LU86960A1 - Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux - Google Patents

Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux Download PDF

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Publication number
LU86960A1
LU86960A1 LU86960A LU86960A LU86960A1 LU 86960 A1 LU86960 A1 LU 86960A1 LU 86960 A LU86960 A LU 86960A LU 86960 A LU86960 A LU 86960A LU 86960 A1 LU86960 A1 LU 86960A1
Authority
LU
Luxembourg
Prior art keywords
oxide
formula
compound
denotes
diamino
Prior art date
Application number
LU86960A
Other languages
English (en)
French (fr)
Inventor
Jean Maignan
Gerard Lang
Serge Restle
Original Assignee
Oreal
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oreal filed Critical Oreal
Priority to LU86960A priority Critical patent/LU86960A1/fr
Priority to EP88112023A priority patent/EP0304648B1/fr
Priority to AT88112023T priority patent/ATE80877T1/de
Priority to DE8888112023T priority patent/DE3874842T2/de
Priority to US07/225,819 priority patent/US4985563A/en
Priority to JP63188536A priority patent/JP2647444B2/ja
Priority to CA000573529A priority patent/CA1318914C/fr
Publication of LU86960A1 publication Critical patent/LU86960A1/fr
Priority to US07/636,126 priority patent/US5126453A/en
Priority to JP9032596A priority patent/JP2726653B2/ja

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50—Three nitrogen atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)
LU86960A 1987-07-31 1987-07-31 Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux LU86960A1 (fr)

Priority Applications (9)

Application Number Priority Date Filing Date Title
LU86960A LU86960A1 (fr) 1987-07-31 1987-07-31 Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux
EP88112023A EP0304648B1 (fr) 1987-07-31 1988-07-26 Procédé de préparation de pipéridino-6 diamino-2,4 pyrimidine oxyde-3 et composés
AT88112023T ATE80877T1 (de) 1987-07-31 1988-07-26 Verfahren zur herstellung von 6-piperidino-2,4diaminopyrimidin-3-oxid, und verbindungen.
DE8888112023T DE3874842T2 (de) 1987-07-31 1988-07-26 Verfahren zur herstellung von 6-piperidino-2,4-diaminopyrimidin-3-oxid, und verbindungen.
US07/225,819 US4985563A (en) 1987-07-31 1988-07-29 Process for the preparation of 6-piperidino-2,4-diamino pyrimidine-3-oxide
JP63188536A JP2647444B2 (ja) 1987-07-31 1988-07-29 ６−ピペリジノ−２，４−ジアミノピリミジン−３−オキシドの調整方法および新規な化合物
CA000573529A CA1318914C (fr) 1987-07-31 1988-08-01 Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux
US07/636,126 US5126453A (en) 1987-07-31 1990-12-31 Process for the preparation of 6-piperidino-2,4-diamino pyrimidine-3-oxide and novel compounds
JP9032596A JP2726653B2 (ja) 1987-07-31 1997-02-03 ジアミノピリミジン誘導体

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU86960A LU86960A1 (fr) 1987-07-31 1987-07-31 Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux
LU86960 1987-07-31

Publications (1)

Publication Number Publication Date
LU86960A1 true LU86960A1 (fr) 1989-03-08

Family

ID=19730956

Family Applications (1)

Application Number Title Priority Date Filing Date
LU86960A LU86960A1 (fr) 1987-07-31 1987-07-31 Procede de preparation de piperidino-6 diamino-2,4 pyrimidine oxyde-3 et composes nouveaux

Country Status (7)

Country Link
US (2) US4985563A (ja)
EP (1) EP0304648B1 (ja)
JP (2) JP2647444B2 (ja)
AT (1) ATE80877T1 (ja)
CA (1) CA1318914C (ja)
DE (1) DE3874842T2 (ja)
LU (1) LU86960A1 (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0467026B1 (de) * 1990-07-17 1993-03-03 Goldwell Aktiengesellschaft Mittel zur Färbung von Haaren und Anwendung desselben
US5502050A (en) * 1993-11-29 1996-03-26 Cornell Research Foundation, Inc. Blocking utilization of tetrahydrobiopterin to block induction of nitric oxide synthesis
BRPI0515944B1 (pt) * 2004-09-29 2021-11-09 Bayer Healthcare Llc Processo para a preparação de 4-{4-[({[4-cloro-3-(trifluorometil)fe-nil]amino}carbonil) amino]fenóxi}nmetilpiridina-2-carboxamida
AU2006259525B2 (en) * 2005-06-14 2012-05-24 Gpcr Therapeutics, Inc Pyrimidine compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3382247A (en) * 1965-11-01 1968-05-07 Upjohn Co 6-amino-1, 2-dihydro-1-hydroxy-2-imino-4-phenoxypyrimidines
US3910928A (en) * 1974-04-26 1975-10-07 Upjohn Co 3-(Cyanimino)-propionitriles
AU519993B2 (en) * 1977-02-04 1982-01-07 F. Hoffmann-La Roche & Co. Pyrimidine derivatives
HU177601B (en) * 1978-10-27 1981-11-28 Egyt Gyogyszervegyeszeti Gyar New process for preparing 6-piperidino-2,4-diamino-pyrimidine-3-oxide

Also Published As

Publication number Publication date
JP2726653B2 (ja) 1998-03-11
CA1318914C (fr) 1993-06-08
DE3874842D1 (de) 1992-10-29
EP0304648A1 (fr) 1989-03-01
EP0304648B1 (fr) 1992-09-23
ATE80877T1 (de) 1992-10-15
JPH09216872A (ja) 1997-08-19
JPH0248570A (ja) 1990-02-19
US5126453A (en) 1992-06-30
US4985563A (en) 1991-01-15
JP2647444B2 (ja) 1997-08-27
DE3874842T2 (de) 1993-02-04

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