MA32012B1 - Octahydroquinolizines destinees au traitement du diabete - Google Patents
Octahydroquinolizines destinees au traitement du diabeteInfo
- Publication number
- MA32012B1 MA32012B1 MA33011A MA33011A MA32012B1 MA 32012 B1 MA32012 B1 MA 32012B1 MA 33011 A MA33011 A MA 33011A MA 33011 A MA33011 A MA 33011A MA 32012 B1 MA32012 B1 MA 32012B1
- Authority
- MA
- Morocco
- Prior art keywords
- treatment
- prevention
- obesity
- diabetes
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/02—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
L'invention concerne de nouvelles octahydroquinolizines utilisées dans le traitement ou la prévention du diabetes mellitus et de ses complications, dans le traitement ou la prévention de l'hyperlipidémie, dans le traitement de la dyslipidémie diabétique, dans le traitement ou la prévention du syndrome métabolique, dans le traitement de maladies liées à un dysfonctionnement métabolique, et dans le traitement de l'obésité ou de maladies liées à l'obésité. L'invention se rapporte aussi à des compositions pharmaceutiques et à des trousses comprenant lesdits composés, seuls ou combinés à d'autres médicaments ou composés, qui ont pour objet d'offrir un traitement ou une prévention améliorés des maladies et syndromes précités chez des humains ou des animaux.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07450235A EP2072515B1 (fr) | 2007-12-19 | 2007-12-19 | Quinazolidines substituées pour traitement antidiabétique |
AT13152008 | 2008-08-25 | ||
PCT/AT2008/000458 WO2009076693A1 (fr) | 2007-12-19 | 2008-12-17 | Octahydroquinolizines destinées au traitement du diabète |
Publications (1)
Publication Number | Publication Date |
---|---|
MA32012B1 true MA32012B1 (fr) | 2011-01-03 |
Family
ID=40430049
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA33011A MA32012B1 (fr) | 2007-12-19 | 2010-07-14 | Octahydroquinolizines destinees au traitement du diabete |
Country Status (16)
Country | Link |
---|---|
US (1) | US20110003808A1 (fr) |
EP (1) | EP2222673A1 (fr) |
JP (1) | JP2011506485A (fr) |
KR (1) | KR20100107469A (fr) |
CN (1) | CN101918402A (fr) |
AP (1) | AP2010005317A0 (fr) |
AU (1) | AU2008338287B2 (fr) |
BR (1) | BRPI0821160A2 (fr) |
CA (1) | CA2710006A1 (fr) |
EA (1) | EA201070750A1 (fr) |
IL (1) | IL205752A0 (fr) |
MA (1) | MA32012B1 (fr) |
MX (1) | MX2010006173A (fr) |
NZ (1) | NZ585307A (fr) |
WO (1) | WO2009076693A1 (fr) |
ZA (1) | ZA201003316B (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2315766A1 (fr) * | 2008-08-25 | 2011-05-04 | 55pharma Drug Discovery & Development AG | Octahydroquinolizines destinées au traitement du diabète |
JP6520440B2 (ja) * | 2014-06-16 | 2019-05-29 | 有限会社バイオシステムコンサルティング | 新規化合物 |
CN110746282A (zh) * | 2019-11-04 | 2020-02-04 | 天津市安凯特科技发展有限公司 | 一种4-氯-2-丁酮的合成方法 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA795318B (en) * | 1978-10-13 | 1980-09-24 | Hoffmann La Roche | Phenyl quinolizidines |
US7538110B2 (en) * | 2005-10-27 | 2009-05-26 | Adolor Corporation | Opioid antagonists |
-
2008
- 2008-12-17 US US12/809,513 patent/US20110003808A1/en not_active Abandoned
- 2008-12-17 NZ NZ585307A patent/NZ585307A/en not_active IP Right Cessation
- 2008-12-17 JP JP2010538265A patent/JP2011506485A/ja active Pending
- 2008-12-17 EP EP08862420A patent/EP2222673A1/fr not_active Withdrawn
- 2008-12-17 AP AP2010005317A patent/AP2010005317A0/en unknown
- 2008-12-17 CN CN2008801225325A patent/CN101918402A/zh active Pending
- 2008-12-17 CA CA2710006A patent/CA2710006A1/fr not_active Abandoned
- 2008-12-17 MX MX2010006173A patent/MX2010006173A/es active IP Right Grant
- 2008-12-17 EA EA201070750A patent/EA201070750A1/ru unknown
- 2008-12-17 KR KR1020107015983A patent/KR20100107469A/ko not_active Application Discontinuation
- 2008-12-17 WO PCT/AT2008/000458 patent/WO2009076693A1/fr active Application Filing
- 2008-12-17 BR BRPI0821160-4A patent/BRPI0821160A2/pt not_active IP Right Cessation
- 2008-12-17 AU AU2008338287A patent/AU2008338287B2/en not_active Expired - Fee Related
-
2010
- 2010-05-11 ZA ZA2010/03316A patent/ZA201003316B/en unknown
- 2010-05-13 IL IL205752A patent/IL205752A0/en unknown
- 2010-07-14 MA MA33011A patent/MA32012B1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
BRPI0821160A2 (pt) | 2015-06-16 |
CA2710006A1 (fr) | 2009-06-25 |
AP2010005317A0 (en) | 2010-08-31 |
JP2011506485A (ja) | 2011-03-03 |
AU2008338287B2 (en) | 2012-06-07 |
MX2010006173A (es) | 2010-09-30 |
ZA201003316B (en) | 2011-08-31 |
IL205752A0 (en) | 2010-11-30 |
WO2009076693A1 (fr) | 2009-06-25 |
AU2008338287A1 (en) | 2009-06-25 |
CN101918402A (zh) | 2010-12-15 |
EP2222673A1 (fr) | 2010-09-01 |
US20110003808A1 (en) | 2011-01-06 |
NZ585307A (en) | 2011-11-25 |
KR20100107469A (ko) | 2010-10-05 |
EA201070750A1 (ru) | 2010-12-30 |
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