LT3643707T - 18f žymėtas junginys, skirtas prostatos vėžio diagnostikai ir jo panaudojimas - Google Patents

18f žymėtas junginys, skirtas prostatos vėžio diagnostikai ir jo panaudojimas

Info

Publication number
LT3643707T
LT3643707T LTEPPCT/KR2018/006869T LT18820848T LT3643707T LT 3643707 T LT3643707 T LT 3643707T LT 18820848 T LT18820848 T LT 18820848T LT 3643707 T LT3643707 T LT 3643707T
Authority
LT
Lithuania
Prior art keywords
diagnosis
prostate cancer
labeled compound
labeled
compound
Prior art date
Application number
LTEPPCT/KR2018/006869T
Other languages
English (en)
Lithuanian (lt)
Inventor
Dae Yoon Chi
Byoung Se Lee
So Young Chu
Min Hwan Kim
Woon Jung Jung
Hyeon Jin Jeong
Kyo Chul Lee
Yong Jin Lee
Ji Ae Park
Mi Hyun Kim
Ran Ji Yoo
Sang Moo Lim
Original Assignee
Futurechem Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Futurechem Co., Ltd. filed Critical Futurechem Co., Ltd.
Priority claimed from PCT/KR2018/006869 external-priority patent/WO2018236115A1/ko
Publication of LT3643707T publication Critical patent/LT3643707T/lt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/0402Organic compounds carboxylic acid carriers, fatty acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K49/00Preparations for testing in vivo
    • A61K49/06Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
    • A61K49/08Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
    • A61K49/085Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier conjugated systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K49/00Preparations for testing in vivo
    • A61K49/06Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
    • A61K49/08Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
    • A61K49/10Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0453Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/0474Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/0497Organic compounds conjugates with a carrier being an organic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Optics & Photonics (AREA)
  • Physics & Mathematics (AREA)
  • Radiology & Medical Imaging (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nuclear Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Magnetic Resonance Imaging Apparatus (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
LTEPPCT/KR2018/006869T 2017-06-19 2018-06-18 18f žymėtas junginys, skirtas prostatos vėžio diagnostikai ir jo panaudojimas LT3643707T (lt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR20170077570 2017-06-19
PCT/KR2018/006869 WO2018236115A1 (ko) 2017-06-19 2018-06-18 전립선암 진단을 위한 18f-표지된 화합물 및 그의 용도

Publications (1)

Publication Number Publication Date
LT3643707T true LT3643707T (lt) 2022-05-25

Family

ID=65008286

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEPPCT/KR2018/006869T LT3643707T (lt) 2017-06-19 2018-06-18 18f žymėtas junginys, skirtas prostatos vėžio diagnostikai ir jo panaudojimas

Country Status (21)

Country Link
US (1) US10870629B2 (https=)
EP (1) EP3643707B1 (https=)
JP (1) JP6913968B2 (https=)
KR (1) KR102015355B1 (https=)
CN (1) CN110770212B (https=)
AU (1) AU2018288907B2 (https=)
CA (1) CA3067696C (https=)
CL (1) CL2019003727A1 (https=)
DK (1) DK3643707T3 (https=)
EA (1) EA037781B1 (https=)
ES (1) ES2912392T3 (https=)
HR (1) HRP20220557T1 (https=)
LT (1) LT3643707T (https=)
MX (1) MX388833B (https=)
MY (1) MY195426A (https=)
PH (1) PH12019502665A1 (https=)
PL (1) PL3643707T3 (https=)
PT (1) PT3643707T (https=)
RS (1) RS63205B1 (https=)
SG (1) SG11201911602RA (https=)
SI (1) SI3643707T1 (https=)

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2494096C2 (ru) 2008-08-01 2013-09-27 Дзе Джонс Хопкинс Юниверсити Агенты, связывающиеся с psma, и их применение
WO2013022797A1 (en) * 2011-08-05 2013-02-14 Molecular Insight Pharmaceuticals Radiolabeled prostate specific membrane antigen inhibitors
WO2013028664A1 (en) 2011-08-22 2013-02-28 Siemens Medical Solutions Usa, Inc. Psma imaging agents
JP2014051442A (ja) * 2012-09-05 2014-03-20 Kyoto Univ 前立腺がんを診断可能な核医学イメージングプローブ
EP3300746B1 (en) * 2013-01-14 2019-05-15 Molecular Insight Pharmaceuticals, Inc. Triazine based radiopharmaceuticals and radioimaging agents
ES3005832T3 (en) 2013-11-13 2025-03-17 Ge Healthcare Ltd Dual run cassette for the synthesis of 18f-labelled compounds
KR20150113801A (ko) * 2014-03-31 2015-10-08 한미약품 주식회사 Tak1 저해 활성을 갖는 피라진 접합고리 유도체
FR3023290B1 (fr) * 2014-07-04 2016-08-19 Pf Medicament Derives de flavaglines
WO2017027870A1 (en) * 2015-08-13 2017-02-16 The Johns Hopkins University Triazole conjugated ureas, thioureas, carbamates, and "reversed" carbamates for psma-targeted imaging agents and uses thereof
EP3493856B1 (en) 2016-06-28 2023-08-09 Cornell University 18f-labeled triazole containing psma inhibitors

Also Published As

Publication number Publication date
CN110770212B (zh) 2022-11-22
DK3643707T3 (da) 2022-05-09
JP2020524175A (ja) 2020-08-13
EP3643707A4 (en) 2021-06-09
RS63205B1 (sr) 2022-06-30
US10870629B2 (en) 2020-12-22
PT3643707T (pt) 2022-05-04
CA3067696A1 (en) 2018-12-27
EA202090071A1 (ru) 2020-04-16
AU2018288907B2 (en) 2020-05-07
AU2018288907A1 (en) 2020-01-23
SI3643707T1 (sl) 2022-06-30
CA3067696C (en) 2022-05-03
HRP20220557T1 (hr) 2022-06-10
KR102015355B1 (ko) 2019-10-23
CL2019003727A1 (es) 2020-07-03
EP3643707B1 (en) 2022-02-23
US20200207724A1 (en) 2020-07-02
CN110770212A (zh) 2020-02-07
SG11201911602RA (en) 2020-01-30
KR20180138169A (ko) 2018-12-28
MY195426A (en) 2023-01-20
EA037781B1 (ru) 2021-05-20
MX388833B (es) 2025-03-12
PH12019502665A1 (en) 2020-10-26
ES2912392T3 (es) 2022-05-25
BR112019027183A2 (pt) 2020-06-30
PL3643707T3 (pl) 2023-06-12
EP3643707A1 (en) 2020-04-29
JP6913968B2 (ja) 2021-08-04
MX2019015616A (es) 2020-02-26

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