MX2010007928A - Imidazolinilmetil aril sulfonamidas novedosas. - Google Patents

Imidazolinilmetil aril sulfonamidas novedosas.

Info

Publication number
MX2010007928A
MX2010007928A MX2010007928A MX2010007928A MX2010007928A MX 2010007928 A MX2010007928 A MX 2010007928A MX 2010007928 A MX2010007928 A MX 2010007928A MX 2010007928 A MX2010007928 A MX 2010007928A MX 2010007928 A MX2010007928 A MX 2010007928A
Authority
MX
Mexico
Prior art keywords
novel
aryl sulfonamides
imidazolinylmethyl
imidazolinylmethyl aryl
methods
Prior art date
Application number
MX2010007928A
Other languages
English (en)
Inventor
Counde O'yang
Robert Greenhouse
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MX2010007928A publication Critical patent/MX2010007928A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D233/24—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Esta invención se refiere a un agonista parcial del receptor alfa-1A, que está representado por la fórmula (I) y a las sales o solvatos del mismo farmacéuticamente aceptables. La invención se refiere además a composiciones farmacéuticas que contienen la fórmula I, a métodos para su uso como agentes terapéuticos, y a métodos de preparación de los mismos.
MX2010007928A 2008-02-04 2009-01-26 Imidazolinilmetil aril sulfonamidas novedosas. MX2010007928A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2584208P 2008-02-04 2008-02-04
PCT/EP2009/050839 WO2009098135A1 (en) 2008-02-04 2009-01-26 Novel imidazolinylmethyl aryl sulfonamides

Publications (1)

Publication Number Publication Date
MX2010007928A true MX2010007928A (es) 2010-08-09

Family

ID=40481825

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010007928A MX2010007928A (es) 2008-02-04 2009-01-26 Imidazolinilmetil aril sulfonamidas novedosas.

Country Status (10)

Country Link
EP (1) EP2238114A1 (es)
JP (1) JP2011511025A (es)
KR (1) KR20100096261A (es)
CN (1) CN101925580A (es)
AU (1) AU2009211505A1 (es)
BR (1) BRPI0906640A2 (es)
CA (1) CA2711726A1 (es)
IL (1) IL206612A0 (es)
MX (1) MX2010007928A (es)
WO (1) WO2009098135A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0906632A2 (pt) * 2008-02-04 2015-07-14 Hoffmann La Roche Imidazolinil metil aril sulfonamidas
CN110041261B (zh) * 2019-05-24 2022-06-24 广东先强药业有限公司 一种盐酸萘甲唑啉的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ535823A (en) * 2002-04-23 2007-07-27 Hoffmann La Roche Imidazolin-2-ylmethyl substituted aralkylsulfonamides

Also Published As

Publication number Publication date
IL206612A0 (en) 2010-12-30
BRPI0906640A2 (pt) 2019-09-17
AU2009211505A1 (en) 2009-08-13
WO2009098135A1 (en) 2009-08-13
JP2011511025A (ja) 2011-04-07
EP2238114A1 (en) 2010-10-13
KR20100096261A (ko) 2010-09-01
CN101925580A (zh) 2010-12-22
CA2711726A1 (en) 2009-08-13

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