MX2009012714A - Nuevas 4-heteroail-imidazol-2-tionas como inhibidores de la tirosinasa, su procedimiento de preparacion y su uso en medicina humana asi como en cosmetica. - Google Patents
Nuevas 4-heteroail-imidazol-2-tionas como inhibidores de la tirosinasa, su procedimiento de preparacion y su uso en medicina humana asi como en cosmetica.Info
- Publication number
- MX2009012714A MX2009012714A MX2009012714A MX2009012714A MX2009012714A MX 2009012714 A MX2009012714 A MX 2009012714A MX 2009012714 A MX2009012714 A MX 2009012714A MX 2009012714 A MX2009012714 A MX 2009012714A MX 2009012714 A MX2009012714 A MX 2009012714A
- Authority
- MX
- Mexico
- Prior art keywords
- heteroaryl
- imidazole
- novel
- thiones
- cosmetology
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Dermatology (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Toxicology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a nuevos compuestos de 4-heteroaril-imidazol-2-tionas que responden a la fórmula general (I) siguiente, a las composiciones que los contienen, 5 a su procedimiento de preparación y a su utilización en composiciones farmacéuticas o cosméticas destinadas al tratamiento o a la prevención de trastornos pigmentarios. (ver fórmula I).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0755473A FR2917089B1 (fr) | 2007-06-05 | 2007-06-05 | Nouveaux 4-heteroaryl-imidazole-2-thiones comme inhibiteurs de la tyrosinase, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique. |
PCT/FR2008/050995 WO2008152332A1 (fr) | 2007-06-05 | 2008-06-04 | Nouveaux 4-héteroaryl-imidazole-2-thiones comme inhibiteurs de la tyrosinase, leur procédé de préparation et leur utilisation en médecine humaine ainsi qu'en cosmétique |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009012714A true MX2009012714A (es) | 2009-12-08 |
Family
ID=38962668
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009012714A MX2009012714A (es) | 2007-06-05 | 2008-06-04 | Nuevas 4-heteroail-imidazol-2-tionas como inhibidores de la tirosinasa, su procedimiento de preparacion y su uso en medicina humana asi como en cosmetica. |
Country Status (12)
Country | Link |
---|---|
US (1) | US7989483B2 (es) |
EP (1) | EP2164845A1 (es) |
JP (1) | JP2010529097A (es) |
KR (1) | KR20100028090A (es) |
CN (1) | CN101679388A (es) |
AR (1) | AR066871A1 (es) |
AU (1) | AU2008263667A1 (es) |
CA (1) | CA2688237A1 (es) |
FR (1) | FR2917089B1 (es) |
MX (1) | MX2009012714A (es) |
RU (1) | RU2009149608A (es) |
WO (1) | WO2008152332A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2917087B1 (fr) * | 2007-06-05 | 2012-09-21 | Galderma Res & Dev | Nouveaux 4-phenyl-imidazole-2-thiones comme inhibiteurs de la tyrosinase, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique. |
TWI508950B (zh) * | 2014-08-29 | 2015-11-21 | Univ Hungkuang | 3-methyl-2-sulfanyl-2,3-dihydro-1H-imidazole-1-carboxylic acid Tertiary butyl ester and its preparation method and use |
JP6553961B2 (ja) * | 2015-06-25 | 2019-07-31 | 花王株式会社 | 美白剤 |
CN116854267B (zh) * | 2023-09-01 | 2024-01-02 | 杭州尚善若水环保科技有限公司 | 一种用于反渗透膜的阻垢剂及其制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4159338A (en) * | 1977-02-09 | 1979-06-26 | E. I. Du Pont De Nemours And Company | Antiinflammatory-4,5-dicyclic-2-(substituted thio)-imidazoles and their corresponding sulfoxides and sulfones |
JPH05124923A (ja) * | 1991-04-09 | 1993-05-21 | Sansho Seiyaku Co Ltd | メラニン生成抑制外用剤 |
JPH05132422A (ja) * | 1991-04-09 | 1993-05-28 | Sansho Seiyaku Co Ltd | メラニン生成抑制外用剤 |
US7115748B2 (en) * | 2004-12-07 | 2006-10-03 | Allergan, Inc. | Method of making imidazole-2-thiones |
FR2917087B1 (fr) * | 2007-06-05 | 2012-09-21 | Galderma Res & Dev | Nouveaux 4-phenyl-imidazole-2-thiones comme inhibiteurs de la tyrosinase, leur procede de preparation et leur utilisation en medecine humaine ainsi qu'en cosmetique. |
-
2007
- 2007-06-05 FR FR0755473A patent/FR2917089B1/fr not_active Expired - Fee Related
-
2008
- 2008-06-04 KR KR1020107000023A patent/KR20100028090A/ko not_active Application Discontinuation
