MC1239A1 - Acides et derives d'acides 4-pyridone-3-carboxyliques leur preparation et leur application en tant que medicaments - Google Patents
Acides et derives d'acides 4-pyridone-3-carboxyliques leur preparation et leur application en tant que medicamentsInfo
- Publication number
- MC1239A1 MC1239A1 MC791356A MC1356A MC1239A1 MC 1239 A1 MC1239 A1 MC 1239A1 MC 791356 A MC791356 A MC 791356A MC 1356 A MC1356 A MC 1356A MC 1239 A1 MC1239 A1 MC 1239A1
- Authority
- MC
- Monaco
- Prior art keywords
- group
- sub
- alkyl
- oxo
- acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/80—Acids; Esters in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Oncology (AREA)
- Psychiatry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Communicable Diseases (AREA)
- Neurosurgery (AREA)
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH51278A CH639073A5 (en) | 1978-01-18 | 1978-01-18 | 4-Pyridone-3-carboxylic acid derivatives and their preparation |
| CH1173478 | 1978-11-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MC1239A1 true MC1239A1 (fr) | 1979-10-26 |
Family
ID=25684790
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MC791356A MC1239A1 (fr) | 1978-01-18 | 1979-01-15 | Acides et derives d'acides 4-pyridone-3-carboxyliques leur preparation et leur application en tant que medicaments |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US4521535A (enExample) |
| EP (1) | EP0003144B1 (enExample) |
| JP (1) | JPS54100382A (enExample) |
| KR (1) | KR820002111B1 (enExample) |
| AR (1) | AR223663A1 (enExample) |
| AT (1) | AT369731B (enExample) |
| AU (1) | AU521148B2 (enExample) |
| CA (1) | CA1110234A (enExample) |
| DE (1) | DE2901868A1 (enExample) |
| DK (1) | DK20279A (enExample) |
| ES (1) | ES476917A1 (enExample) |
| FI (1) | FI790103A7 (enExample) |
| FR (1) | FR2415103A1 (enExample) |
| GB (1) | GB2013190B (enExample) |
| GR (1) | GR73088B (enExample) |
| HU (1) | HU179487B (enExample) |
| IE (1) | IE47784B1 (enExample) |
| IL (1) | IL56421A (enExample) |
| LU (1) | LU80794A1 (enExample) |
| MC (1) | MC1239A1 (enExample) |
| NL (1) | NL7900264A (enExample) |
| NO (1) | NO152089C (enExample) |
| NZ (1) | NZ189379A (enExample) |
| PT (1) | PT69093A (enExample) |
| SE (1) | SE7900318L (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1125762A (en) * | 1979-07-13 | 1982-06-15 | Alexander E. Wick | Dihydronicotinic acid derivatives and process for the preparation thereof |
| NZ197027A (en) * | 1980-05-12 | 1984-03-16 | Rohm & Haas | 4-oxo-2-phenyl-nicotinic acids salts and esters and growth regulating compositions |
| US4964896A (en) * | 1980-05-12 | 1990-10-23 | Monsanto Company | Certain-2,6-diphenyl-1,4-dihydro-4-oxo-nicotinates which are useful for inducing male sterility in cereal grain plants |
| US4936904A (en) * | 1980-05-12 | 1990-06-26 | Carlson Glenn R | Aryl-4-oxonicotinates useful for inducing male sterility in cereal grain plants |
| US4714492A (en) * | 1980-05-12 | 1987-12-22 | Rohm And Haas Company | Certain 2-phenyl-4-oxo-nicotinates and their use for inducing male sterility in a cereal grain plant |
| NZ201395A (en) * | 1981-07-30 | 1987-02-20 | Bayer Ag | Pharmaceutical compositions containing 1,4-dihydropyridines and certain of these dihydropyridines |
| DE3338846A1 (de) * | 1982-10-29 | 1984-05-03 | Toyama Chemical Co. Ltd., Tokyo | Neue 4-oxo-1,4-dihydronicotinsaeurederivate und salze derselben, verfahren zu ihrer herstellung und antibakterielle mittel mit einem gehalt derselben |
| JPS5980665A (ja) * | 1982-10-29 | 1984-05-10 | Toyama Chem Co Ltd | ４−オキソ−１，４−ジヒドロニコチン酸誘導体 |
| GB8502424D0 (en) * | 1985-01-31 | 1985-03-06 | Pharis R P | Promotion of flowering fruit trees |
| GB9317314D0 (en) * | 1993-08-20 | 1993-10-06 | Smithkline Beecham Corp | Compounds |
