LV13089B - 4-oxo-and 4h-imidazo(5,1-c)(1,4)benzoxazines useful as benzodiazepine receptor-binding agents - Google Patents
4-oxo-and 4h-imidazo(5,1-c)(1,4)benzoxazines useful as benzodiazepine receptor-binding agents Download PDFInfo
- Publication number
- LV13089B LV13089B LVP-03-63A LV030063A LV13089B LV 13089 B LV13089 B LV 13089B LV 030063 A LV030063 A LV 030063A LV 13089 B LV13089 B LV 13089B
- Authority
- LV
- Latvia
- Prior art keywords
- alkyl
- imidazo
- aryl
- fluoro
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Adhesives Or Adhesive Processes (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US83664592A | 1992-02-13 | 1992-02-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
LV13089B true LV13089B (en) | 2004-01-20 |
Family
ID=25272407
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
LVP-03-63A LV13089B (en) | 1992-02-13 | 2003-06-12 | 4-oxo-and 4h-imidazo(5,1-c)(1,4)benzoxazines useful as benzodiazepine receptor-binding agents |
Country Status (11)
Country | Link |
---|---|
US (1) | US5610158A (es) |
EP (1) | EP0625982B1 (es) |
JP (1) | JP3512110B2 (es) |
AT (1) | ATE219083T1 (es) |
AU (1) | AU3443593A (es) |
DE (1) | DE69332019T2 (es) |
DK (1) | DK0625982T3 (es) |
ES (1) | ES2177539T3 (es) |
LV (1) | LV13089B (es) |
PT (1) | PT625982E (es) |
WO (1) | WO1993016082A1 (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9410469D0 (en) * | 1994-05-25 | 1994-07-13 | Erba Farmitalia | Imidazolylalkyl derivatives of imidazo (5,1-c) (1,4) benzoxazin-1-one and process for their preparation |
ZA968661B (en) * | 1995-11-17 | 1998-04-14 | Upjohn Co | Oxazolidinone antibacterial agent with tricyclic substituents. |
CA2636043A1 (en) * | 2006-01-23 | 2007-08-02 | Amira Pharmaceuticals, Inc. | Tricyclic inhibitors of 5-lipoxygenase |
CU20090172A7 (es) | 2009-10-09 | 2011-10-05 | Ct De Investigación Y Desarrollo De Medicamentos | Sistemas tricíclicos y tetracíclicos con actividad sobre el sistema nervioso central y vascular |
ES2637113T3 (es) | 2011-01-10 | 2017-10-10 | Infinity Pharmaceuticals, Inc. | Procedimientos para preparar isoquinolinonas y formas sólidas de isoquinolinonas |
US10138233B2 (en) | 2013-06-24 | 2018-11-27 | Merck Patent Gmbh | Imidazole compounds as modulators of FSHR and uses thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1052009B (it) * | 1975-12-30 | 1981-06-20 | Erba Carlo Spa | Imidazo 4.3 c 1.4 benzossazino imidazo 4.3 c 1.4 benzotiazino pirazo 2.1 c 1.4 benzossazino e pirazo 2.1 c 1.4 benzotiazino derivati |
GB2043637B (en) * | 1979-02-09 | 1983-03-16 | Roussel Lab Ltd | Heterotricyclic derivatives |
DK476885D0 (da) * | 1985-10-17 | 1985-10-17 | Ferrosan As | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
DK155524C (da) * | 1987-03-18 | 1989-09-11 | Ferrosan As | Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse |
DK160876C (da) * | 1987-12-08 | 1991-10-14 | Novo Nordisk As | Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar |
-
1993
- 1993-01-14 AT AT93902972T patent/ATE219083T1/de not_active IP Right Cessation
- 1993-01-14 JP JP51405293A patent/JP3512110B2/ja not_active Expired - Fee Related
- 1993-01-14 ES ES93902972T patent/ES2177539T3/es not_active Expired - Lifetime
- 1993-01-14 AU AU34435/93A patent/AU3443593A/en not_active Abandoned
- 1993-01-14 DK DK93902972T patent/DK0625982T3/da active
- 1993-01-14 PT PT93902972T patent/PT625982E/pt unknown
- 1993-01-14 DE DE69332019T patent/DE69332019T2/de not_active Expired - Fee Related
- 1993-01-14 WO PCT/US1993/000095 patent/WO1993016082A1/en active IP Right Grant
- 1993-01-14 EP EP93902972A patent/EP0625982B1/en not_active Expired - Lifetime
-
1994
- 1994-08-03 US US08/285,560 patent/US5610158A/en not_active Expired - Fee Related
-
2003
- 2003-06-12 LV LVP-03-63A patent/LV13089B/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP0625982B1 (en) | 2002-06-12 |
DE69332019T2 (de) | 2002-11-28 |
ATE219083T1 (de) | 2002-06-15 |
ES2177539T3 (es) | 2002-12-16 |
PT625982E (pt) | 2002-10-31 |
DE69332019D1 (de) | 2002-07-18 |
US5610158A (en) | 1997-03-11 |
JPH07503727A (ja) | 1995-04-20 |
DK0625982T3 (da) | 2002-09-30 |
JP3512110B2 (ja) | 2004-03-29 |
EP0625982A1 (en) | 1994-11-30 |
AU3443593A (en) | 1993-09-03 |
WO1993016082A1 (en) | 1993-08-19 |
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