IT1100919B - THERAPEUTIC AGENTS BASED ON CHINAZOLINE DERIVATIVES - Google Patents

THERAPEUTIC AGENTS BASED ON CHINAZOLINE DERIVATIVES

Info

Publication number
IT1100919B
IT1100919B IT29434/78A IT2943478A IT1100919B IT 1100919 B IT1100919 B IT 1100919B IT 29434/78 A IT29434/78 A IT 29434/78A IT 2943478 A IT2943478 A IT 2943478A IT 1100919 B IT1100919 B IT 1100919B
Authority
IT
Italy
Prior art keywords
therapeutic agents
agents based
chinazoline derivatives
chinazoline
derivatives
Prior art date
Application number
IT29434/78A
Other languages
Italian (it)
Other versions
IT7829434A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IT7829434A0 publication Critical patent/IT7829434A0/en
Application granted granted Critical
Publication of IT1100919B publication Critical patent/IT1100919B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/201,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IT29434/78A 1977-11-05 1978-11-03 THERAPEUTIC AGENTS BASED ON CHINAZOLINE DERIVATIVES IT1100919B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4612877 1977-11-05

Publications (2)

Publication Number Publication Date
IT7829434A0 IT7829434A0 (en) 1978-11-03
IT1100919B true IT1100919B (en) 1985-09-28

Family

ID=10439957

Family Applications (1)

Application Number Title Priority Date Filing Date
IT29434/78A IT1100919B (en) 1977-11-05 1978-11-03 THERAPEUTIC AGENTS BASED ON CHINAZOLINE DERIVATIVES

Country Status (36)

Country Link
JP (1) JPS5498792A (en)
AR (2) AR219562A1 (en)
AT (1) AT365186B (en)
AU (1) AU509329B2 (en)
BE (1) BE871771A (en)
CA (1) CA1088059A (en)
CH (1) CH643255A5 (en)
CS (2) CS207671B2 (en)
DD (1) DD139850A5 (en)
DE (1) DE2847623C2 (en)
DK (1) DK154082C (en)
EG (1) EG13594A (en)
ES (2) ES474805A1 (en)
FI (1) FI64366C (en)
FR (1) FR2407929A1 (en)
GR (1) GR81514B (en)
HK (1) HK94284A (en)
HU (1) HU176306B (en)
IE (1) IE47888B1 (en)
IL (1) IL55857A (en)
IN (1) IN148828B (en)
IT (1) IT1100919B (en)
KE (1) KE3350A (en)
LU (2) LU80470A1 (en)
MY (1) MY8500286A (en)
NL (2) NL174549C (en)
NO (1) NO150158C (en)
NZ (1) NZ188813A (en)
PH (1) PH13966A (en)
PL (2) PL119586B1 (en)
PT (1) PT68735A (en)
SE (1) SE437518B (en)
SU (1) SU816403A3 (en)
UA (1) UA8324A1 (en)
YU (2) YU40204B (en)
ZA (1) ZA786184B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985004658A1 (en) * 1984-04-04 1985-10-24 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepine derivatives and their preparation
WO1985002617A1 (en) * 1983-12-14 1985-06-20 Takeda Chemical Industries. Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1986002644A1 (en) * 1984-11-01 1986-05-09 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
EP0849264A1 (en) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Novel polymorphic form of doxazosin mesylate (form I)
ES2282997T3 (en) * 1996-12-20 2007-10-16 Heumann Pcs Gmbh NEW POLYMORM FORM OF MESILATE AND DOXAZOSINE (FORM III).
EP0849265A1 (en) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Novel polymorphic form of doxazosin mesylate (form II)
TW448155B (en) * 1999-03-29 2001-08-01 Dev Center Biotechnology Method for producing amide compounds and quinazolin derivatives
EP1403263B1 (en) * 2002-09-27 2005-06-22 Council of Scientific and Industrial Research Process for the preparation of N-(2,3-dihydrobenzo 1,4 dioxin-2-carbonyl) piperazine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3663706A (en) * 1969-09-29 1972-05-16 Pfizer Use of 2,4-diaminoquinazolines as hypotensive agents
US3669968A (en) * 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines

Also Published As

Publication number Publication date
AR223015A1 (en) 1981-07-15
DD139850A5 (en) 1980-01-23
IL55857A (en) 1982-07-30
NL174549B (en) 1984-02-01
PL210681A1 (en) 1979-11-05
IE782179L (en) 1979-05-05
IT7829434A0 (en) 1978-11-03
NL174549C (en) 1984-07-02
AR219562A1 (en) 1980-08-29
ES8308559A1 (en) 1980-07-16
CA1088059A (en) 1980-10-21
NL930062I2 (en) 1993-11-16
PT68735A (en) 1978-12-01
CH643255A5 (en) 1984-05-30
AU4132278A (en) 1979-05-17
NL7810909A (en) 1979-05-08
LU80470A1 (en) 1980-06-05
PL119419B1 (en) 1981-12-31
FI783347A (en) 1979-05-06
NO150158B (en) 1984-05-21
JPS5498792A (en) 1979-08-03
LU88331I2 (en) 1994-05-04
DK154082B (en) 1988-10-10
ZA786184B (en) 1979-10-31
FR2407929B1 (en) 1981-02-27
FR2407929A1 (en) 1979-06-01
YU40204B (en) 1985-08-31
NO783705L (en) 1979-05-08
NZ188813A (en) 1980-10-08
JPS5625233B2 (en) 1981-06-11
AU509329B2 (en) 1980-05-08
YU38683A (en) 1983-06-30
MY8500286A (en) 1985-12-31
ES474805A1 (en) 1980-01-16
FI64366C (en) 1983-11-10
AT365186B (en) 1981-12-28
PH13966A (en) 1980-11-12
SE437518B (en) 1985-03-04
IE47888B1 (en) 1984-07-11
IL55857A0 (en) 1979-01-31
HU176306B (en) 1981-01-28
EG13594A (en) 1982-03-31
NL930062I1 (en) 1993-09-01
DE2847623C2 (en) 1983-06-01
DK428678A (en) 1979-05-06
BE871771A (en) 1979-05-03
PL119586B1 (en) 1982-01-30
NO150158C (en) 1984-08-29
YU255378A (en) 1983-06-30
CS354491A3 (en) 1992-06-17
IN148828B (en) 1981-06-27
HK94284A (en) 1984-12-07
CS207671B2 (en) 1981-08-31
GR81514B (en) 1984-12-11
YU40419B (en) 1985-12-31
KE3350A (en) 1983-12-16
DK154082C (en) 1989-02-27
ES480121A0 (en) 1980-07-16
UA8324A1 (en) 1996-03-29
FI64366B (en) 1983-07-29
DE2847623A1 (en) 1979-05-23
ATA784378A (en) 1981-05-15
SE7811382L (en) 1979-05-06
SU816403A3 (en) 1981-03-23

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Legal Events

Date Code Title Description
ITCP Complementary protection certificate

Free format text: CCP 72

MEDD Supplementary protection certificate for pharmaceutical products: granted

Free format text: CCP 72, 19920325; PFIZER CORPORATION

TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19961017