) 2016-03-07 2017-10-16 農業保鮮股份有限公司 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法
MA52337A (fr) 2017-03-01 2021-03-03 Anacor Pharmaceuticals Inc Nouveaux analogues d'oxaborole et utilisations de ces derniers
CN107090000B (zh) * 2017-04-27 2019-07-12 上海交通大学 一种苯并硼唑7位脂肪酸的衍生物及其制备与用途
CN108191898B (zh) * 2017-12-18 2020-08-25 上海交通大学 一种苯并硼唑7位查尔酮衍生物及其制备与应用
WO2019153324A1 (en) * 2018-02-12 2019-08-15 Shanghai Jiao Tong University Derivatives of 7-fatty acid substituted benzoxaborole and their preparation and use
WO2020186504A1 (en) * 2019-03-21 2020-09-24 Shanghai Jiao Tong University A new type of antitumor compounds: derivatives of 7-propanamide substituted benzoxaborole
CN111333672B (zh) * 2020-04-07 2022-11-08 中国医学科学院放射医学研究所 一种固醇调控元件结合蛋白和酸性核质dna结合蛋白-1抑制剂及其制备方法和应用
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WO2024094235A1 (en) 2022-11-03 2024-05-10 Univerzita Karlova Use of benzoxaborole-based compounds in therapy of diseases caused by amoebas of the naegleria genus

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Also Published As

Publication number Publication date
WO2011022337A1 (en) 2011-02-24
US20110207701A1 (en) 2011-08-25
IL218163A0 (en) 2012-07-31

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