- 2008-06-04 RU RU2009149608/04A patent/RU2009149608A/ru not_active Application Discontinuation
- 2008-06-04 CN CN200880018930A patent/CN101679388A/zh active Pending
- 2008-06-04 CA CA002688237A patent/CA2688237A1/fr not_active Abandoned
- 2008-06-04 WO PCT/FR2008/050995 patent/WO2008152332A1/fr active Application Filing
- 2008-06-04 EP EP08805935A patent/EP2164845A1/fr not_active Withdrawn
- 2008-06-04 AU AU2008263667A patent/AU2008263667A1/en not_active Abandoned
- 2008-06-04 MX MX2009012714A patent/MX2009012714A/es active IP Right Grant
- 2008-06-04 JP JP2010510857A patent/JP2010529097A/ja active Pending
- 2008-06-05 AR ARP080102387A patent/AR066871A1/es unknown
-
2009
- 2009-12-04 US US12/631,309 patent/US7989483B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US20100144813A1 (en) | 2010-06-10 |
KR20100028090A (ko) | 2010-03-11 |
AR066871A1 (es) | 2009-09-16 |
EP2164845A1 (fr) | 2010-03-24 |
US7989483B2 (en) | 2011-08-02 |
FR2917089B1 (fr) | 2009-07-17 |
JP2010529097A (ja) | 2010-08-26 |
WO2008152332A1 (fr) | 2008-12-18 |
AU2008263667A1 (en) | 2008-12-18 |
FR2917089A1 (fr) | 2008-12-12 |
RU2009149608A (ru) | 2011-07-20 |
CN101679388A (zh) | 2010-03-24 |
CA2688237A1 (fr) | 2008-12-18 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MX2010003258A (es) | Utilizacion de un nuevo agente natural en composiciones cosmeticas. | |
MY179527A (en) | Catecholamine derivatives useful for the treatment of parkinson's disease | |
MX367623B (es) | 6-amino-nicotinamidas sustituidas como moduladores de kcnq2/3. | |
MY146662A (en) | Novel n-(8-heteroaryltetrahydronaphtalene-2yl) or n-(5-heteroarylchromane-3-yl) carboxamide derivatives for the treatment of pain | |
TNSN08370A1 (en) | Tetrahydropyridothienopyrimidine compounds and methods of use thereof | |
MX341211B (es) | Sintesis de un nuevo antioxidante de nitroxido y metodos de uso en composiciones cosmeticas y dermatologicas. | |
WO2009141541A3 (fr) | Utilisation d' inhibiteurs de kif13a et d ' ap-1 pour inhiber la melanogenese | |
TW200738659A (en) | Novel compounds | |
MX2009013131A (es) | Moduladores de gamma secretasa. | |
MX2010009022A (es) | Derivados 16 alfa, 17 alfa-acetal glucocorticoesteroideos y su uso. | |
UA104988C2 (uk) | Похідні піроніндолу та спосіб їх отримання | |
MX2011013130A (es) | Nuevos compuestos de bencensulfonamida, metodo para sintetizarlos y su utilizacion en medicina asi como tambien en cosmeticos. | |
UA101393C2 (ru) | КОМПОЗИЦИИ И ПРИМЕНЕНИЕ ПРОИЗВОДНЫХ ТРИАЗОЛА ДЛЯ ЛЕЧЕНИЯ β-АМИЛОИДОЗОВ И СИНУКЛЕИНОПАТИЙ | |
WO2007049158A3 (en) | Ppar modulating biaromatic compounds | |
WO2008107092A3 (en) | Use of derivatives of 4-hydroxyphenoxy acetic acid | |
MX2009002224A (es) | Composicion a base de xantoxilina y su utilizacion en cosmetica. | |
SI2373310T1 (sl) | Nove spojine 4- (heterocikloalkil) benzen-1, 3- diola kot inhibitorji tirosinaze, postopek njihove priprave in njihova uporaba v humani medicini in tudi v kozmetiki | |
MX2013002118A (es) | 2-oxi-quinolin-3-carboxamidas sustituidas como moduladores de kcnq2/3. | |
MY146802A (en) | Novel drugs for treating respiratory diseases | |
MX2009012712A (es) | Nuevas 4-fenil-imidazol-2-tionas como inhibidores de la tirosinasa, su procedimiento de preparacion y su uso en medicina humana asi como en cosmetica. | |
MX2009012714A (es) | Nuevas 4-heteroail-imidazol-2-tionas como inhibidores de la tirosinasa, su procedimiento de preparacion y su uso en medicina humana asi como en cosmetica. | |
WO2006103119A3 (en) | Tyrosinase inhibitors, process for the preparation thereof and use thereof in human medicine and also in cosmetics | |
CY1111361T1 (el) | Νεα προσδεματα συναγωνιστες των υποδοχεων rar, χρηση στην ανθρωπινη ιατρικη καθως και στην κοσμετολογια | |
MX2013002295A (es) | 1-oxo-dihidroisoquinolin-3-carboxamidas sustituidas como moduladores de kcnq2/3. | |
WO2005056510A3 (en) | Novel ligands that are activators of the rar receptors, use in human medicine and in cosmetics |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration |