MX2010007579A - Preparacion nutriceutica o farmaceutica revestida con una liberacion de sustancia activa de impulsion mejorada. - Google Patents
Preparacion nutriceutica o farmaceutica revestida con una liberacion de sustancia activa de impulsion mejorada.Info
- Publication number
- MX2010007579A MX2010007579A MX2010007579A MX2010007579A MX2010007579A MX 2010007579 A MX2010007579 A MX 2010007579A MX 2010007579 A MX2010007579 A MX 2010007579A MX 2010007579 A MX2010007579 A MX 2010007579A MX 2010007579 A MX2010007579 A MX 2010007579A
- Authority
- MX
- Mexico
- Prior art keywords
- meth
- weight
- weight based
- acrylic
- active substance
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención trata sobre una preparación farmacéutica o nutricéutica que consta de un núcleo que contiene una sustancia farmacéutica o nutricéuticamente activa y una sustancia que actúa en una forma moduladora con respecto a la liberación de las sustancias farmacéutica o nutricéuticamente activas; y una capa controladora que rodea el núcleo y consta de i) 55 a 92% por peso con base en el peso total de copolímeros (met) acrílicos presentes en la capa de un o una mezcla de una variedad de copolímeros de (met) acrilato compuesta de 80 a 98% por peso con base en el peso del copolímero (met) acrílico de unidades estructurales derivadas del C1 a C4 alquil ésteres del ácido (met) acrílico y 2 a 20% por peso con base en el peso del copolímero (met) acrílico de unidades estructurales derivado de monómeros de (met) acrilato con un grupo de amonio cuaternario en el radical alquilo; y ii) 8 a 45% por peso con base en el peso total de los copolímeros (met) acrílicos presentes en la capa de uno o una mezcla de una variedad de copolímeros de (met) acrilato compuesto por más de 5 a 59% por peso con base en el peso del copolímero o unidades estructurales derivadas del ácido acrílico o del ácido metacrílico y tabletas o cápsulas que constan de lo mismo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN96CH2008 | 2008-01-10 | ||
PCT/EP2008/051238 WO2009086941A1 (en) | 2008-01-10 | 2008-02-01 | Coated pharmaceutical or nutraceutical preparation with enhanced pulsed active substance release |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2010007579A true MX2010007579A (es) | 2010-08-03 |
Family
ID=40527442
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2010007579A MX2010007579A (es) | 2008-01-10 | 2008-02-01 | Preparacion nutriceutica o farmaceutica revestida con una liberacion de sustancia activa de impulsion mejorada. |
Country Status (15)
Country | Link |
---|---|
US (1) | US9011907B2 (es) |
EP (1) | EP2227225B1 (es) |
JP (1) | JP2011509265A (es) |
KR (1) | KR101571179B1 (es) |
CN (1) | CN101903017B (es) |
BR (1) | BRPI0822140A8 (es) |
CA (1) | CA2711474C (es) |
ES (1) | ES2715274T3 (es) |
HU (1) | HUE043474T2 (es) |
IL (1) | IL205550A (es) |
MX (1) | MX2010007579A (es) |
PL (1) | PL2227225T4 (es) |
SI (1) | SI2227225T1 (es) |
TR (1) | TR201902212T4 (es) |
WO (1) | WO2009086941A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2983409B1 (fr) * | 2011-12-06 | 2013-12-27 | Ethypharm Sa | Comprime susceptible de lutter contre le detournement par voie injectable |
WO2016044704A1 (en) | 2014-09-19 | 2016-03-24 | The Procter & Gamble Company | Pulsed release phenylephrine dosage forms |
US10278930B2 (en) | 2017-03-16 | 2019-05-07 | The Procter & Gamble Company | Method for relieving sinus congestion |
MX2019008440A (es) | 2019-07-15 | 2021-01-18 | Dva Farma Mexicana S A De C V | Composiciones de recubrimientos en pelicula para tabletas con brillantez incrementada, procedimiento de preparacion y aplicacion. |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE8003805L (sv) | 1980-05-21 | 1981-11-22 | Haessle Ab | En farmaceutisk beredning med forbettrade utlosningsegenskap |
