LU83672A1 - Napsylate de(d-alpha-amino alpha-phenylacetamido)-6 penicillanate de dioxo-1,1 penicillanoyloxymethyle cristallin et ses formes hydratees,leurs procedes de preparation et des medicaments antimicrobiens les contenant comme produits actifs - Google Patents

Napsylate de(d-alpha-amino alpha-phenylacetamido)-6 penicillanate de dioxo-1,1 penicillanoyloxymethyle cristallin et ses formes hydratees,leurs procedes de preparation et des medicaments antimicrobiens les contenant comme produits actifs Download PDF

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Publication number
LU83672A1
LU83672A1 LU83672A LU83672A LU83672A1 LU 83672 A1 LU83672 A1 LU 83672A1 LU 83672 A LU83672 A LU 83672A LU 83672 A LU83672 A LU 83672A LU 83672 A1 LU83672 A1 LU 83672A1
Authority
LU
Luxembourg
Prior art keywords
napsylate
amino
monohydrate
penicillanoyloxymethyl
phenylacetamido
Prior art date
Application number
LU83672A
Other languages
English (en)
French (fr)
Inventor
Wagn O Godtfredsen
Welf Daehne
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of LU83672A1 publication Critical patent/LU83672A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
LU83672A 1980-10-06 1981-10-05 Napsylate de(d-alpha-amino alpha-phenylacetamido)-6 penicillanate de dioxo-1,1 penicillanoyloxymethyle cristallin et ses formes hydratees,leurs procedes de preparation et des medicaments antimicrobiens les contenant comme produits actifs LU83672A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8032147 1980-10-06
GB8032147 1980-10-06

Publications (1)

Publication Number Publication Date
LU83672A1 true LU83672A1 (fr) 1982-05-07

Family

ID=10516500

Family Applications (1)

Application Number Title Priority Date Filing Date
LU83672A LU83672A1 (fr) 1980-10-06 1981-10-05 Napsylate de(d-alpha-amino alpha-phenylacetamido)-6 penicillanate de dioxo-1,1 penicillanoyloxymethyle cristallin et ses formes hydratees,leurs procedes de preparation et des medicaments antimicrobiens les contenant comme produits actifs

Country Status (19)

Country Link
US (1) US4882325A (ja)
JP (1) JPS57131796A (ja)
AT (1) AT373892B (ja)
AU (1) AU547472B2 (ja)
BE (1) BE890649A (ja)
CA (1) CA1178574A (ja)
CH (1) CH648562A5 (ja)
DE (1) DE3139554A1 (ja)
DK (1) DK437481A (ja)
FR (1) FR2491474A1 (ja)
GR (1) GR75774B (ja)
IE (1) IE51516B1 (ja)
IT (1) IT1144892B (ja)
LU (1) LU83672A1 (ja)
NL (1) NL8104527A (ja)
NZ (1) NZ198411A (ja)
PH (1) PH18722A (ja)
SE (1) SE452323B (ja)
ZA (1) ZA816487B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them
US4432987A (en) * 1982-04-23 1984-02-21 Pfizer Inc. Crystalline benzenesulfonate salts of sultamicillin
US5091525A (en) * 1987-10-07 1992-02-25 Eli Lilly And Company Monohydrate and DMF solvates of a new carbacephem antibiotic
CA1324950C (en) * 1988-07-12 1993-12-07 Robert James Joseph Pickford Combating of undesired organisms
MY172561A (en) * 2012-07-17 2019-12-03 Bayer New Zealand Ltd Injectable antibiotic formulations and their methods of use
WO2014014364A1 (en) 2012-07-17 2014-01-23 Bayer New Zealand Limited Injectable antibiotic formulations and their methods of use
BR112015014963B1 (pt) * 2012-12-20 2022-04-12 Alleva Animal Health Limited Formulação de suspensão injetável veterinária

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3180862A (en) * 1962-10-29 1965-04-27 Bristol Myers Co Aryl sulfonic acid salts of alpha-aminobenzylpenicillins
FR1532222A (fr) * 1963-10-28 1968-07-12 Bristol Myers Co Procédé de préparation de dérivés de la pénicilline
GB1241844A (en) * 1968-08-23 1971-08-04 Beecham Group Ltd Penicillins
NZ189945A (en) * 1978-04-01 1981-04-24 Beecham Group Ltd Ampicillin phthalidyl ester naphthalene 2-sulphonate also pharmaceutical compositions
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide

Also Published As

Publication number Publication date
CH648562A5 (de) 1985-03-29
JPH027956B2 (ja) 1990-02-21
ATA416981A (de) 1983-07-15
FR2491474A1 (fr) 1982-04-09
SE8105872L (sv) 1982-04-07
GR75774B (ja) 1984-08-02
CA1178574A (en) 1984-11-27
US4882325A (en) 1989-11-21
AU547472B2 (en) 1985-10-24
DE3139554A1 (de) 1982-07-08
SE452323B (sv) 1987-11-23
IT1144892B (it) 1986-10-29
AU7545281A (en) 1982-04-22
FR2491474B1 (ja) 1984-06-08
IE812145L (en) 1982-04-06
NZ198411A (en) 1985-05-31
NL8104527A (nl) 1982-05-03
JPS57131796A (en) 1982-08-14
IE51516B1 (en) 1987-01-07
AT373892B (de) 1984-02-27
ZA816487B (en) 1983-01-26
DK437481A (da) 1982-04-07
BE890649A (fr) 1982-04-06
DE3139554C2 (ja) 1990-04-26
IT8168281A0 (it) 1981-10-02
PH18722A (en) 1985-09-11

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