| EP2149547A1 (en) * | 2008-07-30 | 2010-02-03 | LEK Pharmaceuticals D.D. | Process for the synthesis of ezetimibe and intermediates useful therefor |
| US9988373B2 (en) | 2013-12-26 | 2018-06-05 | Shionogi & Co., Ltd. | Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3907808A (en) * | 1971-05-17 | 1975-09-23 | Sterling Drug Inc | 1,4-Dihydro-4-oxo-7-pyridyl-3-quinolinecarboxylic acid derivatives |
| IN142614B (enExample) * | 1974-08-28 | 1977-08-06 | Lilly Co Eli | |
| CA1125762A (en) * | 1979-07-13 | 1982-06-15 | Alexander E. Wick | Dihydronicotinic acid derivatives and process for the preparation thereof |
| DE3338846A1 (de) * | 1982-10-29 | 1984-05-03 | Toyama Chemical Co. Ltd., Tokyo | Neue 4-oxo-1,4-dihydronicotinsaeurederivate und salze derselben, verfahren zu ihrer herstellung und antibakterielle mittel mit einem gehalt derselben |
-
1978
- 1978-12-28 CA CA318,702A patent/CA1110234A/en not_active Expired
-
1979
- 1979-01-11 AU AU43296/79A patent/AU521148B2/en not_active Ceased
- 1979-01-12 NL NL7900264A patent/NL7900264A/xx not_active Application Discontinuation
- 1979-01-12 IL IL56421A patent/IL56421A/xx unknown
- 1979-01-12 FI FI790103A patent/FI790103A7/fi unknown
- 1979-01-15 NZ NZ189379A patent/NZ189379A/en unknown
- 1979-01-15 SE SE7900318A patent/SE7900318L/xx unknown
- 1979-01-15 HU HU79HO2130A patent/HU179487B/hu unknown
- 1979-01-15 MC MC791356A patent/MC1239A1/fr unknown
- 1979-01-16 FR FR7900974A patent/FR2415103A1/fr active Granted
- 1979-01-16 JP JP233079A patent/JPS54100382A/ja active Pending
- 1979-01-16 LU LU80794A patent/LU80794A1/de unknown
- 1979-01-16 GR GR58105A patent/GR73088B/el unknown
- 1979-01-17 ES ES476917A patent/ES476917A1/es not_active Expired
- 1979-01-17 AT AT0035079A patent/AT369731B/de not_active IP Right Cessation
- 1979-01-17 GB GB7901668A patent/GB2013190B/en not_active Expired
- 1979-01-17 DK DK20279A patent/DK20279A/da not_active Application Discontinuation
- 1979-01-17 KR KR7900120A patent/KR820002111B1/ko not_active Expired
- 1979-01-17 AR AR275201A patent/AR223663A1/es active
- 1979-01-17 NO NO790165A patent/NO152089C/no unknown
- 1979-01-17 PT PT7969093A patent/PT69093A/pt unknown
- 1979-01-18 DE DE19792901868 patent/DE2901868A1/de not_active Withdrawn
- 1979-01-18 EP EP79100149A patent/EP0003144B1/de not_active Expired
- 1979-01-30 IE IE113/79A patent/IE47784B1/en unknown
-
1982
- 1982-04-19 US US06/369,778 patent/US4521535A/en not_active Expired - Fee Related
-
1984
- 1984-11-02 US US06/667,528 patent/US4549022A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| NO790165L (no) | 1979-07-19 |
| GB2013190A (en) | 1979-08-08 |
| FR2415103B1 (enExample) | 1982-11-05 |
| FI790103A7 (fi) | 1979-07-19 |
| GB2013190B (en) | 1982-07-14 |
| IL56421A0 (en) | 1979-03-12 |
| IE47784B1 (en) | 1984-06-13 |
| GR73088B (enExample) | 1984-02-01 |
| DE2901868A1 (de) | 1979-07-19 |
| CA1110234A (en) | 1981-10-06 |
| NL7900264A (nl) | 1979-07-20 |
| EP0003144A2 (de) | 1979-07-25 |
| NO152089B (no) | 1985-04-22 |
| NO152089C (no) | 1985-08-14 |
| SE7900318L (sv) | 1979-07-19 |
| IL56421A (en) | 1982-08-31 |
| FR2415103A1 (fr) | 1979-08-17 |
| DK20279A (da) | 1979-07-19 |
| US4549022A (en) | 1985-10-22 |
| JPS54100382A (en) | 1979-08-08 |
| EP0003144A3 (en) | 1979-08-08 |
| IE790113L (en) | 1979-07-18 |
| AU521148B2 (en) | 1982-03-18 |
| ES476917A1 (es) | 1979-11-16 |
| AU4329679A (en) | 1979-07-26 |
| AT369731B (de) | 1983-01-25 |
| US4521535A (en) | 1985-06-04 |
| PT69093A (en) | 1979-02-01 |
| EP0003144B1 (de) | 1981-08-05 |
| KR820002111B1 (ko) | 1982-11-10 |
| ATA35079A (de) | 1982-06-15 |
| LU80794A1 (de) | 1980-02-14 |
| NZ189379A (en) | 1984-07-06 |
| HU179487B (en) | 1982-10-28 |
| AR223663A1 (es) | 1981-09-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| YP | Annual fee paid |