LU88331I2 - Doxazosin (Cardura) - Google Patents

Doxazosin (Cardura)

Info

Publication number
LU88331I2
LU88331I2 LU88331C LU88331C LU88331I2 LU 88331 I2 LU88331 I2 LU 88331I2 LU 88331 C LU88331 C LU 88331C LU 88331 C LU88331 C LU 88331C LU 88331 I2 LU88331 I2 LU 88331I2
Authority
LU
Luxembourg
Prior art keywords
cardura
doxazosin
Prior art date
Application number
LU88331C
Other languages
French (fr)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of LU88331I2 publication Critical patent/LU88331I2/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/201,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
LU88331C 1977-11-05 1993-06-24 Doxazosin (Cardura) LU88331I2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4612877 1977-11-05

Publications (1)

Publication Number Publication Date
LU88331I2 true LU88331I2 (en) 1994-05-04

Family

ID=10439957

Family Applications (2)

Application Number Title Priority Date Filing Date
LU80470A LU80470A1 (en) 1977-11-05 1978-11-03 "NEWS DERIVED FROM 4-ANIMO-2- (PIPERAZIN-1-YL OR HOMOPIPE-RAZIN-1-YL) -QUINAZOLINE, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM.
LU88331C LU88331I2 (en) 1977-11-05 1993-06-24 Doxazosin (Cardura)

Family Applications Before (1)

Application Number Title Priority Date Filing Date
LU80470A LU80470A1 (en) 1977-11-05 1978-11-03 "NEWS DERIVED FROM 4-ANIMO-2- (PIPERAZIN-1-YL OR HOMOPIPE-RAZIN-1-YL) -QUINAZOLINE, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM.

Country Status (36)

Country Link
JP (1) JPS5498792A (en)
AR (2) AR219562A1 (en)
AT (1) AT365186B (en)
AU (1) AU509329B2 (en)
BE (1) BE871771A (en)
CA (1) CA1088059A (en)
CH (1) CH643255A5 (en)
CS (2) CS207671B2 (en)
DD (1) DD139850A5 (en)
DE (1) DE2847623C2 (en)
DK (1) DK154082C (en)
EG (1) EG13594A (en)
ES (2) ES474805A1 (en)
FI (1) FI64366C (en)
FR (1) FR2407929A1 (en)
GR (1) GR81514B (en)
HK (1) HK94284A (en)
HU (1) HU176306B (en)
IE (1) IE47888B1 (en)
IL (1) IL55857A (en)
IN (1) IN148828B (en)
IT (1) IT1100919B (en)
KE (1) KE3350A (en)
LU (2) LU80470A1 (en)
MY (1) MY8500286A (en)
NL (2) NL174549C (en)
NO (1) NO150158C (en)
NZ (1) NZ188813A (en)
PH (1) PH13966A (en)
PL (2) PL119419B1 (en)
PT (1) PT68735A (en)
SE (1) SE437518B (en)
SU (1) SU816403A3 (en)
UA (1) UA8324A1 (en)
YU (2) YU40204B (en)
ZA (1) ZA786184B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985002617A1 (en) * 1983-12-14 1985-06-20 Takeda Chemical Industries. Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1986002644A1 (en) * 1984-11-01 1986-05-09 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1985004658A1 (en) * 1984-04-04 1985-10-24 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepine derivatives and their preparation
EP0849264A1 (en) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Novel polymorphic form of doxazosin mesylate (form I)
EP0849265A1 (en) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Novel polymorphic form of doxazosin mesylate (form II)
DK0849266T3 (en) * 1996-12-20 2007-06-04 Heumann Pcs Gmbh New polymorphic form of doxazosin mesylate (form III)
TW448155B (en) * 1999-03-29 2001-08-01 Dev Center Biotechnology Method for producing amide compounds and quinazolin derivatives
EP1403263B1 (en) * 2002-09-27 2005-06-22 Council of Scientific and Industrial Research Process for the preparation of N-(2,3-dihydrobenzo 1,4 dioxin-2-carbonyl) piperazine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3635979A (en) * 1969-09-29 1972-01-18 Pfizer Certain 6- and/or 7-alkoxy-substituted-2 4-bis(disubstituted amino) quinazolines
US3669968A (en) * 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines

Also Published As

Publication number Publication date
YU40419B (en) 1985-12-31
HU176306B (en) 1981-01-28
FR2407929B1 (en) 1981-02-27
FI64366C (en) 1983-11-10
NL930062I1 (en) 1993-09-01
JPS5498792A (en) 1979-08-03
AT365186B (en) 1981-12-28
BE871771A (en) 1979-05-03
NL930062I2 (en) 1993-11-16
SE7811382L (en) 1979-05-06
AR223015A1 (en) 1981-07-15
PL119586B1 (en) 1982-01-30
GR81514B (en) 1984-12-11
PT68735A (en) 1978-12-01
NO150158B (en) 1984-05-21
MY8500286A (en) 1985-12-31
AU509329B2 (en) 1980-05-08
DK154082C (en) 1989-02-27
ATA784378A (en) 1981-05-15
NL174549C (en) 1984-07-02
LU80470A1 (en) 1980-06-05
EG13594A (en) 1982-03-31
CS207671B2 (en) 1981-08-31
UA8324A1 (en) 1996-03-29
AU4132278A (en) 1979-05-17
IE47888B1 (en) 1984-07-11
YU38683A (en) 1983-06-30
IL55857A (en) 1982-07-30
FR2407929A1 (en) 1979-06-01
NL7810909A (en) 1979-05-08
ES8308559A1 (en) 1980-07-16
DK154082B (en) 1988-10-10
FI783347A (en) 1979-05-06
ES474805A1 (en) 1980-01-16
IN148828B (en) 1981-06-27
PL210681A1 (en) 1979-11-05
NO150158C (en) 1984-08-29
SU816403A3 (en) 1981-03-23
ES480121A0 (en) 1980-07-16
NO783705L (en) 1979-05-08
AR219562A1 (en) 1980-08-29
CA1088059A (en) 1980-10-21
CH643255A5 (en) 1984-05-30
IT1100919B (en) 1985-09-28
IL55857A0 (en) 1979-01-31
KE3350A (en) 1983-12-16
FI64366B (en) 1983-07-29
DE2847623C2 (en) 1983-06-01
DE2847623A1 (en) 1979-05-23
NZ188813A (en) 1980-10-08
IT7829434A0 (en) 1978-11-03
NL174549B (en) 1984-02-01
CS354491A3 (en) 1992-06-17
DD139850A5 (en) 1980-01-23
DK428678A (en) 1979-05-06
PH13966A (en) 1980-11-12
SE437518B (en) 1985-03-04
ZA786184B (en) 1979-10-31
JPS5625233B2 (en) 1981-06-11
HK94284A (en) 1984-12-07
YU40204B (en) 1985-08-31
PL119419B1 (en) 1981-12-31
YU255378A (en) 1983-06-30
IE782179L (en) 1979-05-05

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