MX2007007261A - Enantiomeros de 3-heteroaril-8h-8-azabiciclo(3.2.1)oct-2-eno y su uso como inhibidores de la recaptacion del neurotransmisor de monoamina. - Google Patents
Enantiomeros de 3-heteroaril-8h-8-azabiciclo(3.2.1)oct-2-eno y su uso como inhibidores de la recaptacion del neurotransmisor de monoamina.Info
- Publication number
- MX2007007261A MX2007007261A MX2007007261A MX2007007261A MX2007007261A MX 2007007261 A MX2007007261 A MX 2007007261A MX 2007007261 A MX2007007261 A MX 2007007261A MX 2007007261 A MX2007007261 A MX 2007007261A MX 2007007261 A MX2007007261 A MX 2007007261A
- Authority
- MX
- Mexico
- Prior art keywords
- disorder
- oct
- aza
- bicyclo
- pain
- Prior art date
Links
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- 229940095064 tartrate Drugs 0.000 description 1
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- 238000004448 titration Methods 0.000 description 1
- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 description 1
- 238000003325 tomography Methods 0.000 description 1
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- WBYWAXJHAXSJNI-VOTSOKGWSA-M trans-cinnamate Chemical compound [O-]C(=O)\C=C\C1=CC=CC=C1 WBYWAXJHAXSJNI-VOTSOKGWSA-M 0.000 description 1
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- WTVXIBRMWGUIMI-UHFFFAOYSA-N trifluoro($l^{1}-oxidanylsulfonyl)methane Chemical group [O]S(=O)(=O)C(F)(F)F WTVXIBRMWGUIMI-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
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Landscapes
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- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200401950 | 2004-12-17 | ||
| US63686904P | 2004-12-20 | 2004-12-20 | |
| DKPA200500506 | 2005-04-08 | ||
| US66988705P | 2005-04-11 | 2005-04-11 | |
| PCT/EP2005/056801 WO2006064031A1 (en) | 2004-12-17 | 2005-12-15 | Enantiomers of 3-heteroaryl-8h-8-azabicyclo(3.2.1)oct-2-ene and their use as monoamine neurotransmitter re-uptake inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007007261A true MX2007007261A (es) | 2007-08-14 |
Family
ID=35976671
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007007261A MX2007007261A (es) | 2004-12-17 | 2005-12-15 | Enantiomeros de 3-heteroaril-8h-8-azabiciclo(3.2.1)oct-2-eno y su uso como inhibidores de la recaptacion del neurotransmisor de monoamina. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US7781456B2 (enExample) |
| EP (1) | EP1828173A1 (enExample) |
| JP (1) | JP2008524161A (enExample) |
| KR (1) | KR20070089170A (enExample) |
| AU (1) | AU2005315623A1 (enExample) |
| BR (1) | BRPI0519921A2 (enExample) |
| CA (1) | CA2591621A1 (enExample) |
| IL (1) | IL182738A0 (enExample) |
| MX (1) | MX2007007261A (enExample) |
| NO (1) | NO20073652L (enExample) |
| WO (1) | WO2006064031A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| TW200800980A (en) | 2006-02-17 | 2008-01-01 | Neurosearch As | Novel compounds |
| CA2673315A1 (en) * | 2006-12-20 | 2008-06-26 | Neurosearch A/S | Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| AU2007336291A1 (en) * | 2006-12-20 | 2008-06-26 | Neurosearch A/S | Novel chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| TW200904815A (en) | 2007-05-09 | 2009-02-01 | Neurosearch As | Novel compounds |
| CN102216295A (zh) * | 2008-11-18 | 2011-10-12 | 神经研究公司 | 8-氮杂双环[3.2.1]辛-2-烯衍生物及其作为单胺神经递质再摄取抑制剂的用途 |
| AU2010247514A1 (en) | 2009-05-15 | 2011-11-17 | Neurosearch A/S | Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| WO2011092061A1 (en) | 2010-01-29 | 2011-08-04 | Neurosearch A/S | Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| WO2025172422A1 (en) * | 2024-02-13 | 2025-08-21 | Initiator Pharma A/S | Compound for use in the treatment of pain and enantiopure compositions thereof |
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| AU4819099A (en) * | 1998-06-19 | 2000-01-05 | Eli Lilly And Company | Inhibition of serotonin reuptake |
| AU9543601A (en) | 2000-10-13 | 2002-04-22 | Neurosearch As | Treatment of affective disorders by the combined action of a nicotinic receptor agonist and a monoaminergic substance |
| NZ529880A (en) * | 2001-07-06 | 2005-09-30 | Neurosearch As | Novel compounds, their preparation and use |
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2005
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- 2005-12-15 WO PCT/EP2005/056801 patent/WO2006064031A1/en not_active Ceased
- 2005-12-15 KR KR1020077013663A patent/KR20070089170A/ko not_active Withdrawn
- 2005-12-15 MX MX2007007261A patent/MX2007007261A/es not_active Application Discontinuation
- 2005-12-15 EP EP05817471A patent/EP1828173A1/en not_active Withdrawn
- 2005-12-15 BR BRPI0519921-2A patent/BRPI0519921A2/pt not_active IP Right Cessation
- 2005-12-15 JP JP2007546061A patent/JP2008524161A/ja not_active Abandoned
- 2005-12-15 AU AU2005315623A patent/AU2005315623A1/en not_active Abandoned
- 2005-12-15 CA CA002591621A patent/CA2591621A1/en not_active Abandoned
-
2007
- 2007-04-23 IL IL182738A patent/IL182738A0/en unknown
- 2007-07-16 NO NO20073652A patent/NO20073652L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US20080214820A1 (en) | 2008-09-04 |
| NO20073652L (no) | 2007-07-16 |
| EP1828173A1 (en) | 2007-09-05 |
| KR20070089170A (ko) | 2007-08-30 |
| AU2005315623A1 (en) | 2006-06-22 |
| US7781456B2 (en) | 2010-08-24 |
| BRPI0519921A2 (pt) | 2009-08-11 |
| IL182738A0 (en) | 2007-07-24 |
| JP2008524161A (ja) | 2008-07-10 |
| WO2006064031A1 (en) | 2006-06-22 |
| CA2591621A1 (en) | 2006-06-22 |
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