DE69020758T2 (de) | 1989-03-10 | 1995-12-07 | Yamanouchi Pharma Co Ltd | Die Wirkstoffabgabe steuerndes Überzugsmaterial für lang wirksame Formulierungen. |
JPH0674206B2 (ja) * | 1989-12-28 | 1994-09-21 | 田辺製薬株式会社 | 放出制御型製剤およびその製法 |
JPH07112932A (ja) | 1993-08-27 | 1995-05-02 | Mitsui Toatsu Chem Inc | 徐放性医薬製剤 |
JPH08143476A (ja) | 1994-11-18 | 1996-06-04 | Japan Tobacco Inc | 薬物放出制御膜及び固形製剤 |
DE19845358A1 (de) * | 1998-10-02 | 2000-04-06 | Roehm Gmbh | Überzogene Arzneiformen mit kontrollierter Wirkstoffabgabe |
DE10013029A1 (de) * | 2000-03-17 | 2001-09-20 | Roehm Gmbh | Mehrschichtige Arzneiform für die Colonfreigabe |
NZ530511A (en) * | 2001-07-16 | 2005-06-24 | Astrazeneca Ab | A tablet for treating disorders of the gastrointestinal tract comprising a proton pump inhibitor and at least one antacid that has a barrier layer to cover an enteric coating film |
DE10250543A1 (de) * | 2002-10-29 | 2004-05-19 | Röhm GmbH & Co. KG | Mehrschichtige Arzneiform |
RU2372893C2 (ru) * | 2003-10-31 | 2009-11-20 | Хексал Аг | Содержащий фармацевтический агент состав с покрытием |
DE10353196A1 (de) * | 2003-11-13 | 2005-06-16 | Röhm GmbH & Co. KG | Mehrschichtige Arzneiform mit einer die Abgabe einer modulatorischen Substanz beeinflussenden Matrix |
DE10353186A1 (de) | 2003-11-13 | 2005-06-16 | Röhm GmbH & Co. KG | Mehrschichtige Arzneiform, enthaltend eine in Bezug auf die Wirkstoffabgabe modulatorisch wirkende Substanz |
CN101111230B (zh) | 2005-03-29 | 2010-05-19 | 赢创罗姆有限责任公司 | 包含对活性成分具有调节释放作用的小丸的多颗粒药用形式 |
ES2385498T3 (es) * | 2006-08-18 | 2012-07-25 | Evonik Röhm Gmbh | Composición farmacéutica con liberación controlada de la sustancia activa, para sustancias activas con una buena solubilidad en agua |
BRPI0716196A2 (pt) * | 2006-08-31 | 2013-11-12 | Eurand Inc | Sistemas de distribuição de fármacos que compreendem soluções sólidas de fármacos fracamente básicos. |
DE102007009243A1 (de) * | 2007-02-22 | 2008-09-18 | Evonik Röhm Gmbh | Pellets mit einer Wirkstoff-Matrix und einem Polymerüberzug, sowie ein Verfahren zur Herstellung der Pellets |
-
2008
- 2008-02-01 CA CA2711474A patent/CA2711474C/en active Active
- 2008-02-01 MX MX2010007579A patent/MX2010007579A/es active IP Right Grant
- 2008-02-01 WO PCT/EP2008/051238 patent/WO2009086941A1/en active Application Filing
- 2008-02-01 EP EP08708548.6A patent/EP2227225B1/en active Active
- 2008-02-01 US US12/742,945 patent/US9011907B2/en active Active
- 2008-02-01 PL PL08708548T patent/PL2227225T4/pl unknown
- 2008-02-01 KR KR1020107015178A patent/KR101571179B1/ko active IP Right Grant
- 2008-02-01 BR BRPI0822140A patent/BRPI0822140A8/pt not_active Application Discontinuation
- 2008-02-01 HU HUE08708548A patent/HUE043474T2/hu unknown
- 2008-02-01 ES ES08708548T patent/ES2715274T3/es active Active
- 2008-02-01 SI SI200832039T patent/SI2227225T1/sl unknown
- 2008-02-01 JP JP2010541718A patent/JP2011509265A/ja active Pending
- 2008-02-01 CN CN200880122062.2A patent/CN101903017B/zh active Active
- 2008-02-01 TR TR2019/02212T patent/TR201902212T4/tr unknown
-
2010
- 2010-05-05 IL IL205550A patent/IL205550A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
EP2227225B1 (en) | 2018-11-14 |
BRPI0822140A2 (pt) | 2019-10-01 |
KR20100103564A (ko) | 2010-09-27 |
CN101903017A (zh) | 2010-12-01 |
TR201902212T4 (tr) | 2019-06-21 |
IL205550A0 (en) | 2010-12-30 |
CA2711474C (en) | 2016-03-29 |
HUE043474T2 (hu) | 2019-08-28 |
EP2227225A1 (en) | 2010-09-15 |
BRPI0822140A8 (pt) | 2022-07-05 |
KR101571179B1 (ko) | 2015-11-23 |
CN101903017B (zh) | 2014-12-24 |
PL2227225T3 (pl) | 2019-05-31 |
SI2227225T1 (sl) | 2019-04-30 |
JP2011509265A (ja) | 2011-03-24 |
US20100291202A1 (en) | 2010-11-18 |
IL205550A (en) | 2017-06-29 |
US9011907B2 (en) | 2015-04-21 |
ES2715274T3 (es) | 2019-06-03 |
CA2711474A1 (en) | 2009-07-16 |
WO2009086941A1 (en) | 2009-07-16 |
PL2227225T4 (pl) | 2019-05-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration |