LU83327A1 - Procede de preparation de derives de 1,4-thiazine,leur utilisation ainsi que compositions contenant ces derives - Google Patents

Procede de preparation de derives de 1,4-thiazine,leur utilisation ainsi que compositions contenant ces derives Download PDF

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Publication number
LU83327A1
LU83327A1 LU83327A LU83327A LU83327A1 LU 83327 A1 LU83327 A1 LU 83327A1 LU 83327 A LU83327 A LU 83327A LU 83327 A LU83327 A LU 83327A LU 83327 A1 LU83327 A1 LU 83327A1
Authority
LU
Luxembourg
Prior art keywords
group
derivative
formula
thiazane
derivatives
Prior art date
Application number
LU83327A
Other languages
English (en)
French (fr)
Inventor
Claude Gillet
Joseph Roba
Michel Snyers
Georges Lambelin
Original Assignee
Midit
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Midit filed Critical Midit
Priority to LU83327A priority Critical patent/LU83327A1/fr
Priority to JP57501451A priority patent/JPS58500713A/ja
Priority to PCT/BE1982/000009 priority patent/WO1982003860A1/en
Priority to AU83941/82A priority patent/AU8394182A/en
Priority to NL8220153A priority patent/NL8220153A/nl
Priority to GB08235353A priority patent/GB2111056B/en
Priority to PT74813A priority patent/PT74813B/pt
Priority to ES82511759A priority patent/ES8307233A1/es
Priority to KR1019820001874A priority patent/KR830010089A/ko
Priority to ZA822926A priority patent/ZA822926B/xx
Priority to IT20998/82A priority patent/IT1190794B/it
Priority to GR68018A priority patent/GR75996B/el
Priority to BE0/207967A priority patent/BE893025A/fr
Priority to IL65647A priority patent/IL65647A0/xx
Priority to FR8207461A priority patent/FR2509303A1/fr
Priority to DK554382A priority patent/DK554382A/da
Priority to FI771226A priority patent/FI66366C/fi
Priority to SE8207294A priority patent/SE8207294L/xx
Priority to NO824398A priority patent/NO824398L/no
Publication of LU83327A1 publication Critical patent/LU83327A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Facsimiles In General (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
LU83327A 1981-04-29 1981-04-29 Procede de preparation de derives de 1,4-thiazine,leur utilisation ainsi que compositions contenant ces derives LU83327A1 (fr)

Priority Applications (19)

Application Number Priority Date Filing Date Title
LU83327A LU83327A1 (fr) 1981-04-29 1981-04-29 Procede de preparation de derives de 1,4-thiazine,leur utilisation ainsi que compositions contenant ces derives
JP57501451A JPS58500713A (ja) 1981-04-29 1982-04-21 １，４―チアザンカルボン酸誘導体及びその製造方法並びに該誘導体を含有する医薬組成物
PCT/BE1982/000009 WO1982003860A1 (en) 1981-04-29 1982-04-21 Derivatives of 1,4-thiazane-carboxylic acid,preparation and utilization thereof and compositions containing same
AU83941/82A AU8394182A (en) 1981-04-29 1982-04-21 Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same
NL8220153A NL8220153A (nl) 1981-04-29 1982-04-21 1,4-thiazancarbonzuurderivaten, de bereiding en toepassing ervan, alsmede de samenstellingen, die deze derivaten bevatten.
GB08235353A GB2111056B (en) 1981-04-29 1982-04-21 Derivatives of 1, 4-thiazane-carboxylic acid preparation and utilization thereof and compositions containing same
PT74813A PT74813B (fr) 1981-04-29 1982-04-28 Procede de preparation de derives de l'acide 1,4-thiazane-carboxylique
ES82511759A ES8307233A1 (es) 1981-04-29 1982-04-28 Procedimiento para preparar derivados del acido 1,4-tiazan-3-carboxilico.
KR1019820001874A KR830010089A (ko) 1981-04-29 1982-04-29 1,4-티아잔-카르복시산 유도체의 제조방법
ZA822926A ZA822926B (en) 1981-04-29 1982-04-29 1,4-thiazenecarboxylic acid derivatives,their preparation and use and the compositions in which these derivatives are present
IT20998/82A IT1190794B (it) 1981-04-29 1982-04-29 Derivati dell'acido 1,4-tiazancarbossilico,loro preparazione e loro impiego e anche composizioni contenenti questi derivati
GR68018A GR75996B (enrdf_load_stackoverflow) 1981-04-29 1982-04-29
BE0/207967A BE893025A (fr) 1981-04-29 1982-04-29 Derives de l'acide 1,4-thiazane-carboxilique leurs preparation et utilisation ainsi que les compositions contenant ces derives.
IL65647A IL65647A0 (en) 1981-04-29 1982-04-29 Derivatives of 1,4-thiazine-carboxylic acid,preparation thereof,and compositions containing them
FR8207461A FR2509303A1 (fr) 1981-04-29 1982-04-29 Derives de l'acide 1,4-thiazane-carboxylique, leurs preparation et utilisation ainsi que les compositions contenant ces derives
DK554382A DK554382A (da) 1981-04-29 1982-12-14 1,4-tiazankaboxylsyrederivater, deres fremstilling og anvendelse og praeparater hvori disse derivater er til stede
FI771226A FI66366C (fi) 1981-04-29 1982-12-14 Foerfarande foer framstaellning av som laekemedel anvaenda 1,4-tiazin-3-karboxylsyraderivat
SE8207294A SE8207294L (sv) 1981-04-29 1982-12-21 1,4-tiazankarboxylsyraderivat, deras framstellning och anvendning och kompositioner vari dessa derivat ingar
NO824398A NO824398L (no) 1981-04-29 1982-12-28 1,4-tiazankarboksylsyrederivater, fremstilling og bruk av disse og blandinger hvori disse derivater er tilstede

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
LU83327 1981-04-29
LU83327A LU83327A1 (fr) 1981-04-29 1981-04-29 Procede de preparation de derives de 1,4-thiazine,leur utilisation ainsi que compositions contenant ces derives

Publications (1)

Publication Number Publication Date
LU83327A1 true LU83327A1 (fr) 1983-03-24

Family

ID=19729637

Family Applications (1)

Application Number Title Priority Date Filing Date
LU83327A LU83327A1 (fr) 1981-04-29 1981-04-29 Procede de preparation de derives de 1,4-thiazine,leur utilisation ainsi que compositions contenant ces derives

Country Status (16)

Country Link
JP (1) JPS58500713A (enrdf_load_stackoverflow)
KR (1) KR830010089A (enrdf_load_stackoverflow)
BE (1) BE893025A (enrdf_load_stackoverflow)
ES (1) ES8307233A1 (enrdf_load_stackoverflow)
FI (1) FI66366C (enrdf_load_stackoverflow)
FR (1) FR2509303A1 (enrdf_load_stackoverflow)
GB (1) GB2111056B (enrdf_load_stackoverflow)
GR (1) GR75996B (enrdf_load_stackoverflow)
IT (1) IT1190794B (enrdf_load_stackoverflow)
LU (1) LU83327A1 (enrdf_load_stackoverflow)
NL (1) NL8220153A (enrdf_load_stackoverflow)
NO (1) NO824398L (enrdf_load_stackoverflow)
PT (1) PT74813B (enrdf_load_stackoverflow)
SE (1) SE8207294L (enrdf_load_stackoverflow)
WO (1) WO1982003860A1 (enrdf_load_stackoverflow)
ZA (1) ZA822926B (enrdf_load_stackoverflow)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3436386A1 (de) * 1984-10-04 1986-04-10 Merck Patent Gmbh, 6100 Darmstadt (thio)morpholine
FR2618434B1 (fr) * 1987-07-21 1991-02-08 Oreal Esters d'acide thiamorpholinone carboxylique et de ses derives, leur procede de preparation et leur utilisation dans le domaine cosmetique et dermo-pharmaceutique
AU4750990A (en) * 1988-12-14 1990-07-10 Hicks, Richard Method for predicting biological activity of antibiotics, and novel non beta-lactam antibacterial agents derived therefrom
DK2809669T3 (da) 2012-02-03 2017-05-01 Sanofi Sa Kondenserede pyrroldicarboxamider og deres anvendelse som farmaceutika

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2187327B1 (enrdf_load_stackoverflow) * 1972-06-15 1975-06-20 Rech Pharm Scientifiques
US4179276A (en) * 1977-02-01 1979-12-18 E. I. Du Pont De Nemours And Company Novel imidazothiazine-1,3 (2H)-diones
JPS5540658A (en) * 1978-09-19 1980-03-22 Tanabe Seiyaku Co Ltd 1,4-thiazan-3-carboxylic ester derivative and its preparation

Also Published As

Publication number Publication date
ES511759A0 (es) 1983-07-01
GB2111056B (en) 1985-03-06
GR75996B (enrdf_load_stackoverflow) 1984-08-03
PT74813B (fr) 1983-10-26
SE8207294D0 (sv) 1982-12-21
KR830010089A (ko) 1983-12-26
IT1190794B (it) 1988-02-24
ES8307233A1 (es) 1983-07-01
JPH0330592B2 (enrdf_load_stackoverflow) 1991-04-30
IT8220998A0 (it) 1982-04-29
NO824398L (no) 1982-12-28
FI66366C (fi) 1984-10-10
FI66366B (fi) 1984-06-29
FR2509303A1 (fr) 1983-01-14
NL8220153A (nl) 1983-03-01
FI824279L (fi) 1982-12-14
JPS58500713A (ja) 1983-05-06
PT74813A (fr) 1982-05-01
SE8207294L (sv) 1982-12-21
GB2111056A (en) 1983-06-29
BE893025A (fr) 1982-10-29
WO1982003860A1 (en) 1982-11-11
ZA822926B (en) 1983-03-30
FI824279A0 (fi) 1982-12-14

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